125I-Tyr(o)-sauvagine: A novel high affinity radioligand for the pharmacological and biochemical study of human corticotropin-releasing factor(2α) receptors

Molecular Pharmacology

Volumn 50, Issue 3, 1996, Pages 679-686

  Grigoriadis, Dimitri E ^a   Liu, Xin Jun ^a   Vaughn, Joan ^b   Palmer, Scott F ^c   True, C Diane ^c   Vale, Wylie W ^b   Ling, Nicholas ^a   De Souza, Errol B ^a  

^a NEUROCRINE BIOSCIENCES INC   (United States)

^b SALK INSTITUTE FOR BIOLOGICAL STUDIES   (United States)

^c DUPONT COMPANY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CORTICOTROPIN; CORTICOTROPIN RELEASING FACTOR RECEPTOR; RECEPTOR SUBTYPE; CORTICOTROPIN RELEASING FACTOR; CRF(2ALPHA) RECEPTOR; CYCLIC AMP; DRUG DERIVATIVE; GUANINE NUCLEOTIDE; PEPTIDE; PEPTIDE FRAGMENT; RADIOACTIVE IODINE; RECOMBINANT PROTEIN; SAUVAGINE, TYR(0); SAUVAGINE, TYR(0)-;

ANIMAL CELL; ARTICLE; DRUG POTENCY; DRUG RECEPTOR BINDING; HUMAN; ISOTOPE LABELING; LIGAND BINDING; NONHUMAN; PRIORITY JOURNAL; RECEPTOR AFFINITY; ANIMAL; BINDING COMPETITION; CELL MEMBRANE; CHO CELL; DRUG EFFECT; GENETIC TRANSFECTION; HAMSTER; KINETICS; METABOLISM; PHYSIOLOGY; RADIOASSAY; SYNTHESIS;

ANIMALS; BINDING, COMPETITIVE; CELL MEMBRANE; CHO CELLS; CORTICOTROPIN-RELEASING HORMONE; CRICETINAE; CYCLIC AMP; GUANINE NUCLEOTIDES; HUMANS; IODINE RADIOISOTOPES; KINETICS; PEPTIDE FRAGMENTS; PEPTIDES; RADIOLIGAND ASSAY; RECEPTORS, CORTICOTROPIN-RELEASING HORMONE; RECOMBINANT PROTEINS; TRANSFECTION;

EID: 0029665585     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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