Agonist efficacy at the α(2A)-adrenoceptor:G(α15) fusion protein: An analysis based on Ca2+ responses

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 361, Issue 6, 2000, Pages 672-679

  Pauwels, P J ^a   Finana, F ^a   Tardif, S ^a   Colpaert, F C ^a   Wurch, T ^a  

^a INSTITUT DE RECHERCHE PIERRE FABRE   (France)

Author keywords

Ca2+ response; Fusion protein; Ligand efficacy; Recombinant (2A) AR and G( 15) protein

Indexed keywords

2 (2 METHOXY 1,4 BENZODIOXAN 2 YL) 2 IMIDAZOLINE; ADRENALIN; ALPHA 2 ADRENERGIC RECEPTOR STIMULATING AGENT; BRIMONIDINE; CLONIDINE; HYBRID PROTEIN; MEDETOMIDINE; OXYMETAZOLINE; TALIPEXOLE; 2-METHOXYIDAZOXAN; ALPHA 2 ADRENERGIC RECEPTOR; ALPHA ADRENERGIC RECEPTOR STIMULATING AGENT; CALCIUM; DRUG DERIVATIVE; FLUORESCENT DYE; GUANINE NUCLEOTIDE BINDING PROTEIN; IDAZOXAN; LIGAND; QUINOXALINE DERIVATIVE; RECEPTOR, ADRENERGIC, ALPHA 2A; RECEPTOR, ADRENERGIC, ALPHA-2A;

ANIMAL CELL; ARTICLE; CALCIUM MOBILIZATION; CHO CELL; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; HUMAN; LIGAND BINDING; MOLECULAR DYNAMICS; MOUSE; NONHUMAN; NUCLEOTIDE SEQUENCE; ANIMAL; GENETIC TRANSFECTION; GENETICS; HAMSTER; METABOLISM; RADIOASSAY; SIGNAL TRANSDUCTION;

ADRENERGIC ALPHA-AGONISTS; ANIMALS; CALCIUM; CHO CELLS; CRICETINAE; EPINEPHRINE; FLUORESCENT DYES; GTP-BINDING PROTEINS; HUMANS; IDAZOXAN; LIGANDS; MICE; QUINOXALINES; RADIOLIGAND ASSAY; RECEPTORS, ADRENERGIC, ALPHA-2; RECOMBINANT FUSION PROTEINS; SIGNAL TRANSDUCTION; TRANSFECTION;

EID: 0033623847     PISSN: 00281298     EISSN: None     Source Type: Journal    
DOI: 10.1007/s002100000250     Document Type: Article

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