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Volumn 2014, Issue 17, 2014, Pages 3592-3598

Synthesis of trifluoromethyl-substituted 3-azabicyclo[n.1.0]alkanes: Advanced building blocks for drug discovery

Author keywords

Drug discovery; Fluorine; Nitrogen heterocycles; Synthetic methods; Trifluoromethyldiazomethane

Indexed keywords


EID: 84901845043     PISSN: 1434193X     EISSN: 10990690     Source Type: Journal    
DOI: 10.1002/ejoc.201402158     Document Type: Article
Times cited : (63)

References (83)
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    • The search was performed in July 2013 in "Reaxys" database.
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    • Amine 3 is already offered by at least seven chemical suppliers (MDL, ACD database, 2013)
    • Amine 3 is already offered by at least seven chemical suppliers (MDL, ACD database, 2013).
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    • CCDC-969905 (for 9a) contains the supplementary crystallographic data for this paper. These data can be obtained free of charge from The Cambridge Crystallographic Data Centre via
    • CCDC-969905 (for 9a) contains the supplementary crystallographic data for this paper. These data can be obtained free of charge from The Cambridge Crystallographic Data Centre via www.ccdc.cam.ac.uk/data-request/cif.
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    • Application of amine 11 is covered by ca. 40 patents during the past decade (a search of the Reaxys database was performed in November 2013)
    • Application of amine 11 is covered by ca. 40 patents during the past decade (a search of the Reaxys database was performed in November 2013).
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* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.