Synthesis of substituted indole derivatives as a new class of antimalarial agents

Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 12, 2005, Pages 3133-3136

  Agarwal, Anu ^a   Srivastava, Kumkum ^a   Puri, S K ^a   Chauhan, Prem M S ^a  

^a CENTRAL DRUG RESEARCH INSTITUTE   (India)

Author keywords

Antimalarial; Dihydrofolate reductase; Pyrimidine

Indexed keywords

INDOLE DERIVATIVE; PYRIMETHAMINE;

ANTIMALARIAL ACTIVITY; ARTICLE; COMPARATIVE STUDY; CONTROLLED STUDY; DRUG SYNTHESIS; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; PLASMODIUM FALCIPARUM; SUBSTITUTION REACTION;

ANIMALS; ANTIMALARIALS; INDOLES; MICROBIAL SENSITIVITY TESTS; PLASMODIUM FALCIPARUM; PYRIMETHAMINE; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 19844379839     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2005.04.011     Document Type: Article

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