Benzimidazolone p38 inhibitors

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 4, 2004, Pages 919-923

  Dombroski, Mark A ^a   Letavic, Michael A ^a,b   McClure, Kim F ^a   Barberia, John T ^a   Carty, Thomas J ^a   Cortina, Santo R ^a   Csiki, Csilla ^a   Dipesa, Alan J ^a   Elliott, Nancy C ^a   Gabel, Christopher A ^a   Jordan, Crystal K ^a   Labasi, Jeff M ^a   Martin, William H ^a   Peese, Kevin M ^a   Stock, Ingrid A ^a   Svensson, Linne ^a   Sweeney, Francis J ^a   Yu, Chul H ^a  

^a PFIZER GLOBAL RESEARCH AND DEVELOPMENT   (United States)

^b JOHNSON AND JOHNSON PHARMACEUTICAL RESEARCH AND DEVELOPMENT   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BENZIMIDAZOLE DERIVATIVE; ISOENZYME; MITOGEN ACTIVATED PROTEIN KINASE 14; MITOGEN ACTIVATED PROTEIN KINASE INHIBITOR; MITOGEN ACTIVATED PROTEIN KINASE P38; MITOGEN ACTIVATED PROTEIN KINASE P38 INHIBITOR; UNCLASSIFIED DRUG;

AMINO ACID SEQUENCE; ARTICLE; DRUG ACTIVITY; DRUG BINDING; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME ACTIVITY; HYDROGEN BOND; IN VITRO STUDY; STRUCTURE ACTIVITY RELATION;

EID: 10744219681     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2003.12.023     Document Type: Article

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