Synthesis and antimalarial evaluation of new 1,4-bis(3-aminopropyl)piperazine derivatives

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 21, 2003, Pages 3783-3787

  Ryckebusch, Adina ^a   Deprez Poulain, Rébecca ^a   Debreu Fontaine, Marie Ange ^a   Vandaele, Richard ^a   Mouray, Elisabeth ^b   Grellier, Philippe ^b   Sergheraert, Christian ^a  

^a INSTITUT PASTEUR DE LILLE   (France)

^b MUSÉUM NATIONAL D'HISTOIRE NATURELLE   (France)

Author keywords

[No Author keywords available]

Indexed keywords

ANTIMALARIAL AGENT; BENZOXAZOLE DERIVATIVE; BENZYLAMINE DERIVATIVE; BETA HEMATIN; CHLOROQUINE; PIPERAZINE DERIVATIVE; PROTEIN; PROTEIN SYNTHESIS INHIBITOR; UNCLASSIFIED DRUG;

ANTIMALARIAL ACTIVITY; ARTICLE; ARYLATION; CELL LINE; CONTROLLED STUDY; DRUG POTENCY; DRUG SCREENING; DRUG SELECTIVITY; DRUG SYNTHESIS; EMBRYO; HUMAN; HUMAN CELL; NONHUMAN; PLASMODIUM FALCIPARUM; PREDICTION; STRAIN IDENTIFICATION; STRUCTURE ACTIVITY RELATION; STRUCTURE ANALYSIS;

PLASMODIUM FALCIPARUM;

EID: 0141656369     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2003.07.008     Document Type: Article

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