Structural and functional definition of the specificity of a novel caspase-3 inhibitor, Ac-DNLD-CHO

BMC Pharmacology

Volumn 7, Issue , 2007, Pages

  Yoshimori, Atsushi ^a,b   Sakai, Junichi ^b   Sunaga, Satoshi ^b   Kobayashi, Takanobu ^c   Takahashi, Satoshi ^a   Okita, Naoyuki ^b   Takasawa, Ryoko ^b   Tanuma, Sei Ichi ^b  

^a Venture Kanda 504   (Japan)

^b TOKYO UNIVERSITY OF SCIENCE   (Japan)

^c TOKUSHIMA BUNRI UNIVERSITY   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

ALANINE; ASPARAGINE; CASPASE 3; CASPASE 3 INHIBITOR; CASPASE 7; CASPASE 8; CASPASE 9; LEUCINE; SERINE; CYSTEINE PROTEINASE INHIBITOR; OLIGOPEPTIDE; RECOMBINANT PROTEIN;

AMINO ACID SEQUENCE; AMINO ACID SUBSTITUTION; APOPTOSIS; ARTICLE; DRUG DESIGN; DRUG POTENCY; DRUG RESEARCH; DRUG SELECTIVITY; ENZYME ACTIVE SITE; ENZYME ACTIVITY; ENZYME INHIBITION; ENZYME SPECIFICITY; ENZYME STRUCTURE; ENZYME SUBSTRATE; FLUOROMETRY; HYDROPHOBICITY; INFLAMMATION; MOLECULAR RECOGNITION; PROTEIN FAMILY; SITE DIRECTED MUTAGENESIS; X RAY CRYSTALLOGRAPHY; BINDING SITE; CHEMISTRY; DRUG ANTAGONISM; HUMAN; METABOLISM;

BINDING SITES; CASPASE 3; CYSTEINE PROTEINASE INHIBITORS; HUMANS; OLIGOPEPTIDES; RECOMBINANT PROTEINS;

EID: 34547430973     PISSN: None     EISSN: 14712210     Source Type: Journal    
DOI: 10.1186/1471-2210-7-8     Document Type: Article

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