-
1
-
-
67650397861
-
Spread and evolution of Plasmodium falciparum drug resistance
-
Mita, T., Tanabe, K. & Kita, K. Spread and evolution of Plasmodium falciparum drug resistance. Parasitol Int 58, 201-209 (2009).
-
(2009)
Parasitol Int
, vol.58
, pp. 201-209
-
-
Mita, T.1
Tanabe, K.2
Kita, K.3
-
2
-
-
68049123592
-
Artemisinin Resistance in Plasmodium falciparum Malaria
-
Dondorp, A. M. et al. Artemisinin Resistance in Plasmodium falciparum Malaria. New England Journal of Medicine 361, 455-467 (2009).
-
(2009)
New England Journal of Medicine
, vol.361
, pp. 455-467
-
-
Dondorp, A.M.1
-
3
-
-
77956280420
-
Spiroindolones, a potent compound class for the treatment of malaria
-
Rottmann, M. et al. Spiroindolones, a potent compound class for the treatment of malaria. Science 329, 1175-1180 (2010).
-
(2010)
Science
, vol.329
, pp. 1175-1180
-
-
Rottmann, M.1
-
4
-
-
0033646097
-
Atovaquone resistance in malaria parasites
-
Vaidya, A. B. & Mather, M. W. Atovaquone resistance in malaria parasites. Drug Resist Updat 3, 283-287 (2000).
-
(2000)
Drug Resist Updat
, vol.3
, pp. 283-287
-
-
Vaidya, A.B.1
Mather, M.W.2
-
5
-
-
35848951143
-
Strategies to reverse drug resistance in malaria
-
DOI 10.1097/QCO.0b013e3282f1673a, PII 0000143220071200000008
-
Egan, T. J. & Kaschula, C. H. Strategies to reverse drug resistance in malaria. Curr Opin Infect Dis 20, 598-604 (2007). (Pubitemid 350059519)
-
(2007)
Current Opinion in Infectious Diseases
, vol.20
, Issue.6
, pp. 598-604
-
-
Egan, T.J.1
Kaschula, C.H.2
-
6
-
-
84861531462
-
Can we teach an old drug new tricks?
-
Ch'ng, J. H., Renia, L., Nosten, F. & Tan, K. S. Can we teach an old drug new tricks? Trends Parasitol 28, 220-224 (2012).
-
(2012)
Trends Parasitol
, vol.28
, pp. 220-224
-
-
Ch'Ng, J.H.1
Renia, L.2
Nosten, F.3
Tan, K.S.4
-
7
-
-
33751211212
-
Quinoline-resistance reversing agents for the malaria parasite Plasmodium falciparum
-
DOI 10.1016/j.drup.2006.09.002, PII S136876460600063X
-
van Schalkwyk, D. A. & Egan, T. J. Quinoline-resistance reversing agents for the malaria parasite Plasmodium falciparum. Drug Resist Updat 9, 211-226 (2006). (Pubitemid 44781212)
-
(2006)
Drug Resistance Updates
, vol.9
, Issue.4-5
, pp. 211-226
-
-
Van Schalkwyk, D.A.1
Egan, T.J.2
-
8
-
-
77949568358
-
Artemisinin resistance: Current status and scenarios for containment
-
Dondorp, A. M. et al. Artemisinin resistance: current status and scenarios for containment. Nat Rev Microbiol 8, 272-280 (2010).
-
(2010)
Nat Rev Microbiol
, vol.8
, pp. 272-280
-
-
Dondorp, A.M.1
-
9
-
-
7244251635
-
Chloroquine resistance in Plasmodium vivax
-
DOI 10.1128/AAC.48.11.4075-4083.2004
-
Baird, J. K. Chloroquine resistance in Plasmodium vivax. Antimicrob Agents Chemother 48, 4075-4083 (2004). (Pubitemid 39434858)
-
(2004)
Antimicrobial Agents and Chemotherapy
, vol.48
, Issue.11
, pp. 4075-4083
-
-
Baird, J.K.1
-
10
-
-
0024204468
-
Stereoselective protein binding of verapamil enantiomers
-
DOI 10.1016/0006-2952(88)90330-9
-
Gross, A. S., Heuer, B. & Eichelbaum, M. Stereoselective protein binding of verapamil enantiomers. Biochem Pharmacol 37, 4623-4627 (1988). (Pubitemid 19006300)
-
(1988)
Biochemical Pharmacology
, vol.37
, Issue.24
, pp. 4623-4627
-
-
Gross, A.S.1
Heuer, B.2
Eichelbaum, M.3
-
11
-
-
79959227019
-
Vivo and in vitro antimalarial properties of azithromycin-chloroquine combinations that include the resistance reversal agent amlodipine
-
Pereira, M. R. et al. In vivo and in vitro antimalarial properties of azithromycin-chloroquine combinations that include the resistance reversal agent amlodipine. Antimicrob Agents Chemother 55, 3115-3124 (2011).
-
(2011)
Antimicrob Agents Chemother
, vol.55
, pp. 3115-3124
-
-
Pereira, M.R.1
-
12
-
-
44949197772
-
Inhibition of efflux of quinolines as new therapeutic strategy in malaria
-
DOI 10.2174/156802608783955593
-
Henry, M., Alibert, S., Rogier, C., Barbe, J. & Pradines, B. Inhibition of efflux of quinolinesas new therapeutic strategyinmalaria. Curr Top Med Chem8, 563-578 (2008). (Pubitemid 351982580)
-
(2008)
Current Topics in Medicinal Chemistry
, vol.8
, Issue.7
, pp. 563-578
-
-
Henry, M.1
Alibert, S.2
Rogier, C.3
Barbe, J.4
Pradines, B.5
-
13
-
-
38749091374
-
Comparative study of interactions between chloroquine and chlorpheniramine or promethazine in healthy volunteers: A potential combination-therapy phenomenon for resuscitating chloroquine for malaria treatment in Africa
-
DOI 10.1179/136485908X252179
-
Gbotosho, G. O. et al. Comparative study of interactions between chloroquine and chlorpheniramine or promethazine in healthy volunteers: a potential combination-therapy phenomenon for resuscitating chloroquine for malaria treatment in Africa. Ann Trop Med Parasitol 102, 3-9 (2008). (Pubitemid 351185238)
-
(2008)
Annals of Tropical Medicine and Parasitology
, vol.102
, Issue.1
, pp. 3-9
-
-
Gbotosho, G.O.1
Happi, C.T.2
Sijuade, A.3
Ogundahunsi, O.A.T.4
Sowunmi, A.5
Oduola, A.M.J.6
-
14
-
-
0033636607
-
Mutations in the P. falciparum digestive vacuole transmembrane protein PfCRT and evidence for their role in chloroquine resistance
-
Fidock, D. A. et al. Mutations in the P. falciparum digestive vacuole transmembrane protein PfCRT and evidence for their role in chloroquine resistance. Mol Cell 6, 861-871 (2000).
-
(2000)
Mol Cell
, vol.6
, pp. 861-871
-
-
Fidock, D.A.1
-
15
-
-
0023918578
-
Antimalarial agents: Mechanism of chloroquine resistance
-
Krogstad, D. J., Schlesinger, P. H. & Herwaldt, B. L. Antimalarial agents: mechanism of chloroquine resistance. Antimicrob Agents Chemother 32, 799-801 (1988).
-
(1988)
Antimicrob Agents Chemother
, vol.32
, pp. 799-801
-
-
Krogstad, D.J.1
Schlesinger, P.H.2
Herwaldt, B.L.3
-
16
-
-
74549192880
-
A comparative study of a flow-cytometry-based assessment of in vitro Plasmodium falciparum drug sensitivity
-
Karl, S., Wong, R. P., St Pierre, T. G. & Davis, T. M. A comparative study of a flow-cytometry-based assessment of in vitro Plasmodium falciparum drug sensitivity. Malar J 8, 294 (2009).
-
(2009)
Malar J
, vol.8
, pp. 294
-
-
Karl, S.1
Wong, R.P.2
St Pierre, T.G.3
Davis, T.M.4
-
17
-
-
84859738849
-
A rapid and robust tri-color flow cytometry assay for monitoring malaria parasite development
-
Malleret, B. et al. A rapid and robust tri-color flow cytometry assay for monitoring malaria parasite development. Sci Rep 1, 118 (2011).
-
(2011)
Sci Rep
, vol.1
, pp. 118
-
-
Malleret, B.1
-
18
-
-
79959211816
-
A programmed cell death pathway in the malaria parasite Plasmodium falciparum has general features of mammalian apoptosis but is mediated by clan CA cysteine proteases
-
Ch'ng, J. H., Kotturi, S. R., Chong, A. G., Lear, M. J. & Tan, K. S. A programmed cell death pathway in the malaria parasite Plasmodium falciparum has general features of mammalian apoptosis but is mediated by clan CA cysteine proteases. Cell Death Dis 1, e26 (2010).
-
(2010)
Cell Death Dis
, vol.1
-
-
Ch'Ng, J.H.1
Kotturi, S.R.2
Chong, A.G.3
Lear, M.J.4
Tan, K.S.5
-
19
-
-
80055012546
-
Drug-induced permeabilization of parasite's digestive vacuole is a key trigger of programmed cell death in Plasmodium falciparum
-
Ch'ng, J. H., Liew, K., Goh, A. S., Sidhartha, E. & Tan, K. S. Drug-induced permeabilization of parasite's digestive vacuole is a key trigger of programmed cell death in Plasmodium falciparum. Cell Death Dis 2, e216 (2011).
-
(2011)
Cell Death Dis
, vol.2
-
-
Ch'Ng, J.H.1
Liew, K.2
Goh, A.S.3
Sidhartha, E.4
Tan, K.S.5
-
20
-
-
0036791883
-
The pH of the Plasmodium falciparum digestive vacuole: Holy grail or dead-end trail?
-
Spiller, D. G., Bray, P. G., Hughes, R. H., Ward, S. A. & White, M. R. The pH of the Plasmodium falciparum digestive vacuole: holy grail or dead-end trail? Trends Parasitol 18, 441-444 (2002).
-
(2002)
Trends Parasitol
, vol.18
, pp. 441-444
-
-
Spiller, D.G.1
Bray, P.G.2
Hughes, R.H.3
Ward, S.A.4
White, M.R.5
-
21
-
-
0036720312
-
Chloroquine resistance in the malarial parasite, Plasmodium falciparum
-
Ursos, L. M. & Roepe, P. D. Chloroquine resistance in the malarial parasite, Plasmodium falciparum. Med Res Rev 22, 465-491 (2002).
-
(2002)
Med Res Rev
, vol.22
, pp. 465-491
-
-
Ursos, L.M.1
Roepe, P.D.2
-
22
-
-
0033824184
-
The effects of chloroquine and verapamil on digestive vacuolar pH of P. falciparum either sensitive or resistant to chloroquine
-
Ursos, L. M., Dzekunov, S. M. & Roepe, P. D. The effects of chloroquine and verapamil on digestive vacuolar pH of P. falciparum either sensitive or resistant to chloroquine. Mol Biochem Parasitol 110, 125-134 (2000).
-
(2000)
Mol Biochem Parasitol
, vol.110
, pp. 125-134
-
-
Ursos, L.M.1
Dzekunov, S.M.2
Roepe, P.D.3
-
23
-
-
0036708526
-
A 3D QSAR pharmacophore model and quantum chemical structure-activity analysis of chloroquine(CQ)-resistance reversal
-
DOI 10.1021/ci0200265
-
Bhattacharjee, A. K., Kyle, D. E., Vennerstrom, J. L. & Milhous, W. K. A 3D QSAR pharmacophore model and quantum chemical structure-activity analysis of chloroquine(CQ)-resistance reversal. J Chem Inf Comp Sci 42, 1212-1220 (2002). (Pubitemid 35360307)
-
(2002)
Journal of Chemical Information and Computer Sciences
, vol.42
, Issue.5
, pp. 1212-1220
-
-
Bhattacharjee, A.K.1
Kyle, D.E.2
Vennerstrom, J.L.3
Milhous, W.K.4
-
24
-
-
0027043104
-
Localization of agonist and antagonist binding domains of the human neurokinin-1 receptor
-
Fong, T. M., Huang, R. R. & Strader, C. D. Localization of agonist and antagonist binding domains of the human neurokinin-1 receptor. J Biol Chem 267, 25664-25667 (1992). (Pubitemid 23013957)
-
(1992)
Journal of Biological Chemistry
, vol.267
, Issue.36
, pp. 25664-25667
-
-
Tung Ming Fong1
Huang, R.-R.C.2
Strader, C.D.3
-
25
-
-
0032420517
-
Clinical pharmacokinetics of mibefradil
-
DOI 10.2165/00003088-199835060-00001
-
Welker, H. A., Wiltshire, H. & Bullingham, R. Clinical pharmacokinetics of mibefradil. Clin Pharmacokinet 35, 405-423 (1998). (Pubitemid 29010173)
-
(1998)
Clinical Pharmacokinetics
, vol.35
, Issue.6
, pp. 405-423
-
-
Welker, H.A.1
Wiltshire, H.2
Bullingham, R.3
-
26
-
-
79961240592
-
Chemical genomic profiling for antimalarial therapies, response signatures, and molecular targets
-
Yuan, J. et al. Chemical genomic profiling for antimalarial therapies, response signatures, and molecular targets. Science 333, 724-729 (2011).
-
(2011)
Science
, vol.333
, pp. 724-729
-
-
Yuan, J.1
-
27
-
-
0034968177
-
Pharmacokinetic interactions of antimalarial agents
-
Giao, P. T. & de Vries, P. J. Pharmacokinetic interactions of antimalarial agents. Clin Pharmacokinet 40, 343-373 (2001). (Pubitemid 32565596)
-
(2001)
Clinical Pharmacokinetics
, vol.40
, Issue.5
, pp. 343-373
-
-
Giao, P.1
De Vries, P.J.2
-
28
-
-
0345096564
-
Chloroquine resistance in Plasmodium chabaudi: Are chloroquine-resistance transporter (crt) and multi-drug resistance (mdr1) orthologues involved?
-
DOI 10.1016/j.molbiopara.2003.08.010
-
Hunt, P., Cravo, P. V., Donleavy, P., Carlton, J. M. & Walliker, D. Chloroquine resistance in Plasmodium chabaudi: are chloroquine-resistance transporter (crt) and multi-drug resistance (mdr1) orthologues involved? Mol Biochem Parasitol 133, 27-35 (2004). (Pubitemid 37510305)
-
(2004)
Molecular and Biochemical Parasitology
, vol.133
, Issue.1
, pp. 27-35
-
-
Hunt, P.1
Cravo, P.V.L.2
Donleavy, P.3
Carlton, J.M.-R.4
Walliker, D.5
-
29
-
-
79851482799
-
Evidence that mutant PfCRT facilitates the transmission to mosquitoes of chloroquine-treated Plasmodium gametocytes
-
Ecker, A., Lakshmanan, V., Sinnis, P., Coppens, I. & Fidock, D. A. Evidence that mutant PfCRT facilitates the transmission to mosquitoes of chloroquine-treated Plasmodium gametocytes. J Infect Dis 203, 228-236 (2011).
-
(2011)
J Infect Dis
, vol.203
, pp. 228-236
-
-
Ecker, A.1
Lakshmanan, V.2
Sinnis, P.3
Coppens, I.4
Fidock, D.A.5
-
30
-
-
84861658779
-
Quantitative genome re-sequencing defines multiple mutations conferring chloroquine resistance in rodent malaria
-
Kinga Modrzynska, K. et al. Quantitative genome re-sequencing defines multiple mutations conferring chloroquine resistance in rodent malaria. BMC Genomics 13, 106 (2012).
-
(2012)
BMC Genomics
, vol.13
, pp. 106
-
-
Kinga Modrzynska, K.1
-
31
-
-
0026825021
-
Plasmodium chabaudi: Association of reversal of chloroquine resistance with increased accumulation of chloroquine in resistant parasites
-
Miki, A., Tanabe, K., Nakayama, T., Kiryon, C. & Ohsawa, K. Plasmodium chabaudi: association of reversal of chloroquine resistance with increased accumulation of chloroquine in resistant parasites. Exp Parasitol 74, 134-142 (1992).
-
(1992)
Exp Parasitol
, vol.74
, pp. 134-142
-
-
Miki, A.1
Tanabe, K.2
Nakayama, T.3
Kiryon, C.4
Ohsawa, K.5
-
32
-
-
0034597616
-
Interaction between chloroquine and diverse pharmacological agents in chloroquine resistant Plasmodium yoelii nigeriensis
-
Singh, N. & Puri, S. K. Interaction between chloroquine and diverse pharmacological agents in chloroquine resistant Plasmodium yoelii nigeriensis. Acta Trop 77, 185-193 (2000).
-
(2000)
Acta Trop
, vol.77
, pp. 185-193
-
-
Singh, N.1
Puri, S.K.2
-
33
-
-
0038416110
-
Structural properties of dibenzosuberanylpiperazine derivatives for efficient reversal of chloroquine resistance in Plasmodium chabaudi
-
DOI 10.1021/jm020379v
-
Osa, Y. et al. Structural properties of dibenzosuberanylpiperazine derivatives for efficient reversal of chloroquine resistance in Plasmodium chabaudi. J Med Chem 46, 1948-1956 (2003). (Pubitemid 36532237)
-
(2003)
Journal of Medicinal Chemistry
, vol.46
, Issue.10
, pp. 1948-1956
-
-
Osa, Y.1
Kobayashi, S.2
Sato, Y.3
Suzuki, Y.4
Takino, K.5
Takeuchi, T.6
Miyata, Y.7
Sakaguchi, M.8
Takayanagi, H.9
|