Isoform-selective activation of human constitutive androstane receptor by Ginkgo biloba extract: Functional analysis of the SV23, SV24, and SV25 splice variants

Journal of Pharmacology and Experimental Therapeutics

Volumn 339, Issue 2, 2011, Pages 704-715

  Lau, Aik Jiang ^a   Yang, Guixiang ^a   Chang, Thomas K H ^a  

^a UNIVERSITY OF BRITISH COLUMBIA   (Canada)

Author keywords

[No Author keywords available]

Indexed keywords

1,4 BIS [2 (3,5 DICHLOROPYRIDYLOXY)]BENZENE; 6 (4 CHLOROPHENYL)IMIDAZO[2,1 B][1,3]THIAZOLE 5 CARBALDEHYDE O (3,4 DICHLOROBENZYL)OXIME; CONSTITUTIVE ANDROSTANE RECEPTOR; D (2 ETHYLHEXYL)PHTHALATE; GINKGO BILOBA EXTRACT; GINKGOLIDE A; GINKGOLIDE B; GINKGOLIDE C; GINKGOLIDE J; HORMONE RECEPTOR BLOCKING AGENT; LUCIFERASE; PHENOBARBITAL; RETINOID X RECEPTOR ALPHA; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; DRUG ACTIVITY; ENZYME ACTIVATION; ENZYME ACTIVITY; HUMAN; HUMAN CELL; NUCLEOTIDE SEQUENCE; PLASMID; PRIORITY JOURNAL; PROTEIN BINDING; PROTEIN DOMAIN; PROTEIN EXPRESSION; PROTEIN PROTEIN INTERACTION; PROTEIN VARIANT; REPORTER GENE; TRANSACTIVATION;

GENES, REPORTER; GINKGO BILOBA; GINKGOLIDES; HEP G2 CELLS; HUMANS; LIGANDS; PLANT EXTRACTS; PLASMIDS; PROTEIN ISOFORMS; RECEPTORS, CYTOPLASMIC AND NUCLEAR; RETINOID X RECEPTOR ALPHA; TRANSFECTION; TWO-HYBRID SYSTEM TECHNIQUES;

EID: 80054791510     PISSN: 00223565     EISSN: 15210103     Source Type: Journal    
DOI: 10.1124/jpet.111.186130     Document Type: Article

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