Cellular uptake and cytotoxicity of drug-peptide conjugates regulated by conjugation site

Bioconjugate Chemistry

Volumn 24, Issue 4, 2013, Pages 604-613

  Zhang, Pengcheng ^a   Cheetham, Andrew G ^a   Lock, Lye Lin ^a   Cui, Honggang ^a  

^a Johns Hopkins University   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CELL CULTURE; CELLS; DISEASES; PEPTIDES;

ANTICANCER DRUG; CANCEROUS CELLS; CELLULAR CYTOTOXICITY; CELLULAR UPTAKE; DOXORUBICIN; DRUG SOLUBILITY; DRUG-PEPTIDES; HYDROPHILICS; MULTIDRUG RESISTANCE; N-TERMINALS;

CYTOTOXICITY;

DOXORUBICIN; DOXORUBICIN TAT; TAT DOXORUBICIN; TRANSACTIVATOR PROTEIN; UNCLASSIFIED DRUG;

ANTINEOPLASTIC ACTIVITY; ARTICLE; CARBOXY TERMINAL SEQUENCE; CELL CULTURE; CELL TRANSPORT; CIRCULAR DICHROISM; CONJUGATION; CONTROLLED STUDY; COVALENT BOND; CYTOTOXICITY; DRUG POTENCY; DRUG SOLUBILITY; HYDROPHILICITY;

EID: 84876485742     PISSN: 10431802     EISSN: 15204812     Source Type: Journal    
DOI: 10.1021/bc300585h     Document Type: Article

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