Selective histamine H 3 and H 4 receptor agonists exert opposite effects against the gastric lesions induced by HCl in the rat stomach

European Journal of Pharmacology

Volumn 669, Issue 1-3, 2011, Pages 121-127

  Coruzzi, Gabriella ^a   Adami, Maristella ^a   Pozzoli, Cristina ^a   De Esch, Iwan J P ^b   Smits, Rogier ^b   Leurs, Rob ^b  

^a UNIVERSITY OF PARMA   (Italy)

^b VU UNIVERSITY AMSTERDAM   (Netherlands)

Author keywords

Binding; Gastric lesions; HCl; Histamine H 3 receptor; Histamine H 4 receptor

Indexed keywords

1 [2 (AMIDINOTHIO)ETHYL]GUANIDINE; A 331440; HISTAMINE H3 RECEPTOR; HISTAMINE H3 RECEPTOR ANTAGONIST; HISTAMINE H4 RECEPTOR; HISTAMINE H4 RECEPTOR ANTAGONIST; IMMEPIP; IMMETHRIDINE; JNJ 77777120; METHIMEPIP; RANITIDINE; UNCLASSIFIED DRUG; VUF 10460;

ANIMAL EXPERIMENT; ANIMAL MODEL; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG EFFICACY; DRUG INHIBITION; DRUG MEGADOSE; DRUG SELECTIVITY; DRUG STRUCTURE; HUMAN; HUMAN CELL; LIGAND BINDING; MALE; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR BLOCKING; STOMACH LESION; TREATMENT RESPONSE;

ANIMALS; HEK293 CELLS; HISTAMINE AGONISTS; HISTAMINE ANTAGONISTS; HUMANS; HYDROCHLORIC ACID; MALE; PROTEIN BINDING; RADIOLIGAND ASSAY; RATS; RATS, WISTAR; RECEPTORS, G-PROTEIN-COUPLED; RECEPTORS, HISTAMINE; RECEPTORS, HISTAMINE H3; STOMACH ULCER; TRANSFECTION;

EID: 84860404046     PISSN: 00142999     EISSN: 18790712     Source Type: Journal    
DOI: 10.1016/j.ejphar.2011.07.038     Document Type: Article

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