-
1
-
-
85119808332
-
-
National workshop on operational constrains and their feasible solutions for efficient functions of national filaria control program units in the country. December 1991, NICD, Delhi, India.
-
-
-
-
2
-
-
85119802678
-
-
Ottesen, E. A.; Ramachandran, C. P. Lymphatic filariasis infection and disease: control strategies. Parasitology Today 1995 , 2 , 129–131.
-
-
-
-
3
-
-
85119819254
-
-
Cao, W.; Ploeg, C. P. B.; Ren, Z.; Habbema, J. D. F. Success against lymphatic filariasis. World Health Forum 1997 , 18 , 17–20.
-
-
-
-
4
-
-
85119802475
-
-
Sharma, S. Vector borne diseases. Prog. Drug Res. 1990 , 35 , 365–485.
-
-
-
-
5
-
-
85119790519
-
-
Simonsen, P. E.; Meyrowitsch, D. W.; Makunde, W. H. Bancroftian filariasis: long-term effect of the DEC provocative day tool on microfilaraemia. Transactions of the Royal Society of Tropical Medicine and Hygiene 1997 , 91 , 290–293.
-
-
-
-
6
-
-
85119805366
-
-
Bennett, J. L.; Williams, J. F.; Dave, V. Pharmacology of Ivermectin. Parasitology Today 1988 , 4 , 226–228.
-
-
-
-
7
-
-
85119813152
-
-
Ginger, C. D. Advances in Filarial Chemotherapy and Screening. Parasitology Today 1986 , 2 , 38–40.
-
-
-
-
8
-
-
85119816167
-
-
Loiseau, P. M.; Depreux, P. In vitro antifilarial evaluation of phenoxycyclohexane derivatives. Annals of Tropical Medicine and Parasitology 1993 , 87 , 469–476.
-
-
-
-
9
-
-
85119795459
-
-
Chauhan, P. M. S.; Chatterjee, R. K. Synthesis of 1,3-substituted pyrazoles as possible antifilarial agents. Indian J. Chem. 1994 , 33B , 32–37.
-
-
-
-
10
-
-
85119815569
-
-
Srivastava, S. K.; Chauhan, P. M. S.; Agarwal, S. K.; Bhaduri, A. P.; Singh, S. N.; Fatma, N.; Chatterjee, R. K.; Bose, C.; Srivastava, V. M. L. Syntheses and antifilarial profile of 5-amino and 5,8-diamino isoquinoline derivatives: a new class of antifilarial agents. Bioorg. Med. Chem. Lett. 1996 , 6 , 2623–2628.
-
-
-
-
11
-
-
85119799212
-
-
Singh, S. N.; Bhatnagar, S.; Fatma, N.; Chauhan, P. M. S.; Chatterjee, R. K. Antifilarial activity of a synthetic marine alkaloid, aplysinopsin (CDRI Compound 92/138). Tropical Medicine and International Health 1997 , 2 , 535–543.
-
-
-
-
12
-
-
85119802788
-
-
Tewari, S.; Chauhan, P. M. S.; Bhaduri, A. P.; Singh, S. N.; Fatma, N.; Chatterjee, R. K.; Srivastava, V. M. L. 1,1′-Dicyano-2-substituted ethylenes: A new class of glucose uptake inhibitors in antifilarial chemotherapy. Bioorg. Med. Chem. Lett. 1997 , 7 , 1891–1896.
-
-
-
-
13
-
-
85119789916
-
-
Sharma, S. Design of new drugs for helminth diseases: lead optimization in benzimidozole. Adv. Drug Res. 1994 , 25 , 103–172.
-
-
-
-
14
-
-
85119796820
-
-
Townsend, L. B.; Wise D. S. The synthesis and chemistry of certain anthelmintic benzimidazoles. Parasitology Today 1990 , 6 , 107–112.
-
-
-
-
15
-
-
85119819460
-
-
Agarwal, A.; Agarwal, S. K.; Bhakuni, D. S.; Gupta, S.; Katiyar, J. C. Antiparasitic agents: Part VIII—Synthesis of 1,6- and 1,8-disubstituted-9 H -pyrido[3,4- b ]indoles and 2-substituted-1(3),10-dihydro-9-phenylpyrido[3,4- b ]imidazo[4,5-b]indoles and their anthelmintic activity. Indian J. Chem. 1989 , 28B , 943–949.
-
-
-
-
16
-
-
85119811407
-
-
Agarwal, A.; Agarwal, S. K.; Bhakuni, D. S. Antiparasitic agents: Part X—Synthesis of 2,7-disubstituted-1,6-dihydropyrido[3,4- b ]imidazo[4,5-e]indoles as anthelmintic agents. Indian J. Chem. 1990 , 29B , 843–847.
-
-
-
-
17
-
-
85119791343
-
-
Agarwal, A.; Agarwal, S. K.; Bhakuni, D. S.; Gupta, S.; Katiyar, J. C. Antiparasitic agents: Part XIII—Synthesis and anthelmintic activity of 6- and 8-(2,4-dioxoquinazolin-3-yl)-1-substituted-9 H -pyrido[3,4- b ]indoles, 6- and 8-(2-methyl-5-acetamidobenzimidazol-1-yl)-1-substituted-9 H -pyrido[3,4- b ]indoles and 6-[2-carbomethoxyamino-5- N , N ′-dicarbo-methoxyquanidino)benzimidazol-1-yl]-1-phenyl-9 H -pyrido[3,4- b ]indole. Indian J. Chem. 1990 , 29B , 848–854.
-
-
-
-
18
-
-
85119808318
-
-
Kumar, P.; Agarwal, S. K.; Bhakuni, D. S. Antiparasitic agents: Part XI—Synthesis and anthelmintic activity of 6-/8-[(2-carbomethoxyamino)benzimidazole]-5-carbonylamino-1-substituted-9 H -pyrido[3,4- b ]indoles. Indian J. Chem. 1990 , 29B , 1077–1088.
-
-
-
-
19
-
-
85119793669
-
-
Agarwal, A.; Agarwal, S. K.; Bhakuni, D. S.; Singh, S. N.; Chatterjee, R. K. Antiparasitic agents: Part XVI—Synthesis of 5(6)-substituted benzimidazole-2-carbamates as anthelmintic agents. Indian J. Chem. 1993 , 32B , 453–456.
-
-
-
-
20
-
-
85119812952
-
-
Agarwal, A.; Agarwal, S. K.; Singh, S. N.; Fatma, N.; Murthy, P. K.; Chatterjee, R. K. Synthesis and antifilarial activity of pyrido[3,4- b ]imidazo[1,2-c′]quinazolo[4,5-e]/[4,5-g]indoles. Med. Chem. Res. 1994 , 3 , 523–530.
-
-
-
-
21
-
-
85119799268
-
-
Bose, C.; Agarwal, S. K.; Chatterjee, R. K.; Srivastava, V. M. L. Carboline antifilarials: effects on carbohydrate metabolizing enzymes in Litomosides carinii female. Indian J. Exp. Bio. 1994 , 32 , 431–434.
-
-
-
-
22
-
-
85119811291
-
-
Agarwal, A.; Agarwal, S. K.; Singh S. N.; Fatima N.; Chatterjee, R. K., Structure–antifilarial activity relationship of 5/6/7/8-mono or disubstituted 1H/1-phenyl-9H-pyrdo[3,4- b ]indoles—a new class of potential filaricides. Z. Naturforsch 1994 , 49c , 526–529.
-
-
-
-
23
-
-
85119818481
-
-
Agarwal A; Agarwal S. K. Antiparasitic agents: Part XVII. Synthesis of 2-methylmercapto-7-H/phenyl-1H,6H-pyrido[3,4- b ]imidazo[4,5-e]indoles, 6-/8-(4-oxo-2-thioxoquinazoline-3-yl)-1-H/phenyl-9 H -pyrido[3,4- b ]indoles and 6-/8-(2,4-dioxo-1,3-benzoxazin-3-yl)-1-phenyl-9 H -pyrido[3,4- b ]indoles as anthelmintic agents. Indian J. Chem. 1995 , 34B , 323.
-
-
-
-
24
-
-
85119812586
-
-
Agarwal, A.; Agarwal, S. K.; Singh S. N.; Fatima N.; Chatterjee, R. K. Synthesis of neoeudistomin analogues—As potential filaricides. Bioorg. Med. Chem. Lett. 1995 , 5 , 1545–1548.
-
-
-
-
25
-
-
85119813420
-
-
Moore, E. C.; Zedeck, M. S.; Agarwal, K. C.; Sartorelli, A. C. Inhibition of ribonucleoside diphosphate reductase by 1-formylisoquinoline thiosemicarbazone and related compounds. Biochemistry 1970 , 23 , 4492–4498.
-
-
-
-
26
-
-
85119808639
-
-
Campbell, W. C.; Fisher, M. H.; Stapley, E. O.; Albers-Schonberg, G.; Jacob, T. A. Ivermetin: a potent new antiparasitic agent. Science 1983 , 221 , 823–828.
-
-
-
-
27
-
-
85119794263
-
-
Johnston, G. A. R. In GABA in Nervous System Function ; Roberts, E.; Chase, T. N.; Tower, D. B. Ed.; Raven Press, New York, 1978, 395.
-
-
-
-
28
-
-
85119809666
-
-
Wang, C. C. Parastic enzymes as potential targets for antiparasitic chemotherpay. J. Med. Chem. 1984 , 27 , 1–9.
-
-
-
-
29
-
-
85119809552
-
-
Braestrup, C.; Nielson, M.; Olsen, C. E. Urinary and brain β-carboline-3-carboxylates as potent inhibitors of brain benzodiazopine receptors. Proc. Natl. Acad. Sci. USA 1980 , 77 , 2288–2292.
-
-
-
-
30
-
-
85119805806
-
-
Dodd, H. R.; Ovannes, C.; Robert G.; Potier P. Hybrid molecules: growth inhibition of Leishmania donovani promastigotes by thiosemicarbazones of 3-carboxy-β-carbolines. J. Med. Chem. 1989 , 32 , 1272–1276.
-
-
-
-
31
-
-
85119814253
-
-
Cain, M.; Weber, R. W.; Guzman, F.; Cook, J. M.; Barker, S. A.; Rice, K. C.; Grawley, J. N.; Paul, S. M.; Skolnick, P. β-Carbolines: synthesis and neurochemical and pharmacological actions on brain benzodiazepine receptors. J. Med. Chem. 1982 , 25 , 1081–1091.
-
-
-
-
32
-
-
85119817026
-
-
Agarwal, S. K.; Saxena, A. K.; Jain, P. C. Studies on β-carbolines: synthesis of 3-amino-9 H -pyrido[3,4- b ]indoles and its reaction with carbethoxy isothiocyanate and benzoyl isothiocyanate. Indian J. Chem. 1980 , 19B , 45–47.
-
-
-
-
33
-
-
85119799596
-
-
Meyer, M. D.; Kruse, L. I. Ergoline synthons: synthesis of 3,4-dihydro-6-methoxy-benz[cd]indol-5-(1H)-one(6-methoxy-uhle's ketone) and 3,4-dihydrobenz[cd]indol-5(1H)-one(uhle's ketone) via a novel decarboxylation of indole-2-carboxylates. J. Org. Chem. 1984 , 49 , 3195–3199.
-
-
-
-
34
-
-
85119793923
-
-
Hicknbottom, W. J., Reaction of Organic Compounds . Longmans, London, 1959.
-
-
-
-
35
-
-
85119802819
-
-
Kumar, S.; Seth M.; Bhaduri, A. P.; Visen, P. K. S.; Mishra, A.; Gupta S.; Fatima, N.; Katiyar, J. C.; Chatterjee, R. K.; Sen A. B. Syntheses and anthelmintic activity of alkyl 5(6)-(substituted-carbamoyl)- and 5(6)-(disubstituted-carbamoyl)benzimidazole-2-carbamates and related compounds. J. Med. Chem. 1984 , 27 , 1083–1089.
-
-
-
-
36
-
-
85119790850
-
-
Murthy, P. K.; Tyagi, K.; Roy Chowdhury, T. K.; Sen, A. B. Susceptibility of Mastomys natalensis (GRA strain) to a subperiodic strain of human Brugia malayai . Indian J. Med. Res. 1983 , 77 , 623–630.
-
-
-
-
37
-
-
85119812699
-
-
World Health Organisation. Report of the Seventh meeting of the Scientific Working Group on Filariasis: Filaricide screeners. TDR/Fil/SWG(7)82,3 Geneva: World Health Organisation, 1982.
-
-
-
-
38
-
-
85119815975
-
-
Hewitt, R. I.; Kushner, S., Stewart, H., White, E., Wallace, W. S. Subbarow; Y., Experimental chemotherapy of filariasis III. Effect of 1-diethylcarbanyl 4-methylpiperazine hydrochloride against naturally acquired filarial infection in cotton rats and dogs. J. Lab. Clin. Medicine 1947 , 32 , 1314–1329.
-
-
-
-
39
-
-
85119803292
-
-
Worms, M. J.; Terry, R. J.; Terry, A. Dipetalonema witei , filarial parasites of the jird, Meriones libycus , 1. Maintenance in the laboratory. J. Parasit. 1961 , 47 , 963–970.
-
-
-
-
40
-
-
85119790176
-
-
Lammler, G.; Herzog, H.; Saupe E.; Schuetze, H. R. Chemotherapeutic studies on Litomosoides carinii infection of Mastomys natalensis . Bull. Wld. Hlth. Org. 1971 , 44 , 751–756.
-
-
-
-
41
-
-
85119807584
-
-
Misra, S.; Chatterjee, R. K.; Sen, A. B. Antifilarial action of furazolidone. Indian J. Med. Res. 1981 , 73 , 725–728.
-
-
-
-
42
-
-
85119788192
-
-
Howking, F.; Sewell, P. The maintenance of filarial infection ( Litomosoides carinii ) for chemotherapeutic investigations. Br. J. Pharm. Chem. 1948 , 3 , 285.
-
-
-
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