SCOPUS 정보 검색 플랫폼

Volumn 9, Issue 5, 2002, Pages 359-364

Structural characterization of a subtype-selective ligand reveals a novel mode of estrogen receptor antagonism

(9) Shiau, Andrew K a Barstad, Danielle a Radek, James T a Meyers, Marvin J a Nettles, Kendall W a Katzenellenbogen, Benita S a Katzenellenbogen, John A a Agard, David A a Greene, Geoffrey L a

a HOWARD HUGHES MEDICAL INSTITUTE (United States)

Author keywords

[No Author keywords available]

Indexed keywords

5,11 DIETHYL 5,6,11,12 TETRAHYDROCHRYSENE 2,8 DIOL; ANTIESTROGEN; ESTROGEN RECEPTOR; ESTROGEN RECEPTOR ALPHA; ESTROGEN RECEPTOR BETA; HORMONE RECEPTOR AFFECTING AGENT; LIGAND; RECEPTOR SUBTYPE; TRANSCRIPTION FACTOR; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL STRUCTURE; LIGAND BINDING; PRIORITY JOURNAL; PROTEIN CONFORMATION; PROTEIN DOMAIN; PROTEIN STABILITY; PROTEIN STRUCTURE; RECEPTOR BINDING; RECEPTOR BLOCKING;

BINDING SITES; CHRYSENES; CRYSTALLOGRAPHY, X-RAY; ESTROGEN RECEPTOR ALPHA; ESTROGEN RECEPTOR BETA; HUMANS; LIGANDS; MODELS, MOLECULAR; NUCLEAR RECEPTOR COACTIVATOR 2; PEPTIDE FRAGMENTS; PROTEIN STRUCTURE, TERTIARY; RECEPTORS, ESTROGEN; STRUCTURE-ACTIVITY RELATIONSHIP; SUBSTRATE SPECIFICITY; TRANSCRIPTION FACTORS;

EID: 0036234964 PISSN: 10728368 EISSN: None Source Type: Journal
DOI: 10.1038/nsb787 Document Type: Article

Times cited : (359)

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