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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 3, 2013, Pages 764-766

Triazole-based inhibitors of geranylgeranyltransferase II

(6) Zhou, Xiang a Hartman, Sara V b Born, Ella J b Smits, Jacqueline P a Holstein, Sarah A b Wiemer, David F a,b

a University of Iowa (United States)

b UNIVERSITY OF IOWA (United States)

Author keywords

Anti proliferative; Apoptosis; Bioassay; GGTase II; Rab GGTase

Indexed keywords

PHYTOENE SYNTHASE; TRIAZOLE DERIVATIVE;

ARTICLE; BIOLOGICAL ACTIVITY; CANCER CELL CULTURE; CLICK CHEMISTRY; CYTOTOXICITY; ENZYME ASSAY; HUMAN; HUMAN CELL; HYDROPHOBICITY; IC 50; IN VITRO STUDY; MYELOMA CELL;

ALKYL AND ARYL TRANSFERASES; APOPTOSIS; CELL LINE, TUMOR; CLICK CHEMISTRY; DIPHOSPHONATES; ENZYME ACTIVATION; HUMANS; INHIBITORY CONCENTRATION 50; MICROBIAL SENSITIVITY TESTS; MOLECULAR STRUCTURE; TRIAZOLES;

EID: 84872346257 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.11.089 Document Type: Article

Times cited : (28)

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