[3H]8-Ethyl-4-methyl-2-phenyl-(8R)-4,5,7,8-tetrahydro-1H-imidazo [2,1-i]-purin-5-one ([3H]PSB-11), a Novel High-Affinity Antagonist Radioligand for Human A3 Adenosine Receptors

Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 3, 2002, Pages 501-503

  Müller, Christa E ^a   Diekmann, Martina ^a   Thorand, Mark ^a   Ozola, Vita ^a  

^a UNIVERSITY OF BONN   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

2 [4 (2 CARBOXYETHYL)PHENETHYLAMINO]ADENOSINE 5' (N ETHYLCARBOXAMIDE); 2 CHLOROADENOSINE; 3,7 DIMETHYL 1 PROPARGYLXANTHINE; 6 N CYCLOPENTYLADENOSINE; 8 CYCLOPENTYL 1,3 DIPROPYLXANTHINE; 8 ETHYL 4 METHYL 2 PHENYL 4,5,7,8 TETRAHYDRO 1H IMIDAZO[2,1 I]PURIN 5 ONE H 3; ADENOSINE 5' (N ETHYLCARBOXAMIDE); ADENOSINE A3 RECEPTOR; CAFFEINE; KETONE DERIVATIVE; PHENYLISOPROPYLADENOSINE; RADIOLIGAND; RECEPTOR SUBTYPE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING SITE; CHO CELL; CONTROLLED STUDY; DRUG BINDING; DRUG EFFECT; DRUG SYNTHESIS; HYDROGENATION; NONHUMAN; PATHOPHYSIOLOGY; RECEPTOR AFFINITY;

ANIMALS; CATALYSIS; CHO CELLS; CRICETINAE; HUMANS; HYDROGENATION; IMIDAZOLES; KINETICS; MEMBRANES; PURINES; RADIOPHARMACEUTICALS; RECEPTOR, ADENOSINE A3; RECEPTORS, PURINERGIC P1;

CRICETINAE; CRICETULUS GRISEUS;

EID: 0037059931     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(01)00785-5     Document Type: Article

References (11)