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71
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72
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Single-tablet fixed-dose regimen of elvitegravir/emtricitabine/tenofovir diso-proxil fumarate/GS-9350 achieves a high rate of virologic suppression and GS-9350 is an effective booster [Poster 58LB]
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Cohen C, Shamblaw D, Ruane P, et al. Single-tablet, fixed-dose regimen of elvitegravir/emtricitabine/tenofovir diso-proxil fumarate/GS-9350 achieves a high rate of virologic suppression and GS-9350 is an effective booster [Poster 58LB]. 17th CROI; San Francisco, 16-19 February 2010
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17th CROI
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Cohen, C.1
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Ruane, P.3
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73
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77955590835
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S/GSK1349572 is a potent next generation HIV integrase inhibitor 5th IAS
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74
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77955635152
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Underwood M, Johns B, Sato A, et al. S/GSK1349572: a next generation integrase inhibitor with activity against integrase inhibitor resistant clinical isolates from patients experiencing virologic failure while on raltegravir therapy [Poster WePeA098]. 5th IAS; Cape Town, 19-22 July 2009
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5th IAS
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Underwood, M.1
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Sato, A.3
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75
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S/GSK1349572 Is a potent next generation HIV integrase inhibitor and demonstrates a superior resistance profile substantiated with 60 integrase mutant molecular clones [Poster 555]
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San Francisco 16-19 February
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Seki T, Kobayashi M, Wakasa-Morimoto C, et al. S/GSK1349572 Is a potent next generation HIV integrase inhibitor and demonstrates a superior resistance profile substantiated with 60 integrase mutant molecular clones [Poster 555]. 17th CROI; San Francisco, 16-19 February 2010
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Seki, T.1
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76
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80052408105
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Pharmacokinetic (PK) and safety in healthy subjects of S/GSK1349572, a next generation, once-daily HIV integrase inhibitor (INI)
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Cape Town 19-22 July
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Min S, Song I, Borland J, et al. Pharmacokinetic (PK) and safety in healthy subjects of S/GSK1349572, a next generation, once-daily HIV integrase inhibitor (INI). 5th IAS; Cape Town, 19-22 July 2009
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5th IAS
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Min, S.1
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Borland, J.3
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77
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73849124557
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Pharmacokinetics and safety of S/GSK1349572 a next-generation HIV integrase inhibitor in healthy volunteers [Poster A1-1303]
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78
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77955639715
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Lack of interaction between the HIV integrase inhibitor S/GSK1349572 and tenofovir disoproxil fumarate (TDF) in healthy subjects [Poster 616]
-
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-
Song I, Min S, Borland J, et al. Lack of interaction between the HIV integrase inhibitor, S/GSK1349572, and tenofovir disoproxil fumarate (TDF) in healthy subjects [Poster 616]. 49th ICAAC, 12-15 September 2009
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49th ICAAC
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Song, I.1
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79
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79959271980
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Effect of atazanavir and atazanavir/ritonavir on the pharmacokinetics of the next generation integrase inhibitor S/GSK1349572
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Song I, Borland J, Chen S, et al. Effect of atazanavir and atazanavir/ritonavir on the pharmacokinetics of the next generation integrase inhibitor, S/GSK1349572. 17th CROI; San Francisco, 16-19 February 2010
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17th CROI
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Song, I.1
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80
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77955623511
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Evaluation of antacid and multivitamin (MVI) effects on S/GSK1349572 pharmacokinetics (PK) in healthy subjects [Poster A1-1305]
-
San Francisco 12-15 September
-
Song I, Patel A, Min S, et al. Evaluation of antacid and multivitamin (MVI) effects on S/GSK1349572 pharmacokinetics (PK) in healthy subjects [Poster A1-1305]. 49th ICAAC; San Francisco, 12-15 September 2009
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49th ICAAC
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Song, I.1
Patel, A.2
Min, S.3
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81
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77955603647
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Potent antiviral activity of S/GSK1349572, a next generation integrase inhibitor (INI), in INI-Naive HIV-1-infected patients: ING111521 protocol
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Cape Town 19-22 July Abstract TUAB105
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Lalezari J, Sloan L, DeJesus E, et al. Potent antiviral activity of S/GSK1349572, a next generation integrase inhibitor (INI), in INI-Naive HIV-1-infected patients: ING111521 protocol. 5th IAS. Cape Town, 19-22 July 2009. Abstract TUAB105
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5th IAS
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Sloan, L.2
Dejesus, E.3
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82
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77955634467
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Pharmacokinetic (PK) and pharmacodynamic (PD) relationship of S/GSK1349572 a next generation integrase inhibitor (INI) in HIV-a infected patients [Poster WePeB250]
-
Cape Town 19-22 July
-
Song I, Chen S, Lou Y, et al. Pharmacokinetic (PK) and pharmacodynamic (PD) relationship of S/GSK1349572, a next generation integrase inhibitor (INI), in HIV-a infected patients [Poster WePeB250] 5th IAS; Cape Town; 19-22 July 2009
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Song, I.1
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83
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84
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A clinical research study for assessing the effectiveness of the new integrase inhibitor GSK1349572 in HIV-infected persons with prior antiretroviral treatment and resistance to raltegravir
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Available from
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A clinical research study for assessing the effectiveness of the new integrase inhibitor GSK1349572 in HIV-infected persons with prior antiretroviral treatment and resistance to raltegravir. ClinicalTrials.gov identifier: NCT00950859. Available from http://clinicaltrials.gov/ct2/show/NCT00950859
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ClinicalTrials.gov Identifier: NCT00950859
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85
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77955615956
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Pharmacokinetics (PK) and safety in healthy and HIV-infected subjects and short-term antiviral efficacy of S/GSK1265744 a next generation once daily HIV integrase inhibitor [Poster H-1228]
-
San Francisco 12-15 September
-
Min S, DeJesus E, McCurdy L, et al. Pharmacokinetics (PK) and safety in healthy and HIV-infected subjects and short-term antiviral efficacy of S/GSK1265744, a next generation once daily HIV integrase inhibitor [Poster H-1228]. 49th ICAAC; San Francisco, 12-15 September 2009
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Min, S.1
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86
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Characterization and structural analysis of HIV-1 integrase conservation
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Use of LEDGF/p75 Fusion proteins to retarget lentiviral integration outside of genes [Poster 145]
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Ronen, K.1
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Vets, S.3
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94
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