Use of the triazolotriazine [3H]ZM 241385 as a radioligand at recombinant human A(2B) adenosine receptors

Drug Design and Discovery

Volumn 16, Issue 3, 1999, Pages 217-226

  Ji, Xiao Duo ^a   Jacobson, Kenneth A ^a  

^a NATIONAL INSTITUTES OF HEALTH   (United States)

Author keywords

Adenosine analogues; G protein coupled receptors; Purines; Radioligand binding; Xanthines

Indexed keywords

4 [2 [7 AMINO 2 (2 FURYL) 1,2,4 TRIAZOLO[2,3 A][1,3,5]TRIAZIN 5 YLAMINO]ETHYL]PHENOL; 8 [4 (2 AMINOETHYLCARBAMOYL)METHOXYPHENYL] 1,3 DIPROPYLXANTHINE; 8 CYCLOPENTYL 1,3 DIPROPYLXANTHINE; 9 CHLORO 2 (2 FURYL) 5,6 DIHYDRO 5 IMINO 1,2,4 TRIAZOLO[2,3 C]QUINAZOLINE; ADENOSINE 5' (N ETHYLCARBOXAMIDE); ADENOSINE A2B RECEPTOR; ADENOSINE DERIVATIVE; FLAVINE MONONUCLEOTIDE; RADIOLIGAND; RECEPTOR SUBTYPE; RECOMBINANT RECEPTOR; TRITIUM; XANTHINE DERIVATIVE; ADENOSINE RECEPTOR; RECOMBINANT PROTEIN; TRIAZINE DERIVATIVE; TRIAZOLE DERIVATIVE;

ARTICLE; HUMAN; HUMAN CELL; MOLECULAR MODEL; RECEPTOR AFFINITY; RECEPTOR BINDING; ANIMAL; CELL LINE; CHO CELL; DRUG ANTAGONISM; DRUG POTENTIATION; HAMSTER; METABOLISM; RADIOASSAY;

ANIMALS; CELL LINE; CHO CELLS; CRICETINAE; HUMANS; RADIOLIGAND ASSAY; RECEPTOR, ADENOSINE A2B; RECEPTORS, PURINERGIC P1; RECOMBINANT PROTEINS; TRIAZINES; TRIAZOLES; TRITIUM;

EID: 0032585940     PISSN: 10559612     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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