Conservation of functional and pharmacological properties in the distantly related temperature sensors TRVP1 and TRPM8

Molecular Pharmacology

Volumn 68, Issue 2, 2005, Pages 518-527

  Weil, Annette ^a   Moore, Stephen E ^a   Waite, Nicola J ^a   Randall, Andrew ^a   Gunthorpe, Martin J ^a  

^a GLAXOSMITHKLINE   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

4 (3 CHLORO 2 PYRIDINYL) 2 METHYL N [4 (TRIFLUOROMETHYL)PHENYL] 1 PIPERAZINECARBOXAMIDE; ALCOHOL; AMIDE; CAPSAICIN; CAPSAZEPINE; CATION CHANNEL; LIGAND; MENTHOL; N (2 BROMOPHENYL) N' [2 [ETHYL(3 METHYLPHENYL)AMINO]ETHYL]UREA; RECEPTOR; TRANSIENT RECEPTOR POTENTIAL CHANNEL; TRANSIENT RECEPTOR POTENTIAL MELASTATIN 8; UNCLASSIFIED DRUG; UREA DERIVATIVE; VANILLOID RECEPTOR 1;

ACIDIFICATION; ARTICLE; CHANNEL GATING; COLD SENSITIVITY; CONTROLLED STUDY; ELECTRIC POTENTIAL; EMBRYO; HEAT SENSITIVITY; HUMAN; HUMAN CELL; NUCLEOTIDE SEQUENCE; PATCH CLAMP; PRIORITY JOURNAL; PROTEIN FUNCTION; TEMPERATURE; TIME; WHOLE CELL;

CAPSAICIN; CELL LINE; DOSE-RESPONSE RELATIONSHIP, DRUG; HUMANS; ION CHANNELS; NEOPLASM PROTEINS; TEMPERATURE SENSE; TRPM CATION CHANNELS; TRPV CATION CHANNELS;

EID: 23044500197     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.105.012146     Document Type: Article

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