메뉴 건너뛰기




Volumn 54, Issue 1, 1998, Pages 105-112

Differential response of estrogen receptor α and estrogen receptor β to partial estrogen agonists/antagonists

Author keywords

[No Author keywords available]

Indexed keywords

ESTRADIOL; ESTROGEN RECEPTOR; N BUTYL 11 (3,17BETA DIHYDROXYESTRA 1,3,5(10) TRIEN 7ALPHA YL) N METHYLUNDECANAMIDE; RALOXIFENE; TAMOXIFEN;

EID: 0031816540     PISSN: 0026895X     EISSN: None     Source Type: Journal    
DOI: 10.1124/mol.54.1.105     Document Type: Article
Times cited : (741)

References (39)
  • 3
    • 0024545638 scopus 로고
    • Gene regulation by steroid hormones
    • Beato M (1989) Gene regulation by steroid hormones. Cell 56:335-344.
    • (1989) Cell , vol.56 , pp. 335-344
    • Beato, M.1
  • 4
    • 0027521287 scopus 로고
    • Transcriptional activation by the estrogen receptor requires a conformational change in the ligand binding domain
    • Beekman JM, Allan GF, Tsai SY, Tsai M-J, and O'Malley BW (1993) Transcriptional activation by the estrogen receptor requires a conformational change in the ligand binding domain. Mol Endocrinol 7:1266-1274.
    • (1993) Mol Endocrinol , vol.7 , pp. 1266-1274
    • Beekman, J.M.1    Allan, G.F.2    Tsai, S.Y.3    Tsai, M.-J.4    O'Malley, B.W.5
  • 5
    • 0029745382 scopus 로고    scopus 로고
    • Thiazolidinediones produce a conformational change in peroxisomal proliferator-actvated receptor-γ: Binding and activation correlate with antidiabetic actions in db/db mice
    • Berger J, Bailey P, Biswas C, Cullinan CA, Doebber TW, Hayes NS, Saperstein R, Smith RG, and Leibowitz MD (1996) Thiazolidinediones produce a conformational change in peroxisomal proliferator-actvated receptor-γ: binding and activation correlate with antidiabetic actions in db/db mice. Endocrinology 137:4189-4195.
    • (1996) Endocrinology , vol.137 , pp. 4189-4195
    • Berger, J.1    Bailey, P.2    Biswas, C.3    Cullinan, C.A.4    Doebber, T.W.5    Hayes, N.S.6    Saperstein, R.7    Smith, R.G.8    Leibowitz, M.D.9
  • 6
    • 0023932371 scopus 로고
    • Secreted placental alkaline phosphatase: A powerful new quantitative indicator of gene expression in eukaryotic cells
    • Berger J, Hauber J, Hauber R, Geiger R, and Cullen BR (1988) Secreted placental alkaline phosphatase: a powerful new quantitative indicator of gene expression in eukaryotic cells. Gene 66:1-10.
    • (1988) Gene , vol.66 , pp. 1-10
    • Berger, J.1    Hauber, J.2    Hauber, R.3    Geiger, R.4    Cullen, B.R.5
  • 8
    • 0025362718 scopus 로고
    • Nuclear factor I acts as a transcription factor on the MMTV promoter but competes with steroid hormone receptors for DNA binding
    • Brüggemeier U, Rogge L, Winnacker E-L, and Beato M (1990) Nuclear factor I acts as a transcription factor on the MMTV promoter but competes with steroid hormone receptors for DNA binding. EMBO J 9:2233-2239.
    • (1990) EMBO J , vol.9 , pp. 2233-2239
    • Brüggemeier, U.1    Rogge, L.2    Winnacker, E.-L.3    Beato, M.4
  • 10
    • 0023913120 scopus 로고
    • The steroid and thyroid hormone receptor superfamily
    • Evans RM (1988) The steroid and thyroid hormone receptor superfamily. Science (Washington DC) 240:889-895.
    • (1988) Science (Washington DC) , vol.240 , pp. 889-895
    • Evans, R.M.1
  • 12
    • 0025084510 scopus 로고
    • Inhibition of estrogen receptor-DNA binding by the 'pure' antiestrogen ICI 164,384 appears to be mediated by impaired receptor dimerization
    • Fawell SE, White R, Hoare S, Sydenham M, Page M, and Parker MG (1990) Inhibition of estrogen receptor-DNA binding by the 'pure' antiestrogen ICI 164,384 appears to be mediated by impaired receptor dimerization. Proc Natl Acad Sci USA 87:6883-6887.
    • (1990) Proc Natl Acad Sci USA , vol.87 , pp. 6883-6887
    • Fawell, S.E.1    White, R.2    Hoare, S.3    Sydenham, M.4    Page, M.5    Parker, M.G.6
  • 14
    • 0023797380 scopus 로고
    • Nuclear receptors enhance our understanding of transcription regulation
    • Green S and Chambon P (1988) Nuclear receptors enhance our understanding of transcription regulation. Trends Genet 4:309-314.
    • (1988) Trends Genet , vol.4 , pp. 309-314
    • Green, S.1    Chambon, P.2
  • 17
    • 0021078994 scopus 로고
    • Plasmid-encoded hygromycin B resistance: The sequence of hygromycin B phosphotransferase gene and its expression in Escherichia coli and Saccharomyces cerevisiae
    • Gritz L and Davies J (1983) Plasmid-encoded hygromycin B resistance: the sequence of hygromycin B phosphotransferase gene and its expression in Escherichia coli and Saccharomyces cerevisiae. Gene 25:179-188.
    • (1983) Gene , vol.25 , pp. 179-188
    • Gritz, L.1    Davies, J.2
  • 18
    • 0026754249 scopus 로고
    • Control of transcription activation by steroid hormone receptors
    • Gronemeyer H (1992) Control of transcription activation by steroid hormone receptors. FASEB J 6:2524-2529.
    • (1992) FASEB J , vol.6 , pp. 2524-2529
    • Gronemeyer, H.1
  • 19
    • 0029440036 scopus 로고
    • Transcription factors 3: Nuclear receptors
    • Gronemeyer H and Laudet V (1995) Transcription factors 3: nuclear receptors. Protein Profile 2:1167-1322.
    • (1995) Protein Profile , vol.2 , pp. 1167-1322
    • Gronemeyer, H.1    Laudet, V.2
  • 20
    • 0343562790 scopus 로고
    • Hormones and hormone antagonists
    • Goodman-Gilman A, Rall TW, Nies AS, and Taylor P, eds, Pergamon Press, New York
    • Haynes RC, Murad F, Kuret JA, and Wilson JD (1990) Hormones and hormone antagonists, in The Pharmacological Basis of Therapeutics (Goodman-Gilman A, Rall TW, Nies AS, and Taylor P, eds) pp 1332, 1361-1462, 1510-1522, Pergamon Press, New York.
    • (1990) The Pharmacological Basis of Therapeutics , pp. 1332
    • Haynes, R.C.1    Murad, F.2    Kuret, J.A.3    Wilson, J.D.4
  • 22
    • 0021201213 scopus 로고
    • Antiestrogens. 2. Structure-activity studies in a series of 3-aroyl-2-arylbenzo[b]thiophene derivatives leading to [6-hydroxy-2-(4- hydroxyphenyl)benzo[b]thien-3-yl][4-[2-(1-piperidinyl)ethoxy]-phenyl]methanone hydrochloride (LY156758), a remarkably effective estrogen antagonist with only minimal intrinsic estrogenicity
    • Jones CD, Jevnikar MG, Pike AJ, Peters MK, Black LJ, Thompson AR, Falcone JF, and Clemens JA (1984) Antiestrogens. 2. Structure-activity studies in a series of 3-aroyl-2-arylbenzo[b]thiophene derivatives leading to [6-hydroxy-2-(4-hydroxyphenyl)benzo[b]thien-3-yl][4-[2-(1-piperidinyl)ethoxy]- phenyl]methanone hydrochloride (LY156758), a remarkably effective estrogen antagonist with only minimal intrinsic estrogenicity. J Med Chem 27:1057-1066.
    • (1984) J Med Chem , vol.27 , pp. 1057-1066
    • Jones, C.D.1    Jevnikar, M.G.2    Pike, A.J.3    Peters, M.K.4    Black, L.J.5    Thompson, A.R.6    Falcone, J.F.7    Clemens, J.A.8
  • 23
    • 0030071445 scopus 로고    scopus 로고
    • Tripartite steroid hormone receptor pharmacology: Interaction with multiple effector sites as a basis for the cell- and promoter-specific action of these hormones
    • Katzenellenbogen J, O'Malley BW, and Katzenellenbogen BS (1996) Tripartite steroid hormone receptor pharmacology: interaction with multiple effector sites as a basis for the cell- and promoter-specific action of these hormones. Mol Endocrinol 10:119-131.
    • (1996) Mol Endocrinol , vol.10 , pp. 119-131
    • Katzenellenbogen, J.1    O'Malley, B.W.2    Katzenellenbogen, B.S.3
  • 24
    • 0023034983 scopus 로고
    • An estrogen-responsive element derived from the 5′ flanking region of the xenopus vitellogenin A2 gene functions in transfected human cells
    • Klein-Hitpaß L, Schorrp M, Wagner U, and Ryffel GU (1986) An estrogen-responsive element derived from the 5′ flanking region of the xenopus vitellogenin A2 gene functions in transfected human cells. Cell 46:1053-1061.
    • (1986) Cell , vol.46 , pp. 1053-1061
    • Klein-Hitpaß, L.1    Schorrp, M.2    Wagner, U.3    Ryffel, G.U.4
  • 27
    • 0029016829 scopus 로고
    • An antidiabetic thiazolidinedione is a high affinity ligand for peroxisome proliferator-activated receptor γ (PPARγ)
    • Lehman JM, Moore LB, Smith-Oliver TA, Wilkinson WO, Willson TM, and Kliewer SA (1995) An antidiabetic thiazolidinedione is a high affinity ligand for peroxisome proliferator-activated receptor γ (PPARγ). J Biol Chem 270:12953-12956.
    • (1995) J Biol Chem , vol.270 , pp. 12953-12956
    • Lehman, J.M.1    Moore, L.B.2    Smith-Oliver, T.A.3    Wilkinson, W.O.4    Willson, T.M.5    Kliewer, S.A.6
  • 28
    • 0029683157 scopus 로고    scopus 로고
    • Perimenopausal and postmenopausal hormone replacement therapy. Part 1. An update of the literature on benefits and risks
    • Lichtman J (1996) Perimenopausal and postmenopausal hormone replacement therapy. Part 1. An update of the literature on benefits and risks. J Nurse Midwifery 41:3-28.
    • (1996) J Nurse Midwifery , vol.41 , pp. 3-28
    • Lichtman, J.1
  • 29
    • 0024525110 scopus 로고
    • High level expression of nonfused foreign genes with Autographa californica nuclear polyhedrosis virus expression vectors
    • Luckow VA and Summers MD (1989) High level expression of nonfused foreign genes with Autographa californica nuclear polyhedrosis virus expression vectors. Virology 170:31-39.
    • (1989) Virology , vol.170 , pp. 31-39
    • Luckow, V.A.1    Summers, M.D.2
  • 30
    • 0029038986 scopus 로고
    • Analysis of estrogen receptor function in vitro reveals three distinct classes of antiestrogens
    • McDonnell DP, Clemm DL, Hermann T, Goldman ME, and Pike JW (1995) Analysis of estrogen receptor function in vitro reveals three distinct classes of antiestrogens. Mol Endocrinol 9:659-669.
    • (1995) Mol Endocrinol , vol.9 , pp. 659-669
    • McDonnell, D.P.1    Clemm, D.L.2    Hermann, T.3    Goldman, M.E.4    Pike, J.W.5
  • 31
    • 0029796605 scopus 로고    scopus 로고
    • Different regions in activation function-1 of the human estrogen receptor required for antiestrogen- and estradiol-dependent transcription activation
    • McInerney EM and Katzenellenbogen BS (1996) Different regions in activation function-1 of the human estrogen receptor required for antiestrogen- and estradiol-dependent transcription activation. J Biol Chem 271:24172-24178.
    • (1996) J Biol Chem , vol.271 , pp. 24172-24178
    • McInerney, E.M.1    Katzenellenbogen, B.S.2
  • 32
    • 0030593681 scopus 로고    scopus 로고
    • ERβ: Identification and characterization of a novel human estrogen receptor
    • Mosselman S, Polman J, and Dijkema R (1996) ERβ: identification and characterization of a novel human estrogen receptor. FEBS Lett 392:49-53.
    • (1996) FEBS Lett , vol.392 , pp. 49-53
    • Mosselman, S.1    Polman, J.2    Dijkema, R.3
  • 33
    • 0343126830 scopus 로고
    • The use of engineered cells for evaluation of the activity of small organic compounds interacting with the human glucocorticoid receptor
    • Görög S, ed, Akadémiai Kiadó, Budapest, Hungary
    • Nilsson S, Alksnis M, and Ahola H (1993) The use of engineered cells for evaluation of the activity of small organic compounds interacting with the human glucocorticoid receptor, in Proceedings of the 5th Symposium on the Analysis of Steroids (Görög S, ed) pp 57-67, Akadémiai Kiadó, Budapest, Hungary.
    • (1993) Proceedings of the 5th Symposium on the Analysis of Steroids , pp. 57-67
    • Nilsson, S.1    Alksnis, M.2    Ahola, H.3
  • 34
    • 0028146830 scopus 로고
    • Equilibrium hormone binding to human estrogen receptor in highly diluted cell extracts is non-cooperative and has a Kd of approximately 10 pM
    • Salomonsson M, Carlsson B, and Haggblad J (1994) Equilibrium hormone binding to human estrogen receptor in highly diluted cell extracts is non-cooperative and has a Kd of approximately 10 pM. J Steroid Biochem Moc Biol 50:313-318.
    • (1994) J Steroid Biochem Moc Biol , vol.50 , pp. 313-318
    • Salomonsson, M.1    Carlsson, B.2    Haggblad, J.3
  • 36
    • 0019989719 scopus 로고
    • Transformation of mammalian cells to antibiotic resistance with a bacterial gene under control of the SV40 early region promoter
    • Southern PJ and Berg P (1982) Transformation of mammalian cells to antibiotic resistance with a bacterial gene under control of the SV40 early region promoter. J Mol Appl Genet 1:327-341.
    • (1982) J Mol Appl Genet , vol.1 , pp. 327-341
    • Southern, P.J.1    Berg, P.2
  • 38
    • 0028283503 scopus 로고
    • Molecular mechanisms of action of steroid/thyroid receptor superfamily members
    • Tsai MJ and O'Malley BW (1994) Molecular mechanisms of action of steroid/thyroid receptor superfamily members. Annu Rev Biochem 63:451-486.
    • (1994) Annu Rev Biochem , vol.63 , pp. 451-486
    • Tsai, M.J.1    O'Malley, B.W.2
  • 39
    • 0024337858 scopus 로고
    • Determinants of target gene specificity for steroid/thyroid hormone receptors
    • Umesono K and Evans RM (1989) Determinants of target gene specificity for steroid/thyroid hormone receptors. Cell 57:1139-1146.
    • (1989) Cell , vol.57 , pp. 1139-1146
    • Umesono, K.1    Evans, R.M.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.