Synthesis and in vitro and in vivo antimalarial activity of new 4-anilinoquinolines

Journal of Medicinal Chemistry

Volumn 44, Issue 17, 2001, Pages 2827-2833

  Delarue, S ^a   Girault, S ^a   Maes, L ^b   Debreu Fontaine, M A ^a   Labaeid M ^c   Grellier, P ^c   Sergheraert, C ^a  

^a CNRS   (France)

^b MUSÉUM NATIONAL D'HISTOIRE NATURELLE   (France)

^c Virco BVBA   (Belgium)

Author keywords

[No Author keywords available]

Indexed keywords

4 ANILINOQUINOLINE DERIVATIVE; AMODIAQUINE; ANTIMALARIAL AGENT; CHLOROQUINE; MORPHOLINE DERIVATIVE; QUINOLINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIMALARIAL ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG CYTOTOXICITY; DRUG SYNTHESIS; FEMALE; HUMAN; HUMAN CELL; IN VITRO STUDY; IN VIVO STUDY; LUNG ALVEOLUS CELL; MALARIA; MOUSE; NONHUMAN; PARASITEMIA; PERITONEUM MACROPHAGE; PLASMODIUM BERGHEI; PLASMODIUM FALCIPARUM;

ANILINE COMPOUNDS; ANIMALS; ANTIMALARIALS; CELLS, CULTURED; DRUG RESISTANCE; FEMALE; HUMANS; MACROPHAGES, PERITONEAL; MALARIA; MICE; PLASMODIUM BERGHEI; PLASMODIUM FALCIPARUM; QUINOLINES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0035899179     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm010842o     Document Type: Article

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