Bisubstrate analogue structure-activity relationships for p300 histone acetyltransferase inhibitors

Bioorganic and Medicinal Chemistry

Volumn 12, Issue 12, 2004, Pages 3383-3390

  Sagar, Vatsala ^a   Zheng, Weiping ^a   Thompson, Paul R ^a   Cole, Philip A ^a  

^a JOHNS HOPKINS UNIVERSITY SCHOOL OF MEDICINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ACYLTRANSFERASE INHIBITOR; ANTINEOPLASTIC AGENT; COENZYME A; HISTONE ACETYLTRANSFERASE; LYSINE DERIVATIVE; PROTEIN P300;

ARTICLE; DRUG STRUCTURE; DRUG TARGETING; GENE EXPRESSION; STRUCTURE ACTIVITY RELATION;

ACETYLTRANSFERASES; CELL CYCLE PROTEINS; COENZYME A; ENZYME INHIBITORS; HISTONE ACETYLTRANSFERASES; LYSINE; MOLECULAR STRUCTURE; STRUCTURE-ACTIVITY RELATIONSHIP; TRANSCRIPTION FACTORS;

EID: 2542421889     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2004.03.070     Document Type: Article

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