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Volumn 553, Issue 1-3, 2006, Pages 73-81

Involvement of I2-imidazoline binding sites in positive and negative morphine analgesia modulatory effects

Author keywords

Diphenyzoline; I2 IBS (I2 imidazoline binding sites); I2 IBS ligands; Morphine analgesia modulation; Phenyzoline

Indexed keywords

ALPHA 2 ADRENERGIC RECEPTOR; ALPHA 2 ADRENERGIC RECEPTOR BLOCKING AGENT; BENZENE DERIVATIVE; DIPHENYZOLINE; EFAROXAN; IDAZOXAN; IMIDAZOLINE I2 RECEPTOR; MORPHINE; MU OPIATE RECEPTOR; NALOXONE; PHENYZOLINE; TRACIZOLINE; UNCLASSIFIED DRUG; YOHIMBINE; ALPHA ADRENERGIC RECEPTOR BLOCKING AGENT; BENZOFURAN DERIVATIVE; DRUG RECEPTOR; IMIDAZOLE DERIVATIVE; IMIDAZOLINE RECEPTOR 2; NARCOTIC ANALGESIC AGENT; NARCOTIC ANTAGONIST;

EID: 33751190283     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejphar.2006.09.031     Document Type: Article
Times cited : (34)

References (49)
  • 1
    • 0030611203 scopus 로고    scopus 로고
    • 3H]2-(2-benzofuranyl)-2-imidazoline (2-BFI) in rat brain and liver: characterization, regulation and relation to monoamine oxidase enzymes
    • 3H]2-(2-benzofuranyl)-2-imidazoline (2-BFI) in rat brain and liver: characterization, regulation and relation to monoamine oxidase enzymes. Naunyn-Schmiedeberg's Arch. Pharmacol. 356 (1997) 39-47
    • (1997) Naunyn-Schmiedeberg's Arch. Pharmacol. , vol.356 , pp. 39-47
    • Alemany, R.1    Olmos, G.2    Garcìa-Sevilla, J.A.3
  • 3
    • 0035514525 scopus 로고    scopus 로고
    • I1 receptors, cardiovascular function, and metabolism
    • Bousquet P. I1 receptors, cardiovascular function, and metabolism. Am. J. Hypertens. 14 (2001) 317S-321S
    • (2001) Am. J. Hypertens. , vol.14
    • Bousquet, P.1
  • 4
    • 0021153959 scopus 로고
    • Central cardiovascular effects of alpha adrenergic drugs: differences between catecholamines and imidazolines
    • Bousquet P., Feldman J., and Schwartz J. Central cardiovascular effects of alpha adrenergic drugs: differences between catecholamines and imidazolines. J. Pharmacol. Exp. Ther. 230 (1984) 232-236
    • (1984) J. Pharmacol. Exp. Ther. , vol.230 , pp. 232-236
    • Bousquet, P.1    Feldman, J.2    Schwartz, J.3
  • 7
    • 3843115467 scopus 로고    scopus 로고
    • Imidazoline binding sites and their ligands: an overview of the different chemical structures
    • Dardonville C., and Rozas I. Imidazoline binding sites and their ligands: an overview of the different chemical structures. Med. Res. Rev. 24 (2004) 639-661
    • (2004) Med. Res. Rev. , vol.24 , pp. 639-661
    • Dardonville, C.1    Rozas, I.2
  • 8
    • 0018001339 scopus 로고
    • Simultaneous analysis of families of sigmoidal curves: application to bioassay, radioligand assay, and physiological dose-response curves
    • DeLean A., Munson P.J., and Rodbard D. Simultaneous analysis of families of sigmoidal curves: application to bioassay, radioligand assay, and physiological dose-response curves. Am. J. Physiol. 235 (1978) E97-E102
    • (1978) Am. J. Physiol. , vol.235
    • DeLean, A.1    Munson, P.J.2    Rodbard, D.3
  • 9
    • 0033874470 scopus 로고    scopus 로고
    • Autoradiographic mapping of μ-opioid receptors during opiate tolerance and supersensitivity in the rat central nervous system
    • Diaz A., Pazos A., Florez J., and Hurle M.A. Autoradiographic mapping of μ-opioid receptors during opiate tolerance and supersensitivity in the rat central nervous system. Naunyn-Schmiedeberg's Arch. Pharmacol. 362 (2000) 101-109
    • (2000) Naunyn-Schmiedeberg's Arch. Pharmacol. , vol.362 , pp. 101-109
    • Diaz, A.1    Pazos, A.2    Florez, J.3    Hurle, M.A.4
  • 11
    • 0032768991 scopus 로고    scopus 로고
    • Pharmacological characterization of imidazoline receptor proteins identified by immunologic techniques and other methods
    • Escriba P.V., Ozaita A., and Garcia-Sevilla J.A. Pharmacological characterization of imidazoline receptor proteins identified by immunologic techniques and other methods. Ann. N. Y. Acad. Sci. 881 (1999) 8-25
    • (1999) Ann. N. Y. Acad. Sci. , vol.881 , pp. 8-25
    • Escriba, P.V.1    Ozaita, A.2    Garcia-Sevilla, J.A.3
  • 12
    • 0031772025 scopus 로고    scopus 로고
    • Aspects on tail-flick, hot-plate and electrical stimulation tests for morphine antinociception
    • Gardmark M., Hoglund A.U., and Hammarlund-Udenaes M. Aspects on tail-flick, hot-plate and electrical stimulation tests for morphine antinociception. Pharmacol. Toxicol. 83 (1998) 252-258
    • (1998) Pharmacol. Toxicol. , vol.83 , pp. 252-258
    • Gardmark, M.1    Hoglund, A.U.2    Hammarlund-Udenaes, M.3
  • 17
    • 0031752441 scopus 로고    scopus 로고
    • Evidence for the existence of imidazoline-specific binding sites in synaptosomal plasma membranes of the bovine brainstem
    • Heemskerk F.M., Dontenwill M., Greney H., Vonthron C., and Bousquet P. Evidence for the existence of imidazoline-specific binding sites in synaptosomal plasma membranes of the bovine brainstem. J. Neurochem. 71 (1998) 2193-2202
    • (1998) J. Neurochem. , vol.71 , pp. 2193-2202
    • Heemskerk, F.M.1    Dontenwill, M.2    Greney, H.3    Vonthron, C.4    Bousquet, P.5
  • 20
    • 0032520845 scopus 로고    scopus 로고
    • A point mutation (D79N) of the α2A adrenergic receptor abolishes the antiepileptogenic action of endogenous norepinephrine
    • Janumpalli S., Butler L.S., MacMillan L.B., Limbird L.E., and McNamara J.O. A point mutation (D79N) of the α2A adrenergic receptor abolishes the antiepileptogenic action of endogenous norepinephrine. J. Neurosci. 18 (1998) 2004-2008
    • (1998) J. Neurosci. , vol.18 , pp. 2004-2008
    • Janumpalli, S.1    Butler, L.S.2    MacMillan, L.B.3    Limbird, L.E.4    McNamara, J.O.5
  • 21
    • 0034737589 scopus 로고    scopus 로고
    • A new protocol for the synthesis of N(1)-unsubstituted 2-substituted 2-imidazolines
    • Jones R.C.F., and Dimopoulos P. A new protocol for the synthesis of N(1)-unsubstituted 2-substituted 2-imidazolines. Tetrahedron 56 (2000) 2061-2074
    • (2000) Tetrahedron , vol.56 , pp. 2061-2074
    • Jones, R.C.F.1    Dimopoulos, P.2
  • 23
    • 0030610424 scopus 로고    scopus 로고
    • Substitution of a mutant alpha2a-adrenergic receptor via "hit and run" gene targeting reveals the role of this subtype in sedative, analgesic, and anesthetic-sparing responses in vivo
    • Lakhlani P.P., MacMillan L.B., Guo T.Z., McCool B.A., Lovinger D.M., Maze M., and Limbird L.E. Substitution of a mutant alpha2a-adrenergic receptor via "hit and run" gene targeting reveals the role of this subtype in sedative, analgesic, and anesthetic-sparing responses in vivo. Proc. Natl. Acad. Sci. U. S. A. 94 (1997) 9950-9955
    • (1997) Proc. Natl. Acad. Sci. U. S. A. , vol.94 , pp. 9950-9955
    • Lakhlani, P.P.1    MacMillan, L.B.2    Guo, T.Z.3    McCool, B.A.4    Lovinger, D.M.5    Maze, M.6    Limbird, L.E.7
  • 24
    • 0029147286 scopus 로고
    • Hot plate versus tail flick: evaluation of acute tolerance to continuous morphine infusion in the rat model
    • Langerman L., Zakowski M.I., Piskoun B., and Grant G.J. Hot plate versus tail flick: evaluation of acute tolerance to continuous morphine infusion in the rat model. J. Pharmacol. Toxicol. Methods 34 (1995) 23-27
    • (1995) J. Pharmacol. Toxicol. Methods , vol.34 , pp. 23-27
    • Langerman, L.1    Zakowski, M.I.2    Piskoun, B.3    Grant, G.J.4
  • 25
  • 26
    • 0026062486 scopus 로고
    • Possible mechanism of morphine analgesia
    • Lipp J. Possible mechanism of morphine analgesia. Clin. Neuropharmacol. 14 (1991) 131-147
    • (1991) Clin. Neuropharmacol. , vol.14 , pp. 131-147
    • Lipp, J.1
  • 27
    • 0029777474 scopus 로고    scopus 로고
    • Central hypotensive effects of the alpha2a-adrenergic receptor subtype
    • MacMillan L.B., Hein L., Smith M.S., Piascik M.T., and Limbird L.E. Central hypotensive effects of the alpha2a-adrenergic receptor subtype. Science 273 (1996) 801-803
    • (1996) Science , vol.273 , pp. 801-803
    • MacMillan, L.B.1    Hein, L.2    Smith, M.S.3    Piascik, M.T.4    Limbird, L.E.5
  • 28
    • 0006695557 scopus 로고    scopus 로고
    • Models of nociception: hot-plate, tail-flick, and formalin tests in rodents
    • Crawley J.N., Gerfen C.R., Rogawski M.A., Sibley D.R., Skolnick P., and Wray S. (Eds), John Wiley & Sons, New York, NY
    • Malmberg A.B., and Bannon A.W. Models of nociception: hot-plate, tail-flick, and formalin tests in rodents. In: Crawley J.N., Gerfen C.R., Rogawski M.A., Sibley D.R., Skolnick P., and Wray S. (Eds). Current Protocols in Neuroscience (1999), John Wiley & Sons, New York, NY 8.9.1-8.9.15
    • (1999) Current Protocols in Neuroscience
    • Malmberg, A.B.1    Bannon, A.W.2
  • 29
    • 0031181346 scopus 로고    scopus 로고
    • QXP: powerful, rapid computer algorithms for structure-based drug design
    • McMartin C., and Bohacek R.S. QXP: powerful, rapid computer algorithms for structure-based drug design. J. Comput.-Aided Mol. Des. 11 (1997) 333-344
    • (1997) J. Comput.-Aided Mol. Des. , vol.11 , pp. 333-344
    • McMartin, C.1    Bohacek, R.S.2
  • 30
    • 0036277865 scopus 로고    scopus 로고
    • Descending control of pain
    • Millan M.J. Descending control of pain. Prog. Neurobiol. 66 (2002) 355-474
    • (2002) Prog. Neurobiol. , vol.66 , pp. 355-474
    • Millan, M.J.1
  • 31
    • 0029758145 scopus 로고    scopus 로고
    • Antisense technology reveals the alpha2A adrenoceptor to be the subtype mediating the hypnotic response to the highly selective agonist, dexmedetomidine, in the locus coeruleus of the rat
    • Mizobe T., Maghsoudi K., Sitwala K., Tianzhi G., Ou J., and Maze M. Antisense technology reveals the alpha2A adrenoceptor to be the subtype mediating the hypnotic response to the highly selective agonist, dexmedetomidine, in the locus coeruleus of the rat. J. Clin. Invest. 98 (1996) 1076-1080
    • (1996) J. Clin. Invest. , vol.98 , pp. 1076-1080
    • Mizobe, T.1    Maghsoudi, K.2    Sitwala, K.3    Tianzhi, G.4    Ou, J.5    Maze, M.6
  • 32
    • 0030759252 scopus 로고    scopus 로고
    • Imidazoline receptors: basic knowledge, recent advances and future prospects for therapy and diagnosis
    • Molderings G.J. Imidazoline receptors: basic knowledge, recent advances and future prospects for therapy and diagnosis. Drugs Future 22 (1997) 757-772
    • (1997) Drugs Future , vol.22 , pp. 757-772
    • Molderings, G.J.1
  • 33
    • 0345367512 scopus 로고    scopus 로고
    • Imidazoline binding sites and receptors in cardiovascular tissue
    • Molderings G.J., and Gothert M. Imidazoline binding sites and receptors in cardiovascular tissue. Gen. Pharmacol. 32 (1999) 17-22
    • (1999) Gen. Pharmacol. , vol.32 , pp. 17-22
    • Molderings, G.J.1    Gothert, M.2
  • 37
    • 0031008545 scopus 로고    scopus 로고
    • Imidazoline receptors: qualitative structure-activity relationships and discovery of tracizoline and benazoline. Two ligands with high affinity and unprecedented selectivity
    • Pigini M., Bousquet P., Carotti A., Dontenwill M., Giannella M., Moriconi R., Piergentili A., Quaglia W., Tayebati S.K., and Brasili L. Imidazoline receptors: qualitative structure-activity relationships and discovery of tracizoline and benazoline. Two ligands with high affinity and unprecedented selectivity. Bioorg. Med. Chem. 5 (1997) 833-841
    • (1997) Bioorg. Med. Chem. , vol.5 , pp. 833-841
    • Pigini, M.1    Bousquet, P.2    Carotti, A.3    Dontenwill, M.4    Giannella, M.5    Moriconi, R.6    Piergentili, A.7    Quaglia, W.8    Tayebati, S.K.9    Brasili, L.10
  • 40
    • 0032509769 scopus 로고    scopus 로고
    • Immunocytochemical localization of an imidazoline receptor protein in the central nervous system
    • Ruggiero D.A., Regunathan S., Wang H., Milner T.A., and Reis D.J. Immunocytochemical localization of an imidazoline receptor protein in the central nervous system. Brain Res. 780 (1998) 270-293
    • (1998) Brain Res. , vol.780 , pp. 270-293
    • Ruggiero, D.A.1    Regunathan, S.2    Wang, H.3    Milner, T.A.4    Reis, D.J.5
  • 41
    • 0037331173 scopus 로고    scopus 로고
    • Attenuation of acute and chronic effects of morphine by the imidazoline receptor ligand 2-(2-benzofuranyl)-2-imidazoline in rat locus coeruleus neurons
    • Ruiz-Durantez E., Torrecilla M., Pineda J., and Ugedo L. Attenuation of acute and chronic effects of morphine by the imidazoline receptor ligand 2-(2-benzofuranyl)-2-imidazoline in rat locus coeruleus neurons. Br. J. Pharmacol. 138 (2003) 494-500
    • (2003) Br. J. Pharmacol. , vol.138 , pp. 494-500
    • Ruiz-Durantez, E.1    Torrecilla, M.2    Pineda, J.3    Ugedo, L.4
  • 42
    • 0034100844 scopus 로고    scopus 로고
    • 2-imidazoline receptors enhances supraspinal morphine analgesia in mice: a model to detect agonist and antagonist activities at these receptors
    • 2-imidazoline receptors enhances supraspinal morphine analgesia in mice: a model to detect agonist and antagonist activities at these receptors. Br. J. Pharmacol. 130 (2000) 146-152
    • (2000) Br. J. Pharmacol. , vol.130 , pp. 146-152
    • Sanchez-Blazquez, P.1    Boronat, M.A.2    Olmos, G.3    Garcìa-Sevilla, J.A.4    Garzon, J.5
  • 44
    • 0032775303 scopus 로고    scopus 로고
    • Peripheral and central imidazoline receptor-mediated natriuresis in the rat
    • Smyth D.D., and Penner S.B. Peripheral and central imidazoline receptor-mediated natriuresis in the rat. Ann. N. Y. Acad. Sci. 881 (1999) 344-357
    • (1999) Ann. N. Y. Acad. Sci. , vol.881 , pp. 344-357
    • Smyth, D.D.1    Penner, S.B.2
  • 45
    • 0034960352 scopus 로고    scopus 로고
    • Down-regulation of MAO-B activity and imidazoline receptors in rat brain following chronic treatment of morphine
    • Su R.B., Li J., Li X., and Qin B.Y. Down-regulation of MAO-B activity and imidazoline receptors in rat brain following chronic treatment of morphine. Acta Pharmacol. Sin. 22 (2001) 639-644
    • (2001) Acta Pharmacol. Sin. , vol.22 , pp. 639-644
    • Su, R.B.1    Li, J.2    Li, X.3    Qin, B.Y.4
  • 46
    • 0025866818 scopus 로고
    • Identification of an imidazoline-guanidinium receptive site in mitochondria from rabbit cerebral cortex
    • Tesson F., and Parini A. Identification of an imidazoline-guanidinium receptive site in mitochondria from rabbit cerebral cortex. Eur. J. Pharmacol. 208 (1991) 81-83
    • (1991) Eur. J. Pharmacol. , vol.208 , pp. 81-83
    • Tesson, F.1    Parini, A.2
  • 47
    • 0026662748 scopus 로고
    • Tissue-specific localization of mitochondrial imidazoline-guanidinium receptive site
    • Tesson F., Limon I., and Parini A. Tissue-specific localization of mitochondrial imidazoline-guanidinium receptive site. Eur. J. Pharmacol. 219 (1992) 335-338
    • (1992) Eur. J. Pharmacol. , vol.219 , pp. 335-338
    • Tesson, F.1    Limon, I.2    Parini, A.3
  • 49
    • 0025966628 scopus 로고
    • Species differences in μ- and δ-opioid receptors
    • Yoburn B.C., Lutfy K., and Candido J. Species differences in μ- and δ-opioid receptors. Eur. J. Pharmacol. 193 (1991) 105-108
    • (1991) Eur. J. Pharmacol. , vol.193 , pp. 105-108
    • Yoburn, B.C.1    Lutfy, K.2    Candido, J.3


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