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Volumn 2, Issue 3, 2006, Pages 559-571

Characterization of human and rodent native and recombinant adenosine A2B receptors by radioligand binding studies

Author keywords

3H PSB 298; A2B antagonist radioligand; Adenosine A2B receptor; CHO cells; HEK 293 cells; INS 1 cells; NG108 15 cells; Sodium shift assays

Indexed keywords


EID: 33748543969     PISSN: 15739538     EISSN: 15739546     Source Type: Journal    
DOI: 10.1007/s11302-006-9012-4     Document Type: Article
Times cited : (24)

References (40)
  • 2
    • 30444441037 scopus 로고    scopus 로고
    • 2B receptor as a novel therapeutic target in asthma
    • 2B receptor as a novel therapeutic target in asthma. Br J Pharmacol 145:1009-1015
    • (2005) Br J Pharmacol , vol.145 , pp. 1009-1015
    • Holgate, S.T.1
  • 7
    • 0032836645 scopus 로고    scopus 로고
    • q in human embryonic kidney 293 cells and HMC-1 mast cells
    • q in human embryonic kidney 293 cells and HMC-1 mast cells. Mol Pharmacol 56:705-713
    • (1999) Mol Pharmacol , vol.56 , pp. 705-713
    • Linden, J.1    Thai, T.2    Figler, H.3
  • 8
    • 0030428077 scopus 로고    scopus 로고
    • Molecular characterization of recombinant human adenosine receptors
    • Robeva AS, Woodard R, Jin X et al (1996) Molecular characterization of recombinant human adenosine receptors. Drug Dev Res 39:243-252
    • (1996) Drug Dev Res , vol.39 , pp. 243-252
    • Robeva, A.S.1    Woodard, R.2    Jin, X.3
  • 12
    • 21744443649 scopus 로고    scopus 로고
    • 2B receptors in a recombinant system and in peripheral blood cells using a novel selective antagonist radioligand, [3H]MRE 2029-F20
    • 2B receptors in a recombinant system and in peripheral blood cells using a novel selective antagonist radioligand, [3H]MRE 2029-F20. Mol Pharmacol 67:2137-2147
    • (2005) Mol Pharmacol , vol.67 , pp. 2137-2147
    • Gessi, S.1    Varani, K.2    Merighi, S.3
  • 17
    • 0025939740 scopus 로고
    • Synthesis of 3-substituted 6-aminouracils
    • Müller CE (1991) Synthesis of 3-substituted 6-aminouracils. Tetrahedron Lett 32:6539-6540
    • (1991) Tetrahedron Lett , vol.32 , pp. 6539-6540
    • Müller, C.E.1
  • 18
    • 0031931065 scopus 로고    scopus 로고
    • Comparative pharmacology of human adenosine receptor subtypes - Characterization of stable transfected receptors in CHO cells
    • Klotz KN, Hessling J, Hegler J et al (1998) Comparative pharmacology of human adenosine receptor subtypes - characterization of stable transfected receptors in CHO cells. Naunyn Schmiedebergs Arch Pharmacol 357:1-9
    • (1998) Naunyn Schmiedebergs Arch Pharmacol , vol.357 , pp. 1-9
    • Klotz, K.N.1    Hessling, J.2    Hegler, J.3
  • 19
    • 0038390356 scopus 로고    scopus 로고
    • Extracellular metabolism of nucleotides in neuroblastoma x glioma NG108-15 cells determined by capillary electrophoresis
    • Kaulich M, Qurishi R, Müller CE (2003) Extracellular metabolism of nucleotides in neuroblastoma x glioma NG108-15 cells determined by capillary electrophoresis. Cell Mol Neurobiol 23:349-364
    • (2003) Cell Mol Neurobiol , vol.23 , pp. 349-364
    • Kaulich, M.1    Qurishi, R.2    Müller, C.E.3
  • 21
    • 71849104860 scopus 로고
    • Protein measurements with the Folin phenol reagent
    • Lowry OH, Rosebrough NJ, Farr AL et al (1951) Protein measurements with the Folin phenol reagent. J Biol Chem 193:265-275
    • (1951) J Biol Chem , vol.193 , pp. 265-275
    • Lowry, O.H.1    Rosebrough, N.J.2    Farr, A.L.3
  • 22
    • 0036033424 scopus 로고    scopus 로고
    • Constitutive activity of G protein-coupled receptors: Cause of disease and common property of wild-type receptors
    • Seifert R, Wenzel-Seifert K (2002) Constitutive activity of G protein-coupled receptors: Cause of disease and common property of wild-type receptors. Naunyn Schmiedebergs Arch Pharmacol 366:381-416
    • (2002) Naunyn Schmiedebergs Arch Pharmacol , vol.366 , pp. 381-416
    • Seifert, R.1    Wenzel-Seifert, K.2
  • 23
    • 0034016295 scopus 로고    scopus 로고
    • Inverse agonism at G protein-coupled receptors: (patho)Physiological relevance and implications for drug discovery
    • de Ligt RA, Kourounakis AP, IJzerman AP (2000) Inverse agonism at G protein-coupled receptors: (patho)physiological relevance and implications for drug discovery. Br J Pharmacol 130:1-12
    • (2000) Br J Pharmacol , vol.130 , pp. 1-12
    • de Ligt, R.A.1    Kourounakis, A.P.2    IJzerman, A.P.3
  • 24
    • 0037161610 scopus 로고    scopus 로고
    • 2B adenosine receptors of xanthine derivatives substituted at the 1-,3-,7-, and 8-positions
    • 2B adenosine receptors of xanthine derivatives substituted at the 1-,3-,7-, and 8-positions. J Med Chem 45:2131-2138
    • (2002) J Med Chem , vol.45 , pp. 2131-2138
    • Kim, S.A.1    Marshall, M.A.2    Melman, N.3
  • 25
    • 0020603182 scopus 로고
    • Influence of sodium on the alpha 2-adrenergic receptor system of human platelets. Role for intraplatelet sodium in receptor binding
    • Motulsky R, Insel PA (1983) Influence of sodium on the alpha 2-adrenergic receptor system of human platelets. Role for intraplatelet sodium in receptor binding. J Biol Chem 258:3913-3919
    • (1983) J Biol Chem , vol.258 , pp. 3913-3919
    • Motulsky, R.1    Insel, P.A.2
  • 26
    • 0038026057 scopus 로고    scopus 로고
    • Allosteric activation of plasma membrane receptors - Physiological implications and structural origins
    • Conigrave AD, Franks AH (2003) Allosteric activation of plasma membrane receptors - physiological implications and structural origins. Prog Biophys Mol Biol 81:219-240
    • (2003) Prog Biophys Mol Biol , vol.81 , pp. 219-240
    • Conigrave, A.D.1    Franks, A.H.2
  • 27
    • 0018138234 scopus 로고
    • Agonist-specific effects of monovalent and divalent cations on adenylate cyclase-coupled α-adrenergic receptors in rabbit platelets
    • Tsai BS, Lefkowitz RJ (1978) Agonist-specific effects of monovalent and divalent cations on adenylate cyclase-coupled α-adrenergic receptors in rabbit platelets. Mol Pharmacol 14:540-548
    • (1978) Mol Pharmacol , vol.14 , pp. 540-548
    • Tsai, B.S.1    Lefkowitz, R.J.2
  • 28
    • 0030460366 scopus 로고    scopus 로고
    • 1 adenosine receptor: Influences of acidic and hydroxy residues in the first four transmembrane domains on ligand binding
    • 1 adenosine receptor: Influences of acidic and hydroxy residues in the first four transmembrane domains on ligand binding. Mol Pharmacol 50:1635-1642
    • (1996) Mol Pharmacol , vol.50 , pp. 1635-1642
    • Barbhaiya, H.1    McClain, R.2    IJzerman, A.P.3
  • 29
    • 0034284626 scopus 로고    scopus 로고
    • 2A adenosine receptors by amiloride analogues and sodium ions
    • 2A adenosine receptors by amiloride analogues and sodium ions. Biochem Pharmacol 60:669-676
    • (2000) Biochem Pharmacol , vol.60 , pp. 669-676
    • Gao, Z.G.1    IJzerman, A.P.2
  • 30
    • 0035895353 scopus 로고    scopus 로고
    • Salt dependence of the formation and stability state in G protein-coupled receptors: Evidence for the involvement of the Hofmeister effect
    • Vogel R, Fan GB, Sheves M et al (2001) Salt dependence of the formation and stability state in G protein-coupled receptors: Evidence for the involvement of the Hofmeister effect. Biochemistry 40:483-493
    • (2001) Biochemistry , vol.40 , pp. 483-493
    • Vogel, R.1    Fan, G.B.2    Sheves, M.3
  • 32
    • 0028972629 scopus 로고
    • 1 adenosine receptor/G protein coupling: Identification of a membrane protein complex
    • 1 adenosine receptor/G protein coupling: Identification of a membrane protein complex. Mol Pharmacol 48:806-817
    • (1995) Mol Pharmacol , vol.48 , pp. 806-817
    • Nanoff, C.1    Mitterauer, T.2    Roka, F.3
  • 34
    • 0017623546 scopus 로고
    • Structural, electrophysical, biochemical and pharmacological properties of neuroblastoma-glioma cell hybrids in cell culture
    • Hamprecht B (1977) Structural, electrophysical, biochemical and pharmacological properties of neuroblastoma-glioma cell hybrids in cell culture. Int Rev Cytol 49:99-170
    • (1977) Int Rev Cytol , vol.49 , pp. 99-170
    • Hamprecht, B.1
  • 35
    • 0034021926 scopus 로고    scopus 로고
    • Effects of AMP derivatives on cyclic AMP levels in NG108-15 cells
    • Ohkubo S, Nakanishi H, Kimura J et al (2000) Effects of AMP derivatives on cyclic AMP levels in NG108-15 cells. Br J Pharmacol 129:1244-1250
    • (2000) Br J Pharmacol , vol.129 , pp. 1244-1250
    • Ohkubo, S.1    Nakanishi, H.2    Kimura, J.3
  • 38
    • 33748580504 scopus 로고    scopus 로고
    • Control of blood glucose by insulin and adenosine receptor antagonists
    • In: Abstract no. 226 of the Gold Coast, Australia
    • LaNoue KF et al (2002) Control of blood glucose by insulin and adenosine receptor antagonists. In: Abstract no. 226 of the 7th international symposium on adenosine and adenine nucleotides, Gold Coast, Australia
    • (2002) 7th International Symposium on Adenosine and Adenine Nucleotides
    • LaNoue, K.F.1
  • 39
    • 0035653641 scopus 로고    scopus 로고
    • Adenosine receptor antagonists and retinal neovascularization in vivo
    • Mino RP, Spoerri PE, Caballero S et al (2001) Adenosine receptor antagonists and retinal neovascularization in vivo. Investig Ophthalmol Vis Sci 42:332-334
    • (2001) Investig Ophthalmol Vis Sci , vol.42 , pp. 332-334
    • Mino, R.P.1    Spoerri, P.E.2    Caballero, S.3
  • 40
    • 0025603686 scopus 로고    scopus 로고
    • 1 receptor binding and function using 2-amino-3-benzoylthiophenes
    • 1 receptor binding and function using 2-amino-3-benzoylthiophenes. Mol Pharmacol 38:939-949
    • (1996) Mol Pharmacol , vol.38 , pp. 939-949
    • Bruns, R.F.1    Fergus, J.H.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.