Biological redundancy of endogenous GPCR ligands in the gut and the potential for endogenous functional selectivity

Frontiers in Pharmacology

Volumn 5, Issue NOV, 2014, Pages 1-24

  Thompson, Georgina L ^a   Canals, Meritxell ^a   Poole, Daniel P ^a,b  

^a MONASH UNIVERSITY   (Australia)

^b UNIVERSITY OF MELBOURNE   (Australia)

Author keywords

Biased agonism; Enteric nervous system; G protein coupled receptor; Opioid; Opioid receptor; Somatostatin; Somatostatin receptor

Indexed keywords

CORTISTATIN; DELTA OPIATE RECEPTOR; DYNORPHIN; ENDORPHIN; ENKEPHALIN; G PROTEIN COUPLED RECEPTOR; KAPPA OPIATE RECEPTOR; MU OPIATE RECEPTOR; NOCICEPTIN RECEPTOR; OPIATE; PROOPIOMELANOCORTIN; SOMATOSTATIN; SOMATOSTATIN RECEPTOR 1; SOMATOSTATIN RECEPTOR 2; SOMATOSTATIN RECEPTOR 3; SOMATOSTATIN RECEPTOR 4; SOMATOSTATIN RECEPTOR 5;

AMINO ACID SEQUENCE; AMINO TERMINAL SEQUENCE; ARTICLE; GASTROINTESTINAL TRACT; INTESTINE; NONHUMAN; PROTEIN ANALYSIS; PROTEIN CLEAVAGE; PROTEIN DEGRADATION; PROTEIN EXPRESSION; PROTEIN FUNCTION; PROTEIN LOCALIZATION; PROTEIN PROCESSING; PROTEIN SECRETION; PROTEIN SYNTHESIS; PROTEIN TARGETING; SIGNAL TRANSDUCTION;

EID: 84910653530     PISSN: None     EISSN: 16639812     Source Type: Journal    
DOI: 10.3389/fphar.2014.00262     Document Type: Article

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