Selective partial agonism of liver X receptor α is related to differential corepressor recruitment

Molecular Endocrinology

Volumn 22, Issue 10, 2008, Pages 2241-2249

  Phelan, Caroline A ^a   Weaver, Joseph M ^a   Steger, David J ^a   Joshi, Shree ^a   Maslany, Jeffrey T ^a   Collins, Jon L ^b   Zuercher, William J ^b   Willson, Timothy M ^b   Walker, Max ^b   Jaye, Michael ^b   Lazar, Mitchell A ^a  

^a UNIVERSITY OF PENNSYLVANIA   (United States)

^b GLAXOSMITHKLINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

3 [3 [[2 CHLORO 3 (TRIFLUOROMETHYL)BENZYL](2 DIPHENYLETHYL)AMINO]PROPOXY]PHENYLACETIC ACID; GSK 224; GW 965; LIVER X RECEPTOR AGONIST; LIVER X RECEPTOR ALPHA; NUCLEAR RECEPTOR COREPRESSOR; SULFONAMIDE; T 09; T 091317; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DISSOCIATION; DRUG EFFICACY; DRUG POTENCY; DRUG SELECTIVITY; EMBRYO; GENE EXPRESSION; GENE TARGETING; HUMAN; HUMAN CELL; LIGAND BINDING; PRIORITY JOURNAL; PROTEIN BINDING;

BENZOIC ACIDS; BENZYLAMINES; CELL LINE; DIMERIZATION; DNA-BINDING PROTEINS; HUMANS; LIGANDS; MOLECULAR STRUCTURE; NUCLEAR PROTEINS; RECEPTORS, CYTOPLASMIC AND NUCLEAR; REPRESSOR PROTEINS; RETINOID X RECEPTORS; RNA INTERFERENCE; SULFONAMIDES; TRANS-ACTIVATION (GENETICS);

EID: 52949139843     PISSN: 08888809     EISSN: None     Source Type: Journal    
DOI: 10.1210/me.2008-0041     Document Type: Article

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