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Volumn 53, Issue 5, 2010, Pages 2155-2170

Highly potent first examples of dual aromatase-steroid sulfatase inhibitors based on a biphenyl template

Author keywords

[No Author keywords available]

Indexed keywords

3 [(1H 1,2,4 TRIAZOL 1 YL)METHYL) 3' CHLORO 4' HYDROXYBIPHENYL 4 CARBONITRILE; 3 [(1H 1,2,4 TRIAZOL 1 YL)METHYL] 3' HYDROXYBIPHENYL 4 CARBONITRILE; 3 [(1H 1,2,4 TRIAZOL 1 YL)METHYL] 4' HYDROXYBIPHENYL 4 CARBONITRILE; 3' [(1H 1,2,4 TRIAZOL 1 YL)METHYL] 3 CHLORO 4' CYANOBIPHENYL 4 YL SULFAMATE; 3' [(1H 1,2,4 TRIAZOL 1 YL)METHYL] 3 CHLORO-5' CYANOBIPHENYL 4 YL SULFAMATE; 3' [(1H 1,2,4 TRIAZOL 1 YL)METHYL] 3 CHLOROBIPHENYL 4 OL; 3' [(1H 1,2,4 TRIAZOL 1 YL)METHYL] 3 CHLOROBIPHENYL 4 YL SULFAMATE; 3' [(1H 1,2,4 TRIAZOL 1 YL)METHYL] 4' CYANOBIPHENYL 4 YL SULFAMATE; 3' [(1H 1,2,4 TRIAZOL 1 YL)METHYL] 5' CYANOBIPHENYL 4 YL SULFAMATE; 3' [(1H 1,2,4 TRIAZOL 1 YL)METHYL]BIPHENYL 4 OL; 3' [(1H 1,2,4 TRIAZOL 1 YL)METHYL]BIPHENYL 4 YL SULFAMATE; 3;' [(1H 1,2,4 TRIAZOL 1 YL)METHYL] 4' CYANOBIPHENYL 3 YL SULFAMATE; 5 [(1H 1,2,4 TRIAZOL 1 YL)METHYL) 4' FLUOROBIPHENYL 3 CARBONITRILE; 5 [(1H 1,2,4 TRIAZOL 1 YL)METHYL] 3' CHLORO 4' HYDROXYBIPHENYL 2 CARBONITRILE; 5 [(1H 1,2,4 TRIAZOL 1 YL)METHYL] 4' CHLORO 3' HYDROXYBIPHENYL 2 CARBONITRILE; 5 [(1H 1,2,4 TRIAZOL 1 YL)METHYL] 4' HYDROXYBIPHENYL 2 CARBONITRILE; 5 [(1H 1,2,4 TRIAZOL 1 YL)METHYL] 4' HYDROXYBIPHENYL 3 CARBONITRILE; 5 [(1H 1,2,4 TRIAZOL 1 YL)METHYL]BIPHENYL 3 CARBONITRILE; 5 [(1H 1,2,4 TRIAZOL 1 YL)METHYL]BIPHENYL 3' CHLORO 4' HYDROXYBIPHENYL 3 CARBONITRILE; 5 [(1H 1,2,4 TRIAZOL 1 YL)METHYL]BIPHENYL 3,4' DICARBONITRILE; 5' [(1H 1,2,4 TRIAZOL 1 YL)METHYL) 2' CYANOBIPHENYL 4 YL DIMETHYLSULFAMATE; 5' [(1H 1,2,4 TRIAZOL 1 YL)METHYL) 2' CYANOBIPHENYL 4 YL SULFAMATE; 5' [(1H 1,2,4 TRIAZOL 1 YL)METHYL) 3 CHLORO 2' CYANOBIPHENYL 4 YL DIMETHYLSULFAMATE; 5' [(1H 1,2,4 TRIAZOL 1 YL)METHYL) 3 CHLORO 2' CYANOBIPHENYL 4 YL SULFAMATE; 5' [(1H 1,2,4 TRIAZOL 1 YL)METHYL) 4 CHLORO 2' CYANOBIPHENYL 3 YL SULFAMATE; ANASTROZOLE; AROMATASE INHIBITOR; LETROZOLE; STERYL SULFATASE; UNCLASSIFIED DRUG; UNINDEXED DRUG;

EID: 77949346932     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm901705h     Document Type: Article
Times cited : (82)

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