The use of receptor G-protein fusion proteins for the study of ligand activity

Receptors and Channels

Volumn 8, Issue 5-6, 2002, Pages 309-317

  Milligan, Graeme ^a  

^a UNIVERSITY OF GLASGOW   (United Kingdom)

Author keywords

Agonist; G protein; Inverse agonist; Palmitoylation; Receptor

Indexed keywords

G PROTEIN COUPLED RECEPTOR; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANOSINE TRIPHOSPHATASE; HYBRID PROTEIN; LIGAND; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); PALMITIC ACID DERIVATIVE;

ACYLATION; ALPHA CHAIN; AMINO TERMINAL SEQUENCE; CARBOXY TERMINAL SEQUENCE; ENZYME ACTIVATION; LIGAND BINDING; MUTATION; PRIORITY JOURNAL; PROTEIN FUNCTION; PROTEIN PROCESSING; PROTEIN PROTEIN INTERACTION; QUANTITATIVE ANALYSIS; REGULATORY MECHANISM; REVIEW; SIGNAL TRANSDUCTION; ANIMAL; CELL STRAIN COS1; CHEMISTRY; DOSE RESPONSE; GENETIC POLYMORPHISM; HUMAN; KINETICS; METABOLISM; PROTEIN BINDING; PROTEIN TERTIARY STRUCTURE;

ANIMALS; COS CELLS; DOSE-RESPONSE RELATIONSHIP, DRUG; GTP-BINDING PROTEINS; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); HUMANS; KINETICS; LIGANDS; MUTATION; PALMITIC ACIDS; POLYMORPHISM, GENETIC; PROTEIN BINDING; PROTEIN STRUCTURE, TERTIARY; RECOMBINANT FUSION PROTEINS; SIGNAL TRANSDUCTION;

EID: 0036450783     PISSN: 10606823     EISSN: None     Source Type: Journal    
DOI: 10.1080/10606820214639     Document Type: Review

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