-
10
-
-
11044223276
-
-
Danishefsky S.J., Masters J.J., Young W.B., Link J.T., Snyder L.B., Magee T.V., Jung D.K., Isaacs R.C.A., Bornmann W.G., Alaimo C.A., Coburn C.A., and DiGrandi M.J. J. Am. Chem. Soc. 118 (1996) 2843-2859
-
(1996)
J. Am. Chem. Soc.
, vol.118
, pp. 2843-2859
-
-
Danishefsky, S.J.1
Masters, J.J.2
Young, W.B.3
Link, J.T.4
Snyder, L.B.5
Magee, T.V.6
Jung, D.K.7
Isaacs, R.C.A.8
Bornmann, W.G.9
Alaimo, C.A.10
Coburn, C.A.11
DiGrandi, M.J.12
-
11
-
-
0034716749
-
-
Kusama H., Hara R., Kawahara S., Nishimori T., Kashima H., Nakamura N., Morihira K., and Kuwajima I. J. Am. Chem. Soc. 122 (2000) 3811-3820
-
(2000)
J. Am. Chem. Soc.
, vol.122
, pp. 3811-3820
-
-
Kusama, H.1
Hara, R.2
Kawahara, S.3
Nishimori, T.4
Kashima, H.5
Nakamura, N.6
Morihira, K.7
Kuwajima, I.8
-
12
-
-
5644287433
-
-
Kikuno N., Moriyama-Gonda N., Yoshino T., Yoneda T., Urakami S., Terashima M., Yoshida M., Kishi H., Shigeno K., Shiina H., and Igawa M. Cancer Res. 64 (2004) 7526-7532
-
(2004)
Cancer Res.
, vol.64
, pp. 7526-7532
-
-
Kikuno, N.1
Moriyama-Gonda, N.2
Yoshino, T.3
Yoneda, T.4
Urakami, S.5
Terashima, M.6
Yoshida, M.7
Kishi, H.8
Shigeno, K.9
Shiina, H.10
Igawa, M.11
-
13
-
-
13444291204
-
-
Menendez J.A., Vellon L., Mehmi I., Teng P.K., Griggs D.W., and Lupu R. Oncogene 24 (2005) 761-779
-
(2005)
Oncogene
, vol.24
, pp. 761-779
-
-
Menendez, J.A.1
Vellon, L.2
Mehmi, I.3
Teng, P.K.4
Griggs, D.W.5
Lupu, R.6
-
14
-
-
0032959590
-
-
Mark Roe S., Prodromou C., O' Brien R., Ladbury J.E., Piper P.W., and Pearl L.H. J. Med. Chem. 42 (1999) 260-266
-
(1999)
J. Med. Chem.
, vol.42
, pp. 260-266
-
-
Mark Roe, S.1
Prodromou, C.2
O' Brien, R.3
Ladbury, J.E.4
Piper, P.W.5
Pearl, L.H.6
-
16
-
-
0037451452
-
-
Yamamoto K., Garbaccio R.M., Stachel S.J., Solit D.B., Chiosis G., Rosen N., and Danishefsky S.J. Angew. Chem., Int. Ed. 42 (2003) 1280-1284
-
(2003)
Angew. Chem., Int. Ed.
, vol.42
, pp. 1280-1284
-
-
Yamamoto, K.1
Garbaccio, R.M.2
Stachel, S.J.3
Solit, D.B.4
Chiosis, G.5
Rosen, N.6
Danishefsky, S.J.7
-
21
-
-
0038575020
-
-
Yang Z.Q., Kwok B.H., Lin S., Koldobskiy M.A., Crews C.M., and Danishefsky S.J. Chembiochem 6 (2003) 508-513
-
(2003)
Chembiochem
, vol.6
, pp. 508-513
-
-
Yang, Z.Q.1
Kwok, B.H.2
Lin, S.3
Koldobskiy, M.A.4
Crews, C.M.5
Danishefsky, S.J.6
-
22
-
-
0038112083
-
-
Inoue M., Sakazaki H., Furuyama H., and Hirama M. Angew. Chem., Int. Ed. 42 (2003) 2654-2657
-
(2003)
Angew. Chem., Int. Ed.
, vol.42
, pp. 2654-2657
-
-
Inoue, M.1
Sakazaki, H.2
Furuyama, H.3
Hirama, M.4
-
23
-
-
20144377696
-
-
Galsky M.D., Small E.J., Oh W.K., Chen I., Smith D.C., Dimitrios Colevas A., Martone L., Curley T., DeLaCruz A., Scher H.I., and Kelly W.K. J. Clin. Oncol. 23 (2005) 1439-1446
-
(2005)
J. Clin. Oncol.
, vol.23
, pp. 1439-1446
-
-
Galsky, M.D.1
Small, E.J.2
Oh, W.K.3
Chen, I.4
Smith, D.C.5
Dimitrios Colevas, A.6
Martone, L.7
Curley, T.8
DeLaCruz, A.9
Scher, H.I.10
Kelly, W.K.11
-
24
-
-
20244376916
-
-
Zhuang S.H., Agrawal M., Edgerly M., Bakke S., Kotz H., Thambi P., Rutt A., Balis F.M., Bates S., and Fojo T. Cancer 103 (2005) 1932-1938
-
(2005)
Cancer
, vol.103
, pp. 1932-1938
-
-
Zhuang, S.H.1
Agrawal, M.2
Edgerly, M.3
Bakke, S.4
Kotz, H.5
Thambi, P.6
Rutt, A.7
Balis, F.M.8
Bates, S.9
Fojo, T.10
-
25
-
-
33746022358
-
-
Annual Meeting of the American Society of Clinical Oncology (ASCO), Orlando, May 13-17, 2005, Abstract 2050.
-
-
-
-
26
-
-
18744385682
-
Phase 1 dose escalating and pharmacokinetic (PK) study of KOS-862 (epothilone D): Phase 2 dose and schedule defined
-
AACR-NCI-EORTC International Conference: Molecular Targets and Cancer Therapeutics, November 17-21, 2003, Boston, MA, USA
-
Spriggs D., Dupont J., Pezzulli S., Larkin J., Cropp J., and Johnson R. Phase 1 dose escalating and pharmacokinetic (PK) study of KOS-862 (epothilone D): Phase 2 dose and schedule defined. AACR-NCI-EORTC International Conference: Molecular Targets and Cancer Therapeutics, November 17-21, 2003, Boston, MA, USA. Clin. Cancer Res. 9 (2003)
-
(2003)
Clin. Cancer Res.
, vol.9
-
-
Spriggs, D.1
Dupont, J.2
Pezzulli, S.3
Larkin, J.4
Cropp, J.5
Johnson, R.6
-
27
-
-
33745978462
-
-
Annual Meeting of the American Society of Clinical Oncology (ASCO), Orlando, May 13-17, 2005, Abstract 2049.
-
-
-
-
29
-
-
0033757121
-
-
Nakae K., Yoshimoto Y., Sawa T., Homma Y., Hamada M., Takeuchi T., and Imoto M. J. Antibiot. 53 (2000) 1130-1136
-
(2000)
J. Antibiot.
, vol.53
, pp. 1130-1136
-
-
Nakae, K.1
Yoshimoto, Y.2
Sawa, T.3
Homma, Y.4
Hamada, M.5
Takeuchi, T.6
Imoto, M.7
-
30
-
-
0033762667
-
-
Nakae K., Yoshimoto Y., Ueda M., Sawa T., Takahashi Y., Naganawa H., Takeuchi T., and Imoto M. J. Antibiot. 53 (2000) 1228-1230
-
(2000)
J. Antibiot.
, vol.53
, pp. 1228-1230
-
-
Nakae, K.1
Yoshimoto, Y.2
Ueda, M.3
Sawa, T.4
Takahashi, Y.5
Naganawa, H.6
Takeuchi, T.7
Imoto, M.8
-
31
-
-
0035700559
-
-
Takemoto Y., Nakae K., Kawatani M., Takahashi Y., Naganawa H., and Imoto M. J. Antibiot. 54 (2001) 1104-1107
-
(2001)
J. Antibiot.
, vol.54
, pp. 1104-1107
-
-
Takemoto, Y.1
Nakae, K.2
Kawatani, M.3
Takahashi, Y.4
Naganawa, H.5
Imoto, M.6
-
32
-
-
14844343474
-
-
Shan, D.; Chen, L.; Njardarson, J. T.; Gaul, C.; Ma, X.; Danishefsky, S. J.; Huang, X.-Y. In Proceedings of Natural Academy of Science (PNAS), 2005; Vol. 102, pp 3772-3776.
-
-
-
-
34
-
-
0942265463
-
-
Njardarson J.T., Gaul C., Shan D., Huang X.-Y., and Danishefsky S.J. J. Am. Chem. Soc. 126 (2004) 1038-1040
-
(2004)
J. Am. Chem. Soc.
, vol.126
, pp. 1038-1040
-
-
Njardarson, J.T.1
Gaul, C.2
Shan, D.3
Huang, X.-Y.4
Danishefsky, S.J.5
-
35
-
-
4544233786
-
-
Gaul C., Njardarson J.T., Shan D., Dorn D.C., Wu K.-D., Tong W.P., Huang X.-Y., Moore M.A.S., and Danishefsky S.J. J. Am. Chem. Soc. 126 (2004) 11326-11337
-
(2004)
J. Am. Chem. Soc.
, vol.126
, pp. 11326-11337
-
-
Gaul, C.1
Njardarson, J.T.2
Shan, D.3
Dorn, D.C.4
Wu, K.-D.5
Tong, W.P.6
Huang, X.-Y.7
Moore, M.A.S.8
Danishefsky, S.J.9
-
38
-
-
4644228335
-
-
Yu W., Mei Y., Kang Y., Hua Z., and Jin Z. Org. Lett. 6 (2004) 3217-3219
-
(2004)
Org. Lett.
, vol.6
, pp. 3217-3219
-
-
Yu, W.1
Mei, Y.2
Kang, Y.3
Hua, Z.4
Jin, Z.5
-
42
-
-
0034725908
-
-
Ando K., Oishi T., Hirama M., Ohno H., and Ibuka T. J. Org. Chem. 65 (2000) 4745-4749
-
(2000)
J. Org. Chem.
, vol.65
, pp. 4745-4749
-
-
Ando, K.1
Oishi, T.2
Hirama, M.3
Ohno, H.4
Ibuka, T.5
-
43
-
-
33746022661
-
-
note
-
+] 343.1885, found 343.1876.
-
-
-
-
44
-
-
0001616071
-
-
Inanaga J., Hirata K., Saeki H., Katsuki T., and Yamaguchi M. Bull. Chem. Soc. Jpn. 52 (1979) 1989-1993
-
(1979)
Bull. Chem. Soc. Jpn.
, vol.52
, pp. 1989-1993
-
-
Inanaga, J.1
Hirata, K.2
Saeki, H.3
Katsuki, T.4
Yamaguchi, M.5
-
45
-
-
0037149026
-
-
For a recent example, see:
-
For a recent example, see:. Song F., Fidanze S., Benowitz A.B., and Kishi Y. Org. Lett. 4 (2002) 647-650
-
(2002)
Org. Lett.
, vol.4
, pp. 647-650
-
-
Song, F.1
Fidanze, S.2
Benowitz, A.B.3
Kishi, Y.4
-
49
-
-
33745992991
-
-
note
-
+] 423.2147, found 423.2131.
-
-
-
-
50
-
-
0028234484
-
-
Horita K., Sakurai Y., Hachiya S.-I., Nagasawa M., and Yonemitsu O. Chem. Pharm. Bull. 42 (1994) 683-685
-
(1994)
Chem. Pharm. Bull.
, vol.42
, pp. 683-685
-
-
Horita, K.1
Sakurai, Y.2
Hachiya, S.-I.3
Nagasawa, M.4
Yonemitsu, O.5
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