Reversible and irreversible small molecule inhibitors of monoamine oxidase B (MAO-B) investigated by biophysical techniques

Bioorganic and Medicinal Chemistry

Volumn 23, Issue 4, 2015, Pages 770-778

  Rojas, Rafael J ^a   Edmondson, Dale E ^b   Almos, Terri ^a   Scott, Roderick ^a   Massari, Mark E ^a  

^a DART NEUROSCIENCE LLC   (United States)

^b EMORY UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

LAZABEMIDE; MONOAMINE OXIDASE B INHIBITOR; N (2 AMINOETHYL) 4 CHLOROBENZAMIDE; PARGYLINE; PIOGLITAZONE; RASAGILINE; SAFINAMIDE; SELEGILINE;

ANALYTIC METHOD; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG STRUCTURE; ENTHALPY; ISOTHERMAL TITRATION CALORIMETRY; MELTING POINT; NONHUMAN; PHYSICAL CHEMISTRY; PROCESS DEVELOPMENT; THERMAL ANALYSIS; THERMAL SHIFT; THERMODYNAMICS; THERMOSTABILITY;

EID: 84964203185     PISSN: 09680896     EISSN: 14643391     Source Type: Journal    
DOI: 10.1016/j.bmc.2014.12.063     Document Type: Article

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