New selective inhibitors of calcium-activated chloride channels - T16Ainh-A01, CaCCinh-A01 and MONNA - What do they inhibit?

British Journal of Pharmacology

Volumn 172, Issue 16, 2015, Pages 4158-4171

  Boedtkjer, D M B ^a,b   Kim, S ^a   Jensen, A B ^a   Matchkov, V M ^a   Andersson, K E ^a,b  

^a AARHUS UNIVERSITY   (Denmark)

^b AARHUS UNIVERSITY HOSPITAL   (Denmark)

Author keywords

[No Author keywords available]

Indexed keywords

15 HYDROXY 11ALPHA,9ALPHA EPOXYMETHANOPROSTA 5,13 DIENOIC ACID; 2 [(5 ETHYL 1,6 DIHYDRO 4 METHYL 6 OXO 2 PYRIMIDINYL)THIO] N [4 (4 METHOXYPHENYL) 2 THIAZOLYL]ACETAMIDE; 6 (1,1 DIMETHYLETHYL) 2 [(2 FURANYL CARBONYL)AMINO] 4,5,6,7 TETRAHYDROBENZO[B]THIOPHENE 3 CARBOXYLIC ACID; ANOCTAMIN 1 PROTEIN; BARIUM; CALCIUM ACTIVATED CHLORIDE CHANNEL; CHLORIDE; CHLORIDE CHANNEL BLOCKING AGENT; N [(4 METHOXY) 2 NAPHTHYL] 5 NITROANTHRANILIC ACID; NORADRENALIN; POTASSIUM; TMEM16A; UNCLASSIFIED DRUG; 6-T-BUTYL-2-(FURAN-2-CARBOXAMIDO)-4,5,6,7-TETRAHYDROBENZO(B)THIOPHENE-3-CARBOXYLIC ACID; ANTHRANILIC ACID DERIVATIVE; CHLORIDE CHANNEL; N-((4-METHOXY)-2-NAPHTHYL)-5-NITROANTHRANILIC ACID; PYRIMIDINE DERIVATIVE; T16AINH-A01; THIAZOLE DERIVATIVE; THIOPHENE DERIVATIVE; VASODILATOR AGENT;

A7R5 CELL LINE; ADULT; ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTERY RESISTANCE; ARTICLE; CALCIUM CELL LEVEL; CALCIUM CURRENT; CELL LINE; CELL MEMBRANE DEPOLARIZATION; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG EFFICACY; DRUG INHIBITION; DRUG MECHANISM; DRUG SELECTIVITY; ELECTROPHYSIOLOGY; EMBRYO; FEMALE; INHIBITION KINETICS; MALE; MEMBRANE POTENTIAL; MOUSE; NONHUMAN; PRIORITY JOURNAL; RAT; VASOCONSTRICTION; VASODILATATION; VOLTAGE CLAMP TECHNIQUE; VOLTAGE DEPENDENT CALCIUM CURRENT; ANIMAL; ANTAGONISTS AND INHIBITORS; BRAIN ARTERY; C57BL MOUSE; DRUG EFFECTS; IN VITRO STUDY; MESENTERIC ARTERY; PHYSIOLOGY; WISTAR RAT;

ANIMALS; CELL LINE; CEREBRAL ARTERIES; CHLORIDE CHANNELS; FEMALE; IN VITRO TECHNIQUES; MALE; MESENTERIC ARTERIES; MICE, INBRED C57BL; ORTHO-AMINOBENZOATES; PYRIMIDINES; RATS, WISTAR; THIAZOLES; THIOPHENES; VASODILATOR AGENTS;

EID: 84937512484     PISSN: 00071188     EISSN: 14765381     Source Type: Journal    
DOI: 10.1111/bph.13201     Document Type: Article

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