-
1
-
-
0030031782
-
Estrogen receptors: Bioactivities and interactions with cell signaling pathways
-
Katzenellenbogen, B. S. Estrogen Receptors: Bioactivities and Interactions with Cell Signaling Pathways. Biol. Reprod. 1996, 54, 287-293.
-
(1996)
Biol. Reprod.
, vol.54
, pp. 287-293
-
-
Katzenellenbogen, B.S.1
-
2
-
-
0030071445
-
Tripartite steroid hormone receptor pharmacology: Interaction with multiple effector sites as a basis for the cell- and promoter-specific action of these hormones
-
Katzenellenbogen, J. A.; O'Malley, B. W.; Katzenellenbogen, B. S. Tripartite Steroid Hormone Receptor Pharmacology: Interaction with Multiple Effector Sites as a Basis for the Cell- and Promoter-Specific Action of These Hormones. Mol. Endocrinol. 1996, 10, 119-131.
-
(1996)
Mol. Endocrinol.
, vol.10
, pp. 119-131
-
-
Katzenellenbogen, J.A.1
O'Malley, B.W.2
Katzenellenbogen, B.S.3
-
3
-
-
0030593681
-
ERβ: Identification and characterization of a novel human estrogen receptor
-
Mosselman, S.; Polman, J.; Dijkema, R. ERβ: Identification and Characterization of a Novel Human Estrogen Receptor. FEBS Lett. 1996, 392, 49-53.
-
(1996)
FEBS Lett.
, vol.392
, pp. 49-53
-
-
Mosselman, S.1
Polman, J.2
Dijkema, R.3
-
4
-
-
0030579801
-
Cloning of a novel estrogen receptor ex-pressed in rat prostate and ovary
-
Kuiper, G. G. J. M.; Enmark, E.; Pelto-Huikko, M.; Nilsson, S.; Gustafsson, J.-Å. Cloning of a Novel Estrogen Receptor Ex-pressed in Rat Prostate and Ovary. Proc. Natl. Acad. Sci. U.S.A. 1996, 93, 5925-5930.
-
(1996)
Proc. Natl. Acad. Sci. U.S.A
, vol.93
, pp. 5925-5930
-
-
Kuiper, G.G.J.M.1
Enmark, E.2
Pelto-Huikko, M.3
Nilsson, S.4
Gustafsson, J.-Å.5
-
5
-
-
0031039888
-
Comparison of the ligand binding specificity and transcript tissue distribution of estrogen receptors α and β
-
Kuiper, G. G. J. M.; Carlsson, B.; Grandien, K.; Enmark, E.; Häggblad, J.; Nilsson, S.; Gustafsson, J.-Å. Comparison of the Ligand Binding Specificity and Transcript Tissue Distribution of Estrogen Receptors α and β. Endocrinology 1997, 138, 863-870.
-
(1997)
Endocrinology
, vol.138
, pp. 863-870
-
-
Kuiper, G.G.J.M.1
Carlsson, B.2
Grandien, K.3
Enmark, E.4
Häggblad, J.5
Nilsson, S.6
Gustafsson, J.-Å.7
-
6
-
-
0030824020
-
Expression of oestrogen receptor beta (ERβ) in multiple rat tissues visualised by immunohistochemistry
-
Saunders, P. T. K.; Maguire, S. M.; Gaughan, J.; Millar, M. R. Expression of Oestrogen Receptor Beta (ERβ) in Multiple Rat Tissues Visualised by Immunohistochemistry. J. Endocrinol. 1997, 154, R13-R16.
-
(1997)
J. Endocrinol.
, vol.154
-
-
Saunders, P.T.K.1
Maguire, S.M.2
Gaughan, J.3
Millar, M.R.4
-
7
-
-
0031943993
-
Coronary artery and cultured aortic smooth muscle cells express mRNA for both the classical estrogen receptor and the newly described estrogen receptor beta
-
Register, T. C.; Adams, M. R. Coronary Artery and Cultured Aortic Smooth Muscle Cells Express mRNA for Both the Classical Estrogen Receptor and the Newly Described Estrogen Receptor Beta. J. Steroid Biochem. Mol. Biol. 1998, 64, 187-191.
-
(1998)
J. Steroid Biochem. Mol. Biol.
, vol.64
, pp. 187-191
-
-
Register, T.C.1
Adams, M.R.2
-
8
-
-
0030801841
-
Differential ligand activation of estrogen receptors ERa and ERβ at API sites
-
Paech, K.; Webb, P.; Kuiper, G. G. J. M.; Nilsson, S.; Gustafsson, J.-Å.; Kushner, P. J.; Scanlan, T. S. Differential Ligand Activation of Estrogen Receptors ERa and ERβ at API Sites. Science 1997, 277, 1508-1510.
-
(1997)
Science
, vol.277
, pp. 1508-1510
-
-
Paech, K.1
Webb, P.2
Kuiper, G.G.J.M.3
Nilsson, S.4
Gustafsson, J.-Å.5
Kushner, P.J.6
Scanlan, T.S.7
-
9
-
-
0032566547
-
Transcriptional regulation of the human quinone reductase gene by antiestrogen-liganded estrogen receptor-α and estrogen receptor-β
-
Montano, M. M.; Jaiswal, A. K.; Kaztenellenbogen, B. S. Transcriptional Regulation of the Human Quinone Reductase Gene by Antiestrogen-Liganded Estrogen Receptor-α and Estrogen Receptor-β. J. Biol. Chem. 1998, 273, 25443-25449.
-
(1998)
J. Biol. Chem.
, vol.273
, pp. 25443-25449
-
-
Montano, M.M.1
Jaiswal, A.K.2
Kaztenellenbogen, B.S.3
-
10
-
-
0031816540
-
Differential response of estrogen receptor α and estrogen receptor β to partial estrogen Agonists/Antagonists
-
Barkhem, T.; Carlsson, B.; Nilsson, Y.; Enmark, E.; Gustafsson, J.-Å.; Nilsson, S. Differential Response of Estrogen Receptor α and Estrogen Receptor β to Partial Estrogen Agonists/Antagonists. Mol. Pharmacol. 1998, 54, 105-112.
-
(1998)
Mol. Pharmacol.
, vol.54
, pp. 105-112
-
-
Barkhem, T.1
Carlsson, B.2
Nilsson, Y.3
Enmark, E.4
Gustafsson, J.-Å.5
Nilsson, S.6
-
11
-
-
0004752110
-
Novel ligands that function as selective estrogens or antiestrogens for estrogen receptor-a or estrogen receptor-β
-
Sun, J.; Meyers, M. J.; Fink, B. E.; Rajendran, R.; Katzenellenbogen, J. A.; Katzenellenbogen, B. S. Novel Ligands that Function as Selective Estrogens or Antiestrogens for Estrogen Receptor-a or Estrogen Receptor-β. Endocrinology 1999, 140, 800-804.
-
(1999)
Endocrinology
, vol.140
, pp. 800-804
-
-
Sun, J.1
Meyers, M.J.2
Fink, B.E.3
Rajendran, R.4
Katzenellenbogen, J.A.5
Katzenellenbogen, B.S.6
-
12
-
-
0018718637
-
The structure and function of oestrogens. I. Synthesis of 4b-Methyl-trans-4b,5,6,10b,11,12-hexahydrochrysene-2,8-diol
-
Collins, D. J.; Matthews, W. A. The Structure and Function of Oestrogens. I. Synthesis of 4b-Methyl-trans-4b,5,6,10b,11,12-hexahydrochrysene-2,8-diol. Aust. J. Chem. 1979, 32, 1093-1106.
-
(1979)
Aust. J. Chem.
, vol.32
, pp. 1093-1106
-
-
Collins, D.J.1
Matthews, W.A.2
-
13
-
-
0026590257
-
5,6,11,12-Tetrahydrochrysenes: Synthesis of rigid stilbene systems designed to be fluorescent ligands for the estrogen receptor
-
Hwang, K.-J.; O'Neil, J. P.; Katzenellenbogen, J. A. 5,6,11,12-Tetrahydrochrysenes: Synthesis of Rigid Stilbene Systems Designed To Be Fluorescent Ligands for the Estrogen Receptor. J. Org. Chem. 1992, 57, 1262-1271.
-
(1992)
J. Org. Chem.
, vol.57
, pp. 1262-1271
-
-
Hwang, K.-J.1
O'Neil, J.P.2
Katzenellenbogen, J.A.3
-
14
-
-
0030810476
-
Pseudoephedrine as a practical chiral auxiliary for the synthesis of highly enantiomerically enriched carboxylic acids, alcohols, aldehydes, and ketones
-
Myers, A. G.; Yang, B. H.; Chen, H.; McKinstry, L.; Kopecky, D. J.; Gleason, J. L. Pseudoephedrine as a Practical Chiral Auxiliary for the Synthesis of Highly Enantiomerically Enriched Carboxylic Acids, Alcohols, Aldehydes, and Ketones. J. Am. Chem. Soc. 1997, 119, 6496-6511.
-
(1997)
J. Am. Chem. Soc.
, vol.119
, pp. 6496-6511
-
-
Myers, A.G.1
Yang, B.H.2
Chen, H.3
McKinstry, L.4
Kopecky, D.J.5
Gleason, J.L.6
-
15
-
-
85065179340
-
Die unsetzung von carbonsäureestern mit natrium in gegenwart von trimethylchlorsilan
-
Rühlmann, K. Die Unsetzung von Carbonsäureestern mit Natrium in Gegenwart von Trimethylchlorsilan. Synthesis 1971, 236-253.
-
(1971)
Synthesis
, pp. 236-253
-
-
Rühlmann, K.1
-
16
-
-
0030663411
-
7-α,11-β-disubstituted estrogens: Probes for the shape of the ligand binding pocket in the estrogen receptor
-
Tedesco, R.; Katzenellenbogen, J. A.; Napolitano, E. 7-α,11-β-Disubstituted Estrogens: Probes for the Shape of the Ligand Binding Pocket in the Estrogen Receptor. Bioorg. Med. Chem. Lett. 1997, 7, 2919-2924.
-
(1997)
Bioorg. Med. Chem. Lett.
, vol.7
, pp. 2919-2924
-
-
Tedesco, R.1
Katzenellenbogen, J.A.2
Napolitano, E.3
-
17
-
-
85078007309
-
Uber die präparative nutzung der 1,3-thiazoliumsalz-katalysierten acyloin - Und benzoin-bildung; IV. Herstellung von acyloinen mit funktionellen gruppen
-
Stetter, H.; Rämsch, R. Y. Uber die präparative Nutzung der 1,3-Thiazoliumsalz-Katalysierten Acyloin - und Benzoin-Bildung; IV. Herstellung von Acyloinen mit Funktionellen Gruppen. Synthesis 1981, 477-478.
-
(1981)
Synthesis
, pp. 477-478
-
-
Stetter, H.1
Rämsch, R.Y.2
-
18
-
-
0015902629
-
Photoaffinity labels for estrogen binding proteins of rat uterus
-
Katzenellenbogen, J. A.; Johnson, H. J., Jr.; Myers, H. N. Photoaffinity Labels for Estrogen Binding Proteins of Rat Uterus. Biochemistry 1973, 12, 4085-4092.
-
(1973)
Biochemistry
, vol.12
, pp. 4085-4092
-
-
Katzenellenbogen, J.A.1
Johnson H.J., Jr.2
Myers, H.N.3
-
19
-
-
0030734795
-
Altered ligand binding properties and enhanced stability of a constitutively active estrogen receptor: Evidence that an open-pocket conformation is required for ligand interaction
-
Carlson, K. E.; Choi, I.; Gee, A.; Katzenellenbogen, B. S.; Katzenellenbogen, J. A. Altered Ligand Binding Properties and Enhanced Stability of a Constitutively Active Estrogen Receptor: Evidence That an Open-Pocket Conformation Is Required for Ligand Interaction. Biochemistry 1997, 36, 14897-14905.
-
(1997)
Biochemistry
, vol.36
, pp. 14897-14905
-
-
Carlson, K.E.1
Choi, I.2
Gee, A.3
Katzenellenbogen, B.S.4
Katzenellenbogen, J.A.5
-
20
-
-
0031059270
-
The estradiol pharmacophore: Ligand structure-estrogen receptor binding affinity relationships and a model for the receptor binding site
-
Anstead, G. M.; Carlson, K. E.; Katzenellenbogen, J. A. The Estradiol Pharmacophore: Ligand Structure-Estrogen Receptor Binding Affinity Relationships and a Model for the Receptor Binding Site. Steroids 1997, 62, 268-303.
-
(1997)
Steroids
, vol.62
, pp. 268-303
-
-
Anstead, G.M.1
Carlson, K.E.2
Katzenellenbogen, J.A.3
-
21
-
-
0030667676
-
Molecular basis of agonism and antagonism in the oestrogen receptor
-
Brzozowski, A. M.; Pike, A. C. W.; Dauter, Z.; Hubbard, R. E.; Bonn, T.; Engström, O.; Öhman, L.; Greene, G. L.; Gustafsson, J.-Å.; Carlquist, M. Molecular Basis of Agonism and Antagonism in the Oestrogen Receptor. Nature 1997, 389, 753-758.
-
(1997)
Nature
, vol.389
, pp. 753-758
-
-
Brzozowski, A.M.1
Pike, A.C.W.2
Dauter, Z.3
Hubbard, R.E.4
Bonn, T.5
Engström, O.6
Öhman, L.7
Greene, G.L.8
Gustafsson, J.-A.9
Carlquist, M.10
-
22
-
-
0032568527
-
Crystallographic comparison of the estrogen and progesterone receptor's ligand binding domains
-
Tanenbaum, D. M.; Wang, Y.; Williams, S. P.; Sigler, P. B. Crystallographic Comparison of the Estrogen and Progesterone Receptor's Ligand Binding Domains. Proc. Natl. Acad. Sci. U.S.A. 1998, 95, 5998-6003.
-
(1998)
Proc. Natl. Acad. Sci. U.S.A.
, vol.95
, pp. 5998-6003
-
-
Tanenbaum, D.M.1
Wang, Y.2
Williams, S.P.3
Sigler, P.B.4
-
23
-
-
0032446607
-
The structural basis of estrogen receptor/coactivator recognition and the antagonism of this interaction by tamoxifen
-
Shiau, A. K.; Barstad, D.; Loria, P. M.; Cheng, L.; Kushner, P. J.; Agard, D. A.; Greene, G. L. The Structural Basis of Estrogen Receptor/Coactivator Recognition and the Antagonism of This Interaction by Tamoxifen. Cell 1998, 95, 927-937.
-
(1998)
Cell
, vol.95
, pp. 927-937
-
-
Shiau, A.K.1
Barstad, D.2
Loria, P.M.3
Cheng, L.4
Kushner, P.J.5
Agard, D.A.6
Greene, G.L.7
-
24
-
-
0344725601
-
-
note
-
If one of the cis-THC enantiomers bound with the ligand core flipped 180° about the C-2/C-8 axis, the substituents from both enantiomers would project in the same direction. In the flipped orientation, however, the central two rings of the THC occupy quite a different spatial position.
-
-
-
-
25
-
-
0029058152
-
The carboxyl-terminal F domain of the human estrogen receptor: Role in the transcriptional activity of the receptor and the effectiveness of antiestrogens as estrogen antagonists
-
Montano, M. M.; Müller, V.; Trobaugh, A.; Katzenellenbogen, B. S. The Carboxyl-Terminal F Domain of the Human Estrogen Receptor: Role in the Transcriptional Activity of the Receptor and the Effectiveness of Antiestrogens as Estrogen Antagonists. Mol. Endocrinol 1995, 9, 814-825.
-
(1995)
Mol. Endocrinol
, vol.9
, pp. 814-825
-
-
Montano, M.M.1
Müller, V.2
Trobaugh, A.3
Katzenellenbogen, B.S.4
-
26
-
-
0029796605
-
Different regions in activation function-1 of the human estrogen receptor required for antiestrogen- and estradiol-dependent transcription activation
-
McInerney, E. M.; Katzenellenbogen, B. S. Different Regions in Activation Function-1 of the Human Estrogen Receptor Required for Antiestrogen- and Estradiol-Dependent Transcription Activation. J. Biol. Chem. 1996, 271, 24172-24178.
-
(1996)
J. Biol. Chem.
, vol.271
, pp. 24172-24178
-
-
McInerney, E.M.1
Katzenellenbogen, B.S.2
-
27
-
-
0031789876
-
Transcription activation by the human estrogen receptor subtype β (ERβ) studied with ERβ and ERα receptor chimeras
-
McInerney, E. M.; Weis, K. E.; Sun, J.; Mosselman, S.; Katzenellenbogen, B. S. Transcription Activation by the Human Estrogen Receptor Subtype β (ERβ) Studied with ERβ and ERα Receptor Chimeras. Endocrinology 1998, 139, 4513-4522.
-
(1998)
Endocrinology
, vol.139
, pp. 4513-4522
-
-
McInerney, E.M.1
Weis, K.E.2
Sun, J.3
Mosselman, S.4
Katzenellenbogen, B.S.5
-
28
-
-
0001557536
-
Diazomethane
-
Wiley: New York, Collect
-
Arndt, F. Diazomethane. Organic Syntheses; Wiley: New York, 1943; Collect. Vol. 2, pp 165-167.
-
(1943)
Organic Syntheses
, vol.2
, pp. 165-167
-
-
Arndt, F.1
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