Selective aminopeptidase-N (CD13) inhibitors with relevance to cancer chemotherapy

Bioorganic and Medicinal Chemistry

Volumn 21, Issue 7, 2013, Pages 2135-2144

  Schmitt, Céline ^a   Voegelin, Manon ^b   Marin, Aurélie ^a   Schmitt, Marjorie ^a   Schegg, Fabienne ^a   Hénon, Philippe ^c   Guenot, Dominique ^b   Tarnus, Céline ^a  

^a UNIVERSITÉ DE HAUTE ALSACE   (France)

^b UNIVERSITÉ DE STRASBOURG   (France)

^c Hopital du Hasenrain CH de Mulhouse   (France)

Author keywords

Aminopeptidase; Antitumor; HIF 1 ; Metalloenzyme; Rapamycin

Indexed keywords

AMINOBENZOSUBERONE DERIVATIVE; ENZYME INHIBITOR; HYPOXIA INDUCIBLE FACTOR 1ALPHA; MICROSOMAL AMINOPEPTIDASE; RAPAMYCIN; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIANGIOGENIC ACTIVITY; ANTIGEN EXPRESSION; ANTINEOPLASTIC ACTIVITY; ARTICLE; CANCER CHEMOTHERAPY; CANCER INHIBITION; CELL MOTILITY; COLON TUMOR; CONCENTRATION RESPONSE; CONTROLLED STUDY; DOWN REGULATION; DRUG EFFICACY; DRUG POTENCY; DRUG SCREENING; DRUG TOLERABILITY; ENDOTHELIUM CELL; FEMALE; HUMAN; HUMAN CELL; HUMAN TISSUE; IN VITRO STUDY; IN VIVO STUDY; MALE; MOUSE; NONHUMAN; NUCLEOTIDE SEQUENCE; SOLID TUMOR; STRUCTURE ACTIVITY RELATION; TUMOR XENOGRAFT;

ANGIOGENESIS INHIBITORS; ANIMALS; ANISOLES; ANTIGENS, CD13; ANTINEOPLASTIC AGENTS; CELL LINE, TUMOR; CELL MOVEMENT; CYCLOHEPTANES; GENE EXPRESSION REGULATION, NEOPLASTIC; HUMANS; HYPOXIA-INDUCIBLE FACTOR 1, ALPHA SUBUNIT; MICE; MICE, NUDE; MOLECULAR TARGETED THERAPY; NEOPLASMS;

MUS; MUS MUSCULUS;

EID: 84875217801     PISSN: 09680896     EISSN: 14643391     Source Type: Journal    
DOI: 10.1016/j.bmc.2012.12.038     Document Type: Article

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