Pharmacological characterization of GABAB receptor subtypes assembled with auxiliary KCTD subunits

Neuropharmacology

Volumn 88, Issue , 2015, Pages 145-154

  Rajalu, Mathieu ^a   Fritzius, Thorsten ^a   Adelfinger, Lisa ^a   Jacquier, Valerie ^a   Besseyrias, Valerie ^a   Gassmann, Martin ^a   Bettler, Bernhard ^a  

^a UNIVERSITY OF BASEL   (Switzerland)

Author keywords

Baclofen; G protein coupled receptor; GABA B; GS93783; KCTD; Kir3

Indexed keywords

4 AMINOBUTYRIC ACID; 4 AMINOBUTYRIC ACID B RECEPTOR; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANINE NUCLEOTIDE BINDING PROTEIN BETA SUBUNIT; GUANINE NUCLEOTIDE BINDING PROTEIN GAMMA SUBUNIT; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); INWARDLY RECTIFYING POTASSIUM CHANNEL; INWARDLY RECTIFYING POTASSIUM CHANNEL SUBUNIT KIR3; MEMBRANE PROTEIN; N,N' DICYCLOPENTYL 2 METHYLTHIO 5 NITRO 4,6 PYRIMIDINEDIAMINE; POTASSIUM CHANNEL TETRAMERIZATION DOMAIN 16 SUBUNIT; POTASSIUM CHANNEL TETRAMERIZATION DOMAIN 8 SUBUNIT; UNCLASSIFIED DRUG; 4 AMINOBUTYRIC ACID B RECEPTOR STIMULATING AGENT; BACLOFEN; BENZODIAZEPINE RECEPTOR AFFECTING AGENT; CYCLOPENTANE DERIVATIVE; G PROTEIN COUPLED INWARDLY RECTIFYING POTASSIUM CHANNEL; N,N'-DICYCLOPENTYL-2-METHYLSULFANYL-5-NITRO-PYRIMIDINE-4,6-DIAMINE; POTASSIUM; PYRIMIDINE DERIVATIVE; RECOMBINANT PROTEIN;

ALLOSTERISM; ANIMAL CELL; ARTICLE; BINDING AFFINITY; BRAIN NERVE CELL; CHO CELL LINE; CONTROLLED STUDY; EMBRYO; FEMALE; GENETIC TRANSFECTION; HEK293 CELL LINE; HIPPOCAMPUS; HUMAN; HUMAN CELL; NONHUMAN; POTASSIUM CURRENT; PROTEIN ANALYSIS; PROTEIN ASSEMBLY; PROTEIN INDUCTION; PROTEIN PROTEIN INTERACTION; SIGNAL TRANSDUCTION; ANIMAL; CELL CULTURE; CRICETULUS; DRUG EFFECTS; GENETICS; METABOLISM; MOUSE; NERVE CELL; PHYSIOLOGY; RAT;

ALLOSTERIC REGULATION; ANIMALS; BACLOFEN; CELLS, CULTURED; CHO CELLS; CRICETULUS; CYCLOPENTANES; G PROTEIN-COUPLED INWARDLY-RECTIFYING POTASSIUM CHANNELS; GABA MODULATORS; GABA-B RECEPTOR AGONISTS; GAMMA-AMINOBUTYRIC ACID; GTP-BINDING PROTEINS; HEK293 CELLS; HIPPOCAMPUS; HUMANS; MICE; NEURONS; POTASSIUM; PYRIMIDINES; RATS; RECEPTORS, GABA-B; RECOMBINANT PROTEINS;

EID: 84908374412     PISSN: 00283908     EISSN: 18737064     Source Type: Journal    
DOI: 10.1016/j.neuropharm.2014.08.020     Document Type: Article

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