Combinatorial synthesis of CCR5 antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 11, Issue 24, 2001, Pages 3137-3141

  Willoughby, Christopher A ^a   Berk, Scott C ^a   Rosauer, Keith G ^a   Degrado, Silvia ^a   Chapman, Kevin T ^a   Gould, Sandra L ^a   Springer, Martin S ^a   Malkowitz, Lorraine ^a   Schleif, William A ^a   Hazuda, Daria ^a   Miller, Michael ^a   Kessler, Joseph ^a   Danzeisen, Renee ^a   Holmes, Karen ^a   Lineberger, Janet ^a   Carella, Anthony ^a   Carver, Gwen ^a   Emini, Emilio A ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ANTI HUMAN IMMUNODEFICIENCY VIRUS AGENT; CHEMOKINE RECEPTOR CCR5; GLYCOPROTEIN GP 120; MACROPHAGE INFLAMMATORY PROTEIN 1ALPHA; RECEPTOR BLOCKING AGENT;

ANTIVIRAL ACTIVITY; ARTICLE; DRUG DESIGN; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; RECEPTOR AFFINITY; STRUCTURE ACTIVITY RELATION;

COMBINATORIAL CHEMISTRY TECHNIQUES; HIV-1; RECEPTORS, CCR5; STRUCTURE-ACTIVITY RELATIONSHIP;

HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 0035904882     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(01)00652-7     Document Type: Article

References (28)