Erratum: Synthesis and biological evaluation of the first dual tyrosyl-DNA phosphodiesterase I (Tdp1)-topoisomerase I (Top1) inhibitors (Journal of Medicinal Chemistry (2012) 55 (4457-4478) DOI:10.1021/jm300335n);Synthesis and biological evaluation of the first dual tyrosyl-DNA phosphodiesterase i (Tdp1)-topoisomerase i (Top1) inhibitors

Journal of Medicinal Chemistry

Volumn 55, Issue 9, 2012, Pages 4457-4478

  Nguyen, Trung Xuan ^a   Morrell, Andrew ^a   Conda Sheridan, Martin ^a   Marchand, Christophe ^b   Agama, Keli ^b   Bermingam, Alun ^c   Stephen, Andrew G ^d   Chergui, Adel ^b   Naumova, Alena ^b   Fisher, Robert ^d   O'Keefe, Barry R ^c   Pommier, Yves ^b   Cushman, Mark ^a  

^a PURDUE UNIVERSITY   (United States)

^b NATIONAL CANCER INSTITUTE   (United States)

^c NATIONAL CANCER INSTITUTE   (United States)

^d SAIC FREDERICK INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

2,5 BIS(4 AMIDINOPHENYL)FURAN; CAMPTOTHECIN; DNA TOPOISOMERASE INHIBITOR; ESTER DERIVATIVE; INDENOISOQUINOLINE DERIVATIVE; ISOQUINOLINE DERIVATIVE; LACTONE; NEOMYCIN; NSC 88915; PHOSPHODIESTERASE I; PHOSPHODIESTERASE INHIBITOR; STEROID; SULFONAMIDE; SULFONIC ACID DERIVATIVE; THYMINE; TOPOTECAN; TYROSYL DNA PHOSPHODIESTERASE I INHIBITOR; UNCLASSIFIED DRUG; VANADIC ACID;

ARTICLE; DNA BINDING; DRUG POTENCY; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME ACTIVE SITE; ENZYME INHIBITION; HYDROPHOBICITY; PHARMACOPHORE; STRUCTURE ACTIVITY RELATION;

EID: 84861078122     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm301167v     Document Type: Erratum

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