Structure of the GCN5 histone acetyltransferase bound to a bisubstrate inhibitor

Proceedings of the National Academy of Sciences of the United States of America

Volumn 99, Issue 22, 2002, Pages 14065-14070

  Poux, Arienne N ^a   Cebrat, Marek ^b,c   Kim, Cheol M ^b,d   Cole, Philip A ^b   Marmorstein, Ronen ^a  

^a UNIVERSITY OF PENNSYLVANIA   (United States)

^b JOHNS HOPKINS UNIVERSITY   (United States)

^c UNIVERSITY OF WROC AW   (Poland)

^d LG Chemical Ltd   (South Korea)

Author keywords

[No Author keywords available]

Indexed keywords

ACETYL COENZYME A; COENZYME A; CYCLIC AMP RESPONSIVE ELEMENT BINDING PROTEIN BINDING PROTEIN; ENZYME INHIBITOR; HISTONE; HISTONE ACETYLTRANSFERASE; HISTONE ACETYLTRANSFERASE GCN5; LYSINE; PROTEIN P53; TRANSCRIPTION FACTOR; UNCLASSIFIED DRUG;

ACETYLATION; ARTICLE; CARBOXY TERMINAL SEQUENCE; CATALYSIS; ENZYME STRUCTURE; ENZYME SUBSTRATE COMPLEX; GENE ACTIVATION; GENE REARRANGEMENT; PRIORITY JOURNAL; PROTEIN DOMAIN;

ACETYLTRANSFERASES; ANIMALS; CATALYSIS; CELL CYCLE PROTEINS; COENZYME A; DRUG DESIGN; ENZYME INHIBITORS; HISTONE ACETYLTRANSFERASES; HUMANS; MODELS, MOLECULAR; PEPTIDES; PROTEIN STRUCTURE, TERTIARY; PROTOZOAN PROTEINS; SACCHAROMYCES CEREVISIAE PROTEINS; SUBSTRATE SPECIFICITY; TETRAHYMENINA; TRANS-ACTIVATORS; TRANSCRIPTION FACTORS;

EID: 0037195124     PISSN: 00278424     EISSN: None     Source Type: Journal    
DOI: 10.1073/pnas.222373899     Document Type: Article

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