-
2
-
-
0025485084
-
A new vasoconstrictor peptide, endothelin: Profiles as vasoconstrictor and neuropeptide
-
Shigeno T, Mima T: A new vasoconstrictor peptide, endothelin: profiles as vasoconstrictor and neuropeptide. Cerebrovasc Brain Metab Rev (1992) 2:227-239.
-
(1992)
Cerebrovasc Brain Metab Rev
, vol.2
, pp. 227-239
-
-
Shigeno, T.1
Mima, T.2
-
3
-
-
0026077104
-
Molecular and cellular mechanism of endothelin regulation. Implications for vascular function
-
Masaki T, Kimura S, Yanagisawa M, Goto K: Molecular and cellular mechanism of endothelin regulation. Implications for vascular function. Circulation (1991) 84:1457-1468.
-
(1991)
Circulation
, vol.84
, pp. 1457-1468
-
-
Masaki, T.1
Kimura, S.2
Yanagisawa, M.3
Goto, K.4
-
5
-
-
0025605930
-
Cloning of a cDNA encoding a non-isopeptide-selective subtype of the endothelin receptor
-
Sakurai T, Yanagisawa M, Takuwa Y, Miyazaki H, Kimura S, Goto K, Masaki T: Cloning of a cDNA encoding a non-isopeptide-selective subtype of the endothelin receptor. Nature (1990) 348:732-735.
-
(1990)
Nature
, vol.348
, pp. 732-735
-
-
Sakurai, T.1
Yanagisawa, M.2
Takuwa, Y.3
Miyazaki, H.4
Kimura, S.5
Goto, K.6
Masaki, T.7
-
6
-
-
0026547777
-
Distinct tissue distribution and cellular localization of two messenger ribonucleic acids encoding different subtypes of rat endothelin receptors
-
Hori S, Komatsu Y, Shigemoto R, Mizuno N, Nakanishi S: Distinct tissue distribution and cellular localization of two messenger ribonucleic acids encoding different subtypes of rat endothelin receptors. Endocrinology (1992) 130:1885-1895.
-
(1992)
Endocrinology
, vol.130
, pp. 1885-1895
-
-
Hori, S.1
Komatsu, Y.2
Shigemoto, R.3
Mizuno, N.4
Nakanishi, S.5
-
7
-
-
0027538163
-
Characterization and localization of endothelin receptor subtypes in the human atrioventricular conducting system and myocardium
-
Molenaar P, O'Reilly G, Sharkey A, Kuc RE, Harding DP, Plumpton C, Gresham GA, Devenport AP: Characterization and localization of endothelin receptor subtypes in the human atrioventricular conducting system and myocardium. Circ Res (1993) 72:526-538.
-
(1993)
Circ Res
, vol.72
, pp. 526-538
-
-
Molenaar, P.1
O'Reilly, G.2
Sharkey, A.3
Kuc, R.E.4
Harding, D.P.5
Plumpton, C.6
Gresham, G.A.7
Devenport, A.P.8
-
8
-
-
85047675578
-
Endothelin receptors in cultured adult rat cardiac fibroblasts
-
Katwa LC, Guarda E, Weber KT: Endothelin receptors in cultured adult rat cardiac fibroblasts. Cardiovasc Res (1993) 27:2125-2129.
-
(1993)
Cardiovasc Res
, vol.27
, pp. 2125-2129
-
-
Katwa, L.C.1
Guarda, E.2
Weber, K.T.3
-
9
-
-
0025605345
-
Cloning and expression of a cDNA encoding an endothelin receptor
-
Arai H, Hori S, Aramori I, Ohkubo H, Nakanishi S: Cloning and expression of a cDNA encoding an endothelin receptor. Nature (1990) 348:730-732.
-
(1990)
Nature
, vol.348
, pp. 730-732
-
-
Arai, H.1
Hori, S.2
Aramori, I.3
Ohkubo, H.4
Nakanishi, S.5
-
11
-
-
0025718651
-
Cloning and characterization of cDNA encoding human A-type endothelin receptor
-
Adachi M, Yang YY, Furuichi Y, Miyamoto C: Cloning and characterization of cDNA encoding human A-type endothelin receptor. Biochem Biophys Res Commun (1991) 180:1265-1272.
-
(1991)
Biochem Biophys Res Commun
, vol.180
, pp. 1265-1272
-
-
Adachi, M.1
Yang, Y.Y.2
Furuichi, Y.3
Miyamoto, C.4
-
12
-
-
0026563306
-
Molecular cloning and characterization of the major endothelin receptor subtype in porcine cerebellum
-
Elshourbagy NA, Lee JA, Korman DR, Nuthalaganti P, Sylvester DR, Dilella AG, Sutiphong JA, Kumar CS: Molecular cloning and characterization of the major endothelin receptor subtype in porcine cerebellum. Mol Pharmacol (1992) 41:465-473.
-
(1992)
Mol Pharmacol
, vol.41
, pp. 465-473
-
-
Elshourbagy, N.A.1
Lee, J.A.2
Korman, D.R.3
Nuthalaganti, P.4
Sylvester, D.R.5
Dilella, A.G.6
Sutiphong, J.A.7
Kumar, C.S.8
-
13
-
-
0025221768
-
Cellular signaling by peptides of the endothelin gene family
-
Simonson MS, Dunn MJ: Cellular signaling by peptides of the endothelin gene family. FASEB J (1990) 4:2989-3000.
-
(1990)
FASEB J
, vol.4
, pp. 2989-3000
-
-
Simonson, M.S.1
Dunn, M.J.2
-
14
-
-
0023859136
-
A novel potent vasoconstrictor peptide produced by vascular endothelial cells
-
Yanagisawa M, Kurihara H, Kimura S: A novel potent vasoconstrictor peptide produced by vascular endothelial cells. Nature (1989) 322:411-415.
-
(1989)
Nature
, vol.322
, pp. 411-415
-
-
Yanagisawa, M.1
Kurihara, H.2
Kimura, S.3
-
15
-
-
0009488762
-
-
Humana press Inc, Totowa, NJ
-
Brookes DP, Jorkasky DK, Freed MI, Ohlstein EH: Pathophysiological role of endothelin and potential therapeutic targets for receptor antagonists, in Endothelin: molecular biology, physiology and pathology. Humana press Inc, Totowa, NJ (1998) 223-268.
-
(1998)
Pathophysiological Role of Endothelin and Potential Therapeutic Targets for Receptor Antagonists, in Endothelin: Molecular Biology, Physiology and Pathology
, pp. 223-268
-
-
Brookes, D.P.1
Jorkasky, D.K.2
Freed, M.I.3
Ohlstein, E.H.4
-
16
-
-
0033537345
-
Endothelin antagonists
-
Benigni A, Remuzzi G: Endothelin antagonists. Lancet (1999) 353:133-138.
-
(1999)
Lancet
, vol.353
, pp. 133-138
-
-
Benigni, A.1
Remuzzi, G.2
-
18
-
-
0032996418
-
Heart failure and endothelin antagonists
-
Miyauchi T, Goto K: Heart failure and endothelin antagonists. Trends Pharmacol Sci (1999) 20:210-217.
-
(1999)
Trends Pharmacol Sci
, vol.20
, pp. 210-217
-
-
Miyauchi, T.1
Goto, K.2
-
19
-
-
0032968208
-
Endothelin antagonism with bosentan: A review of potential applications
-
Roux S, Breu V, Ertel SI, Clozel M: Endothelin antagonism with bosentan: a review of potential applications. J Molecular Med (1999) 77:364-376.
-
(1999)
J Molecular Med
, vol.77
, pp. 364-376
-
-
Roux, S.1
Breu, V.2
Ertel, S.I.3
Clozel, M.4
-
20
-
-
0032780617
-
Endothelins and their receptors in cirrhotic and neoplastic livers of Canadian and Chinese populations
-
Cai L, Wang GJ, Mukherjee K, Xu ZL, Khalil M, Cherian MG, Chakrabarti S: Endothelins and their receptors in cirrhotic and neoplastic livers of Canadian and Chinese populations. Anticancer Res (1999) 19:2243-2248.
-
(1999)
Anticancer Res
, vol.19
, pp. 2243-2248
-
-
Cai, L.1
Wang, G.J.2
Mukherjee, K.3
Xu, Z.L.4
Khalil, M.5
Cherian, M.G.6
Chakrabarti, S.7
-
21
-
-
0032942944
-
Anti-ulcerogenic properties of endothelin receptor antagonists in the rat
-
Padol I, Huang JQ, Hunt RH: Anti-ulcerogenic properties of endothelin receptor antagonists in the rat. Aliment Pharmacol Ther (1999) 13:537-544.
-
(1999)
Aliment Pharmacol Ther
, vol.13
, pp. 537-544
-
-
Padol, I.1
Huang, J.Q.2
Hunt, R.H.3
-
22
-
-
0027310294
-
Endothelins: Homeostatic and compensatory actions in the circulatory and endocrine systems
-
Masaki T: Endothelins: Homeostatic and compensatory actions in the circulatory and endocrine systems. Endocr Rev (1993) 14:256-268.
-
(1993)
Endocr Rev
, vol.14
, pp. 256-268
-
-
Masaki, T.1
-
23
-
-
0030038443
-
Endothelin receptors and activity differ in human, dog, and rabbit lung
-
McKay KO, Armour CL, Black JL: Endothelin receptors and activity differ in human, dog, and rabbit lung. Am J Physiol (1996) 270:L37-L43.
-
(1996)
Am J Physiol
, vol.270
-
-
McKay, K.O.1
Armour, C.L.2
Black, J.L.3
-
24
-
-
0026641543
-
Endothelin rapidly stimulates mitogen-activated protein kinase activity in rat mesangial cells
-
Wang Y, Simonson MS, Poussegur J, Dunn MJ: Endothelin rapidly stimulates mitogen-activated protein kinase activity in rat mesangial cells. Biochem J (1992) 287:589-594.
-
(1992)
Biochem J
, vol.287
, pp. 589-594
-
-
Wang, Y.1
Simonson, M.S.2
Poussegur, J.3
Dunn, M.J.4
-
25
-
-
3142651526
-
Studies on type IV collagen production in culture mesangial cells
-
Sawada T, Haneda M, Togawa M, Kikkawa R: Studies on type IV collagen production in culture mesangial cells. Jpn J Nephrol (1996) 38:469-474.
-
(1996)
Jpn J Nephrol
, vol.38
, pp. 469-474
-
-
Sawada, T.1
Haneda, M.2
Togawa, M.3
Kikkawa, R.4
-
26
-
-
0033609032
-
Role of endothelin in deterioration of heart failure due to cardiomyopathy in hamsters: Increase in endothelin-1 production in the heart and beneficial effect of endothelin-A receptor antagonist on survival and cardiac function
-
Yamauchi-Kohno R, Miyauchi T, Hoshino T, Kobayashi T, Aihara H, Sakai S, Yabana H, Goto K, Sugishita Y, Murata S: Role of endothelin in deterioration of heart failure due to cardiomyopathy in hamsters: increase in endothelin-1 production in the heart and beneficial effect of endothelin-A receptor antagonist on survival and cardiac function. Circulation (1999) 99:2171-2176.
-
(1999)
Circulation
, vol.99
, pp. 2171-2176
-
-
Yamauchi-Kohno, R.1
Miyauchi, T.2
Hoshino, T.3
Kobayashi, T.4
Aihara, H.5
Sakai, S.6
Yabana, H.7
Goto, K.8
Sugishita, Y.9
Murata, S.10
-
27
-
-
0032898256
-
Macrophage and myofibroblast involvement in ischemic acute renal failure is attenuated by endothelin receptor antagonists
-
Forbes JM, Leaker B, Hewitson TD, Becker GJ, Jones CL: Macrophage and myofibroblast involvement in ischemic acute renal failure is attenuated by endothelin receptor antagonists. Kidney Int (1999) 55:198-208.
-
(1999)
Kidney Int
, vol.55
, pp. 198-208
-
-
Forbes, J.M.1
Leaker, B.2
Hewitson, T.D.3
Becker, G.J.4
Jones, C.L.5
-
28
-
-
0030694639
-
Clinical development of endothelin receptor antagonists
-
Douglas SA: Clinical development of endothelin receptor antagonists. Trends Pharmacol Sci (1997) 18:408-412.
-
(1997)
Trends Pharmacol Sci
, vol.18
, pp. 408-412
-
-
Douglas, S.A.1
-
30
-
-
0033514321
-
Effects of a specific endothelin-converting enzyme inhibitor on cardiac, renal, and neurohumoral functions in congestive heart failure
-
Wada A, Tsutamoto T, Ohnishi M, Sawaki M, Fukai D, Maeda Y, Kinoshita M: Effects of a specific endothelin-converting enzyme inhibitor on cardiac, renal, and neurohumoral functions in congestive heart failure. Circulation (1999) 99:570-577.
-
(1999)
Circulation
, vol.99
, pp. 570-577
-
-
Wada, A.1
Tsutamoto, T.2
Ohnishi, M.3
Sawaki, M.4
Fukai, D.5
Maeda, Y.6
Kinoshita, M.7
-
31
-
-
0027052320
-
Cochinmicins, novel and potent cyclodepsipeptide endothelin antagonists from a Microbispora sp.
-
Lam YKT, Willims DL, Sigmund JM, Sawchez M, Genilloud O, Koug YL, Stevens-Miles S, Huang L, Garrity GM: Cochinmicins, novel and potent cyclodepsipeptide endothelin antagonists from a Microbispora sp. J Antibiot (1992) 45:1709-1716.
-
(1992)
J Antibiot
, vol.45
, pp. 1709-1716
-
-
Lam, Y.K.T.1
Willims, D.L.2
Sigmund, J.M.3
Sawchez, M.4
Genilloud, O.5
Koug, Y.L.6
Stevens-Miles, S.7
Huang, L.8
Garrity, G.M.9
-
32
-
-
0027092420
-
Cochinmicins, novel and potent cyclodepsipeptide endothelin antagonists from a Microspora sp
-
Zink D, Hensens OD, Iam YKT, Reamer R, Liesch JM: Cochinmicins, novel and potent cyclodepsipeptide endothelin antagonists from a Microspora sp. J Antibiot (1992) 45:1717-1722.
-
(1992)
J Antibiot
, vol.45
, pp. 1717-1722
-
-
Zink, D.1
Hensens, O.D.2
Iam, Y.K.T.3
Reamer, R.4
Liesch, J.M.5
-
33
-
-
0026319175
-
Endothelin-binding inhibitors, BE-18257a and BE-18257B. I. Taxonomy, fermentation, isolation and characterization
-
Kojiri K, Ihara M, Nakajima S, Kawamura K, Funaishi K, Yano M, Suda H: Endothelin-binding inhibitors, BE-18257a and BE-18257B. I. Taxonomy, fermentation, isolation and characterization. J Antibiot (1991) 44:1342-1347.
-
(1991)
J Antibiot
, vol.44
, pp. 1342-1347
-
-
Kojiri, K.1
Ihara, M.2
Nakajima, S.3
Kawamura, K.4
Funaishi, K.5
Yano, M.6
Suda, H.7
-
34
-
-
0029854741
-
The combinatorial chemistry of nature
-
Verdine, GL: The combinatorial chemistry of nature. Nature (1996) 384:11-13.
-
(1996)
Nature
, vol.384
, pp. 11-13
-
-
Verdine, G.L.1
-
35
-
-
0342288717
-
Attack as the best form of defense: Natural product in the forefront of contemporary drug research
-
Moore, M: Attack as the best form of defense: Natural product in the forefront of contemporary drug research. J Biomol Screen (1996) 1:19-23.
-
(1996)
J Biomol Screen
, vol.1
, pp. 19-23
-
-
Moore, M.1
-
36
-
-
0029911948
-
For medical purposes
-
Petsko GA: For medical purposes. Nature (1996) 384:7-9.
-
(1996)
Nature
, vol.384
, pp. 7-9
-
-
Petsko, G.A.1
-
37
-
-
0002441921
-
Endophytic microbes embody pharmaceutical potential
-
Strobel GA, Long DM: Endophytic microbes embody pharmaceutical potential. ASM News (1998) 64:263-268.
-
(1998)
ASM News
, vol.64
, pp. 263-268
-
-
Strobel, G.A.1
Long, D.M.2
-
38
-
-
0031595885
-
Paclitaxol (Taxol): A success story with valuable lessons for natural product drug discovery and development
-
Cragg GM: Paclitaxol (Taxol): a success story with valuable lessons for natural product drug discovery and development. Med Res Rev (1998) 18:315-331.
-
(1998)
Med Res Rev
, vol.18
, pp. 315-331
-
-
Cragg, G.M.1
-
39
-
-
0029671145
-
History of Cyclosporin A (Sandimmune) revisited
-
Stahelin HF: History of Cyclosporin A (Sandimmune) revisited. Experientia (1996) 52:5-13.
-
(1996)
Experientia
, vol.52
, pp. 5-13
-
-
Stahelin, H.F.1
-
41
-
-
0028052780
-
Pathway engineering in secondary meatbolite-producing actinomycetes
-
Pipersberg W: Pathway engineering in secondary meatbolite-producing actinomycetes. Crit Rev Biotechnol (1994) 14:251-285.
-
(1994)
Crit Rev Biotechnol
, vol.14
, pp. 251-285
-
-
Pipersberg, W.1
-
42
-
-
0033014645
-
Analysis of fungal diversity in the wheat rhizosphere by sequencing of cloned PCR-amplified genes encoding 18S rRNA and temperature gradient gel electrophoresis
-
Smit E, Leeflang P, Glandorf B, van Elsas JD, Wemars K: Analysis of fungal diversity in the wheat rhizosphere by sequencing of cloned PCR-amplified genes encoding 18S rRNA and temperature gradient gel electrophoresis. Appl Environ Microbiol (1999) 65:2614-2621.
-
(1999)
Appl Environ Microbiol
, vol.65
, pp. 2614-2621
-
-
Smit, E.1
Leeflang, P.2
Glandorf, B.3
Van Elsas, J.D.4
Wemars, K.5
-
43
-
-
0033023519
-
Combination ACE inhibitor and angiotensin II receptor antagonist therapy in diabetic nephropathy
-
Hebert LA, Falkenhain ME, Nahman Jr NS, Cosio FG, O'Dorisio TM: Combination ACE inhibitor and angiotensin II receptor antagonist therapy in diabetic nephropathy. Am J Nephrol (1999) 19:1-6.
-
(1999)
Am J Nephrol
, vol.19
, pp. 1-6
-
-
Hebert, L.A.1
Falkenhain, M.E.2
Nahman Jr., N.S.3
Cosio, F.G.4
O'Dorisio, T.M.5
-
44
-
-
0032960827
-
Mitogen-activated protein kinase cascade is involved in endothelin-1-induced rat puerperal uterine contraction
-
Kimura A, Ohmichi M, Takeda T, Kurachi H, Ikegami H, Koike K, Masuhara K, Hayakawa J, Kanzaki T, Kobayashi M, Akabane M, Inoue M, Miyake A, Murata Y: Mitogen-activated protein kinase cascade is involved in endothelin-1-induced rat puerperal uterine contraction. Endocrinology (1999) 140:722-731.
-
(1999)
Endocrinology
, vol.140
, pp. 722-731
-
-
Kimura, A.1
Ohmichi, M.2
Takeda, T.3
Kurachi, H.4
Ikegami, H.5
Koike, K.6
Masuhara, K.7
Hayakawa, J.8
Kanzaki, T.9
Kobayashi, M.10
Akabane, M.11
Inoue, M.12
Miyake, A.13
Murata, Y.14
-
45
-
-
0029985798
-
Protective effect of the specific endothelin-1 antagonist BQ610 on mechanical function and energy metabolism during ischemia/reperfusion injury in isolated perfused rat hearts
-
Illing B, Horn M, Han H, Hahn S, Bureik P, Ertl G, Neubauer S: Protective effect of the specific endothelin-1 antagonist BQ610 on mechanical function and energy metabolism during ischemia/reperfusion injury in isolated perfused rat hearts. J Cardiovasc Pharmacol (1996) 27:487-494.
-
(1996)
J Cardiovasc Pharmacol
, vol.27
, pp. 487-494
-
-
Illing, B.1
Horn, M.2
Han, H.3
Hahn, S.4
Bureik, P.5
Ertl, G.6
Neubauer, S.7
-
46
-
-
0031630062
-
Efficacy of CI-020, an endothelin-A receptor antagonist, in hypoxic pulmonary hypertension
-
Haleen S, Schroeder R, Walker D, Quenby-Brown E, Welch K, Hallak H, Uprichard A, Keiser J: Efficacy of CI-020, an endothelin-A receptor antagonist, in hypoxic pulmonary hypertension. J Cardiovasc Pharmacol (1998) 31:S331-S335.
-
(1998)
J Cardiovasc Pharmacol
, vol.31
-
-
Haleen, S.1
Schroeder, R.2
Walker, D.3
Quenby-Brown, E.4
Welch, K.5
Hallak, H.6
Uprichard, A.7
Keiser, J.8
-
47
-
-
0032217194
-
A antagonist CI-1020 Inhibits hypoxic pulmonary vasoconstriction in small isolated rat pulmonary arteries
-
A antagonist CI-1020 Inhibits hypoxic pulmonary vasoconstriction in small isolated rat pulmonary arteries. Pulm Pharmacol Ther (1998) 11:177-181.
-
(1998)
Pulm Pharmacol Ther
, vol.11
, pp. 177-181
-
-
Jones, R.D.1
Morice, A.H.2
-
49
-
-
15144360873
-
A antagonist (A-216546)
-
A antagonist (A-216546). J Med Chem (1998) 41:3261-3275.
-
(1998)
J Med Chem
, vol.41
, pp. 3261-3275
-
-
Liu, G.1
Henry Jr., K.J.2
Szczepankiewicz, B.G.3
Winn, M.4
Kozmina, N.S.5
Boyd, S.A.6
Wasicak, J.7
Von Geldern, T.W.8
Wu-Wong, J.R.9
Chiou, W.J.10
Dixon, D.B.11
Nguyen, B.12
Marsh, K.C.13
Opgenorth, T.J.14
-
50
-
-
0032008565
-
A receptor antagonist, BMS-182874, reduces acute hypoxic pulmonary hypertension in pigs in vivo
-
A receptor antagonist, BMS-182874, reduces acute hypoxic pulmonary hypertension in pigs in vivo. Cardiovasc Res (1998), 37:765-771.
-
(1998)
Cardiovasc Res
, vol.37
, pp. 765-771
-
-
Holm, P.1
Liska, J.2
Franco-Cereceda, A.3
-
51
-
-
0031760395
-
Systemic administration of the endothelin-A receptor antagonist TBC 11251 attenuates cerebral vasospasm after experimental subarachnoid hemorrhage: Dose study and review of endothelin-based therapies in the literature on cerebral vasospasm
-
Wanebo JE, Arthur AS, Louis HG, West K, Kassell NF, Lee KS, Helm GA: Systemic administration of the endothelin-A receptor antagonist TBC 11251 attenuates cerebral vasospasm after experimental subarachnoid hemorrhage: dose study and review of endothelin-based therapies in the literature on cerebral vasospasm. Neurosurgery (1998) 43:1409-1417.
-
(1998)
Neurosurgery
, vol.43
, pp. 1409-1417
-
-
Wanebo, J.E.1
Arthur, A.S.2
Louis, H.G.3
West, K.4
Kassell, N.F.5
Lee, K.S.6
Helm, G.A.7
-
52
-
-
0032588243
-
A receptor blockade attenuates cardiac hypertrophy independent of blood pressure effects in renovascular hypertensive rats
-
A receptor blockade attenuates cardiac hypertrophy independent of blood pressure effects in renovascular hypertensive rats. Hypertension (1999) 33:954-960.
-
(1999)
Hypertension
, vol.33
, pp. 954-960
-
-
Ehmke, H.1
Faulhaber, J.2
Munter, K.3
Kirchengast, M.4
Wiesner, R.J.5
-
53
-
-
0008901574
-
Effects of an endothelin ET(A)-receptor antagonist, S-0139, on cerebral vasospasm and behavioral changes in dogs intracisternally administered endothelin-1
-
Sato S, Yonetani Y, Fujimoto M, Kita K, Kubo K, Nakashima T: Effects of an endothelin ET(A)-receptor antagonist, S-0139, on cerebral vasospasm and behavioral changes in dogs intracisternally administered endothelin-1. Life Sci (1998) 62:191-197.
-
(1998)
Life Sci
, vol.62
, pp. 191-197
-
-
Sato, S.1
Yonetani, Y.2
Fujimoto, M.3
Kita, K.4
Kubo, K.5
Nakashima, T.6
-
54
-
-
0033034854
-
A receptor
-
A receptor. Eur J Pharmacol (1999) 366:189-201.
-
(1999)
Eur J Pharmacol
, vol.366
, pp. 189-201
-
-
Wu-Wong, J.R.1
Dixon, D.B.2
Chiou, W.J.3
Dayton, B.D.4
Novosad, E.I.5
Adler, A.L.6
Wessale, J.L.7
Calzadilla, S.V.8
Hemandez, L.9
Marsh, K.C.10
Liu, G.11
Szczepankiewicz, B.12
Von Geldern, T.W.13
Opgenorth, T.J.14
-
55
-
-
0032493194
-
A selective antagonist
-
A selective antagonist. Bioorg Med Chem Lett (1998) 8:1771-1776.
-
(1998)
Bioorg Med Chem Lett
, vol.8
, pp. 1771-1776
-
-
Mederski, W.W.1
Dorsch, D.2
Osswald, M.3
Anzali, S.4
Christadler, M.5
Schmitges, C.J.6
Schelling, P.7
Wilm, C.8
Ruck, M.9
-
56
-
-
0031456079
-
Ro 61-1790, a new hydrosoluble endothelin antagonist: General pharmacology and effects on experimental cerebral vasospasm
-
Roux S, Breu V, Giller T, Neidhart W, Ramuz H, Coassolo P, Clozel JP, Clozel M: Ro 61-1790, a new hydrosoluble endothelin antagonist: general pharmacology and effects on experimental cerebral vasospasm. J Pharmacol Exp Ther (1997) 283:1110-1118.
-
(1997)
J Pharmacol Exp Ther
, vol.283
, pp. 1110-1118
-
-
Roux, S.1
Breu, V.2
Giller, T.3
Neidhart, W.4
Ramuz, H.5
Coassolo, P.6
Clozel, J.P.7
Clozel, M.8
-
57
-
-
0001650691
-
SB 234551, a novel endothelin-A receptor antagonist, unmasks endothelin-induced renal vasodilatation in the dog
-
Brooks DP, DePalma PD, Pullen M, Elliott JD, Ohlstein EH, Nambi P: SB 234551, a novel endothelin-A receptor antagonist, unmasks endothelin-induced renal vasodilatation in the dog. J Cardiovasc Pharmacol (1998) 31:5339-8341.
-
(1998)
J Cardiovasc Pharmacol
, vol.31
, pp. 5339-8341
-
-
Brooks, D.P.1
Depalma, P.D.2
Pullen, M.3
Elliott, J.D.4
Ohlstein, E.H.5
Nambi, P.6
-
58
-
-
0031854946
-
A novel orally active endothelin-A receptor antagonist, ZD1611, prevents chronic hypoxia-induced pulmonary hypertension in the rat
-
Bialecki RA, Stinson-Fisher C, Murdoch W, Bertelsen D, Desiato M, Rumsey W: A novel orally active endothelin-A receptor antagonist, ZD1611, prevents chronic hypoxia-induced pulmonary hypertension in the rat. Chest (1998) 114:91S.
-
(1998)
Chest
, vol.114
-
-
Bialecki, R.A.1
Stinson-Fisher, C.2
Murdoch, W.3
Bertelsen, D.4
Desiato, M.5
Rumsey, W.6
-
59
-
-
0032424117
-
Pharmacological profile of T-0201, a highly potent and orally active endothelin receptor antagonist
-
Hoshino T, Yamauchi R, Kikkawa K, Yabana H, Murata S: Pharmacological profile of T-0201, a highly potent and orally active endothelin receptor antagonist. J Pharmacol Exp Ther (1998) 286:643-649.
-
(1998)
J Pharmacol Exp Ther
, vol.286
, pp. 643-649
-
-
Hoshino, T.1
Yamauchi, R.2
Kikkawa, K.3
Yabana, H.4
Murata, S.5
-
60
-
-
0031879390
-
Increased expression of endothelin receptors in the vasculature of portal hypertensive rats: Role in splanchnic hemodynamics
-
Cahill PA, Hou MC, Hendrickson R, Wang YN, Zhang S, Redmond EM, Sitzman JV: Increased expression of endothelin receptors in the vasculature of portal hypertensive rats: role in splanchnic hemodynamics. Hepatology (1998) 28:396-403.
-
(1998)
Hepatology
, vol.28
, pp. 396-403
-
-
Cahill, P.A.1
Hou, M.C.2
Hendrickson, R.3
Wang, Y.N.4
Zhang, S.5
Redmond, E.M.6
Sitzman, J.V.7
-
61
-
-
0032544150
-
B affinity
-
B affinity. Bioorg Med Chem Lett (1998) 8:2241-2246.
-
(1998)
Bioorg Med Chem Lett
, vol.8
, pp. 2241-2246
-
-
Sakaki, J.1
Murata, T.2
Yuumoto, Y.3
Nakamura, I.4
Trueh, T.5
Pittema, T.6
Iwasaki, G.7
Oda, K.8
Yamamura, T.9
Hayakawa, K.10
-
62
-
-
0032442833
-
Hybrid peptides constructed from RES-701-1, an endothelin B receptor antagonist, and endothelin; binding selectivity for endothelin receptors and their pharmacological activity
-
Shibata K, Suzawa T, Ohno T, Yamada K, Tanaka T, Tsukuda E, Matsuda Y, Yamasaki M: Hybrid peptides constructed from RES-701-1, an endothelin B receptor antagonist, and endothelin; binding selectivity for endothelin receptors and their pharmacological activity. Bioorg Med Chem (1998) 6:2459-2467.
-
(1998)
Bioorg Med Chem
, vol.6
, pp. 2459-2467
-
-
Shibata, K.1
Suzawa, T.2
Ohno, T.3
Yamada, K.4
Tanaka, T.5
Tsukuda, E.6
Matsuda, Y.7
Yamasaki, M.8
-
63
-
-
0033135846
-
BQ788, an endothelin ET(B) receptor antagonist, attenuates stab wound injury-induced reactive astrocytes in rat brain
-
Koyama Y, Takemura M, Fujiki K, Ishikawa N, Shigenaga Y, Baba A: BQ788, an endothelin ET(B) receptor antagonist, attenuates stab wound injury-induced reactive astrocytes in rat brain. Glia (1999) 26:268-271.
-
(1999)
Glia
, vol.26
, pp. 268-271
-
-
Koyama, Y.1
Takemura, M.2
Fujiki, K.3
Ishikawa, N.4
Shigenaga, Y.5
Baba, A.6
-
64
-
-
0033042155
-
Different contributions of endothelin-A and endothelin-B receptors in the pathogenesis of deoxycorticosterone acetate-salt-induced hypertension in rats
-
Matsumura Y, Hashimoto N, Taira S, Kuro T, Kitano R, Ohkita M, Opgenorth TJ, Takaoka M: Different contributions of endothelin-A and endothelin-B receptors in the pathogenesis of deoxycorticosterone acetate-salt-induced hypertension in rats. Hypertension (1999) 33:759-765.
-
(1999)
Hypertension
, vol.33
, pp. 759-765
-
-
Matsumura, Y.1
Hashimoto, N.2
Taira, S.3
Kuro, T.4
Kitano, R.5
Ohkita, M.6
Opgenorth, T.J.7
Takaoka, M.8
-
65
-
-
0029613835
-
Stachybocins, novel endothelin receptor antagonists, produced by Stachybotrys sp. M6222.II. Structure determination and stachybocins A, B and C
-
Ogawa K, Nakamura M, Yaginuma S, Yamamoto S, Furihata K, Shin-Ya K, Seta H: Stachybocins, novel endothelin receptor antagonists, produced by Stachybotrys sp. M6222.II. Structure determination and stachybocins A, B and C. J Antibiot (1995) 48:1396-1400.
-
(1995)
J Antibiot
, vol.48
, pp. 1396-1400
-
-
Ogawa, K.1
Nakamura, M.2
Yaginuma, S.3
Yamamoto, S.4
Furihata, K.5
Shin-Ya, K.6
Seta, H.7
-
66
-
-
0029669946
-
B receptor antagonist Ro 46-8443
-
B receptor antagonist Ro 46-8443. FEBS Letters (1996) 383:42-45.
-
(1996)
FEBS Letters
, vol.383
, pp. 42-45
-
-
Clozel, M.1
Breu, V.2
-
67
-
-
0031647397
-
PD 142893, SB 209670, and BQ 788 selectively antagonize vascular endothelial versus vascular smooth muscle ET(B)-receptor activity in the rat
-
Schroeder RL, Keiser JA, Cheng XM, Haleen SJ: PD 142893, SB 209670, and BQ 788 selectively antagonize vascular endothelial versus vascular smooth muscle ET(B)-receptor activity in the rat. J Cardiovasc Pharmacol (1998) 32:935-943.
-
(1998)
J Cardiovasc Pharmacol
, vol.32
, pp. 935-943
-
-
Schroeder, R.L.1
Keiser, J.A.2
Cheng, X.M.3
Haleen, S.J.4
-
68
-
-
0031031076
-
Cardiovascular and renal effects of endothelin receptor blockade with PD 145065 and interaction with urodilatin
-
Dobrowolski L, Endlich K, Sadowski J, Steinhausen M: Cardiovascular and renal effects of endothelin receptor blockade with PD 145065 and interaction with urodilatin. Acta Physiol Scand (1997) 159:7-13.
-
(1997)
Acta Physiol Scand
, vol.159
, pp. 7-13
-
-
Dobrowolski, L.1
Endlich, K.2
Sadowski, J.3
Steinhausen, M.4
-
69
-
-
0032907460
-
Effect of non-selective endothelin blockade, TAK-044, on the ischemic cellular injury of rat heart
-
Geshi E, Nomizo A, Arata Y, Nakatani M, Katagiri T: Effect of non-selective endothelin blockade, TAK-044, on the ischemic cellular injury of rat heart. Basic Res Cardiol (1999) 94:94-101.
-
(1999)
Basic Res Cardiol
, vol.94
, pp. 94-101
-
-
Geshi, E.1
Nomizo, A.2
Arata, Y.3
Nakatani, M.4
Katagiri, T.5
-
70
-
-
0030746698
-
Design of a potent combined pseudopeptide endothelin-A/endothelin-B receptor antagonist, Ac-DBhg16-Leu-Asp-Ile-[NMe]Ile-Trp21 (PD 156252): Examination of its pharmacokinetic and spectral properties
-
Cody WL, He JX, Reily MD, Haleen SJ, Walker DM, Reyner EL, Stewart BH, Doherty AM: Design of a potent combined pseudopeptide endothelin-A/endothelin-B receptor antagonist, Ac-DBhg16-Leu-Asp-Ile-[NMe]Ile-Trp21 (PD 156252): examination of its pharmacokinetic and spectral properties. J Med Chem (1997) 40:2228-2240.
-
(1997)
J Med Chem
, vol.40
, pp. 2228-2240
-
-
Cody, W.L.1
He, J.X.2
Reily, M.D.3
Haleen, S.J.4
Walker, D.M.5
Reyner, E.L.6
Stewart, B.H.7
Doherty, A.M.8
-
71
-
-
0032774168
-
Protective effect of the endothelin antagonist bosentan against ischemic skeletal muscle necrosis
-
Hvaal K, Mathisen SR, Svindland A, Nordsletten L, Skjeldal S: Protective effect of the endothelin antagonist bosentan against ischemic skeletal muscle necrosis. Acta Orthop Scand (1999) 70:293-297.
-
(1999)
Acta Orthop Scand
, vol.70
, pp. 293-297
-
-
Hvaal, K.1
Mathisen, S.R.2
Svindland, A.3
Nordsletten, L.4
Skjeldal, S.5
-
72
-
-
0032766706
-
Pharmacology of tezosentan, new endothelin receptor antagonist designed for parenteral use
-
Clozel M, Ramuz H, Clozel JP, Breu V, Hess P, Loffler BM, Coassolo P, Roux S: Pharmacology of tezosentan, new endothelin receptor antagonist designed for parenteral use. J Pharmacol Exp Ther (1999) 290:840-846.
-
(1999)
J Pharmacol Exp Ther
, vol.290
, pp. 840-846
-
-
Clozel, M.1
Ramuz, H.2
Clozel, J.P.3
Breu, V.4
Hess, P.5
Loffler, B.M.6
Coassolo, P.7
Roux, S.8
-
73
-
-
0031837024
-
Efficacy of administering an endothelin-receptor antagonist (SB209670) in ameliorating ischemia-reperfusion injury in lung allografts
-
Shennib H, Lee AG, Kuang JQ, Yanagisawa M, Ohlstein EH, Giaid A: Efficacy of administering an endothelin-receptor antagonist (SB209670) in ameliorating ischemia-reperfusion injury in lung allografts. Am J Respir Crit Care Med (1998), 157:1975-1981.
-
(1998)
Am J Respir Crit Care Med
, vol.157
, pp. 1975-1981
-
-
Shennib, H.1
Lee, A.G.2
Kuang, J.Q.3
Yanagisawa, M.4
Ohlstein, E.H.5
Giaid, A.6
-
74
-
-
0032499652
-
Application of serial in vivo magnetic resonance imaging to evaluate the efficacy of endothelin receptor antagonist SB 217242 in the rat carotid artery model of neointime formation
-
Chandra S, Clark LV, Coatney RW, Phan L, Sarkar SK, Ohlstein EH: Application of serial in vivo magnetic resonance imaging to evaluate the efficacy of endothelin receptor antagonist SB 217242 in the rat carotid artery model of neointime formation. Circulation (1998) 97:2252-2258.
-
(1998)
Circulation
, vol.97
, pp. 2252-2258
-
-
Chandra, S.1
Clark, L.V.2
Coatney, R.W.3
Phan, L.4
Sarkar, S.K.5
Ohlstein, E.H.6
-
75
-
-
0029551537
-
Pharmacology of L-754,142, a highly potent, orally active, nonpeptidyl endothelin antagonist
-
Williams Jr DL, Murphy KL, Nolan NA, O'Brien JA, Pittibone DJ, Kivlighn SD, Krause SM, Lis Jr EV, Zingaro GJ, Gabei RA, Clayton FC, Siegl PKS, Zhang K, Naue J, Vyas K, Walsh TF, Fitch KJ, Chakravarty PK, Greenlee WJ, Clineschmidt BV: Pharmacology of L-754,142, a highly potent, orally active, nonpeptidyl endothelin antagonist. J Pharmacol Exp Ther (1995) 275:1518-1526.
-
(1995)
J Pharmacol Exp Ther
, vol.275
, pp. 1518-1526
-
-
Williams Jr., D.L.1
Murphy, K.L.2
Nolan, N.A.3
O'Brien, J.A.4
Pittibone, D.J.5
Kivlighn, S.D.6
Krause, S.M.7
Lis Jr., E.V.8
Zingaro, G.J.9
Gabei, R.A.10
Clayton, F.C.11
Siegl, P.K.S.12
Zhang, K.13
Naue, J.14
Vyas, K.15
Walsh, T.F.16
Fitch, K.J.17
Chakravarty, P.K.18
Greenlee, W.J.19
Clineschmidt, B.V.20
more..
-
76
-
-
0032958019
-
The ET(A) receptor blocker LU 135252 prevents chronic transplant nephropathy in the "Fisher to Lewis" model
-
Orth SR, Odoni G, Amann K, Strzelczyk P, Raschack M, Ritz E: The ET(A) receptor blocker LU 135252 prevents chronic transplant nephropathy in the "Fisher to Lewis" model. J Am Soc Nephrol (1999) 10:387-391.
-
(1999)
J Am Soc Nephrol
, vol.10
, pp. 387-391
-
-
Orth, S.R.1
Odoni, G.2
Amann, K.3
Strzelczyk, P.4
Raschack, M.5
Ritz, E.6
-
77
-
-
0029925702
-
The unusual binding properties of the endothelin receptor antagonist CGS 27830 distinguishes receptor/agonist interactions
-
Chin MH, Cioffi CL, Garay M, Neale RF, Shetty SS, DelGrande D, Mugrage B, Sills MA, Lipson KE: The unusual binding properties of the endothelin receptor antagonist CGS 27830 distinguishes receptor/agonist interactions. J Pharmacol Exp Ther (1996) 276:74-83.
-
(1996)
J Pharmacol Exp Ther
, vol.276
, pp. 74-83
-
-
Chin, M.H.1
Cioffi, C.L.2
Garay, M.3
Neale, R.F.4
Shetty, S.S.5
DelGrande, D.6
Mugrage, B.7
Sills, M.A.8
Lipson, K.E.9
-
78
-
-
0001271975
-
LU302872 and its racemate (LU224332) show balanced endothelin-A/B receptor affinity, high oral activity, and inhibit human prostate tissue contractions
-
Raschack M, Gock S, Unger L, Hahn A, Amberg W, Jansen R, Alken P, Weber A, Hergenroder S: LU302872 and its racemate (LU224332) show balanced endothelin-A/B receptor affinity, high oral activity, and inhibit human prostate tissue contractions. J Cardiovasc Pharmacol (1998) 31:5241-244.
-
(1998)
J Cardiovasc Pharmacol
, vol.31
, pp. 5241-5244
-
-
Raschack, M.1
Gock, S.2
Unger, L.3
Hahn, A.4
Amberg, W.5
Jansen, R.6
Alken, P.7
Weber, A.8
Hergenroder, S.9
-
79
-
-
0033032181
-
B endothelin receptor antagonist
-
B endothelin receptor antagonist. J Pharmacol Exp Ther (1999) 289:1262-1270.
-
(1999)
J Pharmacol Exp Ther
, vol.289
, pp. 1262-1270
-
-
Nishikibe, M.1
Ohta, H.2
Okada, M.3
Ishikawa, K.4
Hayama, T.5
Fukuroda, T.6
Noguchi, K.7
Saito, M.8
Kanoh, T.9
Ozaki, S.10
Kamei, T.11
Hara, K.12
William, D.13
Kivlighn, S.14
Krause, S.15
Gabel, R.16
Zingaro, G.17
Nolan, N.18
O'Brien, J.19
Clayton, F.20
Lynch, J.21
Pettibone, D.22
Siegl, P.23
more..
-
80
-
-
0028810898
-
WS75624 a and B, new endothelin converting enzyme inhibitors isolated from Saccharothrix sp. No. 75624. II. Structure elucidation of WS75624 a and B
-
Yoshimura S, Tsurumi Y, Takase S, Okuhara M: WS75624 A and B, new endothelin converting enzyme inhibitors isolated from Saccharothrix sp. No. 75624. II. Structure elucidation of WS75624 A and B. J Antibiot (1995) 48:1073-1075.
-
(1995)
J Antibiot
, vol.48
, pp. 1073-1075
-
-
Yoshimura, S.1
Tsurumi, Y.2
Takase, S.3
Okuhara, M.4
-
81
-
-
0030799481
-
Prevention and reversal of cerebral vasospasm by an endothelin-converting enzyme inhibitor, CGS 26303, in an experimental model of subarachnoid hemorrhage
-
Kwan AL, Bavbek M, Jeng AY, Maniara W, Toyoda T, Lappe RW, Kassell NF, Lee KS: Prevention and reversal of cerebral vasospasm by an endothelin-converting enzyme inhibitor, CGS 26303, in an experimental model of subarachnoid hemorrhage. J Neurosurg (1997) 87:281-286.
-
(1997)
J Neurosurg
, vol.87
, pp. 281-286
-
-
Kwan, A.L.1
Bavbek, M.2
Jeng, A.Y.3
Maniara, W.4
Toyoda, T.5
Lappe, R.W.6
Kassell, N.F.7
Lee, K.S.8
-
82
-
-
0032481287
-
Novel selective quinazoline inhibitors of endothelin converting enzyme-1
-
Ahn K, Sisneros AM, Herman SB, Pan SM, Hupe D, Lee C, Nikam S, Cheng XM, Doherty AM, Schroeder RL, Haleen SJ, Kaw S, Emoto N, Yanagisawa M: Novel selective quinazoline inhibitors of endothelin converting enzyme-1. Biochem Biophys Res Commun (1998) 243:184-190.
-
(1998)
Biochem Biophys Res Commun
, vol.243
, pp. 184-190
-
-
Ahn, K.1
Sisneros, A.M.2
Herman, S.B.3
Pan, S.M.4
Hupe, D.5
Lee, C.6
Nikam, S.7
Cheng, X.M.8
Doherty, A.M.9
Schroeder, R.L.10
Haleen, S.J.11
Kaw, S.12
Emoto, N.13
Yanagisawa, M.14
-
83
-
-
15144355006
-
B-90063, a novel endothelin converting enzyme inhibitor isolated from a new marine bacterium, Blastobacter sp. SANK 71894
-
Takaishi S, Tuchiya N, Sato A, Negishi T, Takamatsu Y, Malsushita Y, Watanabe T, Iijima Y, Haruyama H, Kinoshita T, Tanaka M, Kodama K.: B-90063, a novel endothelin converting enzyme inhibitor isolated from a new marine bacterium, Blastobacter sp. SANK 71894. J Antibiot (1998) 51:805-815.
-
(1998)
J Antibiot
, vol.51
, pp. 805-815
-
-
Takaishi, S.1
Tuchiya, N.2
Sato, A.3
Negishi, T.4
Takamatsu, Y.5
Malsushita, Y.6
Watanabe, T.7
Iijima, Y.8
Haruyama, H.9
Kinoshita, T.10
Tanaka, M.11
Kodama, K.12
-
84
-
-
0032498249
-
Phosphoramidon, an inhibitor of endothelin-converting enzyme, prevents indomethacin-induced gastric mucosal damage in rats
-
Matsumaru K, Kashimura H, Hassan M, Nakahara A, Goto K, Fukutomi H, Muto H, Tanaka N: Phosphoramidon, an inhibitor of endothelin-converting enzyme, prevents indomethacin-induced gastric mucosal damage in rats. Life Sci (1998) 62:PL79-84.
-
(1998)
Life Sci
, vol.62
-
-
Matsumaru, K.1
Kashimura, H.2
Hassan, M.3
Nakahara, A.4
Goto, K.5
Fukutomi, H.6
Muto, H.7
Tanaka, N.8
-
85
-
-
0030048610
-
RES-1149-1 and 2, novel non-peptidic type B receptor produced by Aspergillus sp. I. Taxonomy of producing strain, fermentation, isolation and physico-chemical and biological properties
-
Ogawa T, Ando K, Tanaka T, Uosaki Y, Matsuda Y: RES-1149-1 and 2, novel non-peptidic type B receptor produced by Aspergillus sp. I. Taxonomy of producing strain, fermentation, isolation and physico-chemical and biological properties. J Antibiot (1996) 49:1-5.
-
(1996)
J Antibiot
, vol.49
, pp. 1-5
-
-
Ogawa, T.1
Ando, K.2
Tanaka, T.3
Uosaki, Y.4
Matsuda, Y.5
-
86
-
-
0028350179
-
RES-701-1, a novel and selective endothelin type B receptor antagonist produced by Streptomyces sp. RE-701. II. Determination of the primary sequence
-
Yamasaki M, Yano K, Yoshida M, Matsuda Y, Yamaguchi K: RES-701-1, a novel and selective endothelin type B receptor antagonist produced by Streptomyces sp. RE-701. II. Determination of the primary sequence. J Antibiot (1994) 47:276-280.
-
(1994)
J Antibiot
, vol.47
, pp. 276-280
-
-
Yamasaki, M.1
Yano, K.2
Yoshida, M.3
Matsuda, Y.4
Yamaguchi, K.5
-
87
-
-
0028220239
-
RES-701-1, a novel and selective endothelin type B receptor antagonist produced by Streptomyces sp. RE-701. I. Characterization of producing strain, fermentation, isolation, physico-chemical and biological properties
-
Morishita Y, Chiba S, Tsukuda E, Tanaka T, Ogawa T, Yamasaki M, Yoshida M, Kawamoto I, Matsuda Y: RES-701-1, a novel and selective endothelin type B receptor antagonist produced by Streptomyces sp. RE-701. I. Characterization of producing strain, fermentation, isolation, physico-chemical and biological properties. J Antibiot (1994) 47:269-275.
-
(1994)
J Antibiot
, vol.47
, pp. 269-275
-
-
Morishita, Y.1
Chiba, S.2
Tsukuda, E.3
Tanaka, T.4
Ogawa, T.5
Yamasaki, M.6
Yoshida, M.7
Kawamoto, I.8
Matsuda, Y.9
-
88
-
-
8944221184
-
Novel drimane sesquiterpene esters from Aspergillus ustus var. pseudodeflectus with endothelin receptor binding activity
-
Hayes MA, Wrigley SK, Chetland I, Reynolds EE, Ainsworth AM, Renno DV, Latif MA, Cheng XM, Hupe DJ, Charlton P, Doherty AM: Novel drimane sesquiterpene esters from Aspergillus ustus var. pseudodeflectus with endothelin receptor binding activity. J Antibiot (1996) 49:505-512.
-
(1996)
J Antibiot
, vol.49
, pp. 505-512
-
-
Hayes, M.A.1
Wrigley, S.K.2
Chetland, I.3
Reynolds, E.E.4
Ainsworth, A.M.5
Renno, D.V.6
Latif, M.A.7
Cheng, X.M.8
Hupe, D.J.9
Charlton, P.10
Doherty, A.M.11
-
89
-
-
0030048611
-
RES-1149-1 and -2, novel non-peptidic endothelin type B receptor antagonists produced by Aspergillus sp. II. Structure determination and derivatization
-
Uosaki Y, Yoshida M, Ogawa T, Saitoh Y: RES-1149-1 and -2, novel non-peptidic endothelin type B receptor antagonists produced by Aspergillus sp. II. Structure determination and derivatization. J Antibiot (1996) 49:6-12.
-
(1996)
J Antibiot
, vol.49
, pp. 6-12
-
-
Uosaki, Y.1
Yoshida, M.2
Ogawa, T.3
Saitoh, Y.4
-
90
-
-
0026499039
-
Asterric acid, a new endothelin binding inhibitor
-
Ohashi H, Akiyama H, Nishikori K, Mochizuki J: Asterric acid, a new endothelin binding inhibitor. J Antibiot (1992) 45:1684-1685.
-
(1992)
J Antibiot
, vol.45
, pp. 1684-1685
-
-
Ohashi, H.1
Akiyama, H.2
Nishikori, K.3
Mochizuki, J.4
-
91
-
-
0029965387
-
Novel spirodihydrobenzofuranlactams as antagonists of endothelin and as inhibitors of HIV-1 protease produced by Stachybotrys sp. II. Structure determination
-
Roggo BE, Hug P, Moss S, stampfli A, Kriemler HP, Pater HH: Novel spirodihydrobenzofuranlactams as antagonists of endothelin and as inhibitors of HIV-1 protease produced by Stachybotrys sp. II. Structure determination. J Antibiot (1996) 49:374-379.
-
(1996)
J Antibiot
, vol.49
, pp. 374-379
-
-
Roggo, B.E.1
Hug, P.2
Moss, S.3
Stampfli, A.4
Kriemler, H.P.5
Pater, H.H.6
-
92
-
-
0028867063
-
Azphilones with endothelin receptor binding activity produced by Penicillium sclerotiorum: Taxonomy, fermentation, structure elucidation and biological activity
-
Pairet L, Wrigley SK, Chetland I, Reynolds EE, Hayes MA, Holloway J, Ainsworth AM, Katzer W, Cheng XM, Hupe DJ: Azphilones with endothelin receptor binding activity produced by Penicillium sclerotiorum: Taxonomy, fermentation, structure elucidation and biological activity. J Antibiot (1995) 48:913-923.
-
(1995)
J Antibiot
, vol.48
, pp. 913-923
-
-
Pairet, L.1
Wrigley, S.K.2
Chetland, I.3
Reynolds, E.E.4
Hayes, M.A.5
Holloway, J.6
Ainsworth, A.M.7
Katzer, W.8
Cheng, X.M.9
Hupe, D.J.10
-
93
-
-
0029613837
-
RES-1214-1 and -2, novel non-peptidic endothelin type a receptor antagonists produced by Pestalotiopsis sp
-
Ogawa T, Ando K, Aotani Y, Shinoda K, Tanaka T, Tsukuda E, Yishida M, Matsuda Y: RES-1214-1 and -2, novel non-peptidic endothelin type A receptor antagonists produced by Pestalotiopsis sp. J Antibiot (1995) 48:1401-1406.
-
(1995)
J Antibiot
, vol.48
, pp. 1401-1406
-
-
Ogawa, T.1
Ando, K.2
Aotani, Y.3
Shinoda, K.4
Tanaka, T.5
Tsukuda, E.6
Yishida, M.7
Matsuda, Y.8
-
94
-
-
0028241416
-
Aselacins, novel compounds that inhibit binding of endothelin to its receptor. I. the producing organism, fermentation and biological activity
-
Jackson M, Burres NS, Karwowski JP, Alder LA, Humphrey PE, Kohl WL, McAlpine JB: Aselacins, novel compounds that inhibit binding of endothelin to its receptor. I. The producing organism, fermentation and biological activity. J Antibiot (1994) 47:523-527.
-
(1994)
J Antibiot
, vol.47
, pp. 523-527
-
-
Jackson, M.1
Burres, N.S.2
Karwowski, J.P.3
Alder, L.A.4
Humphrey, P.E.5
Kohl, W.L.6
McAlpine, J.B.7
-
95
-
-
0028308270
-
Aselacins, novel compounds that inhibit binding of endothelin to its receptor. I. Isolation and elucidation of structures
-
Hochlowski JF Hill P, Whittem DN, Scherr MH, Rasmussen RR, Dorwin SA, McAlpine JB: Aselacins, novel compounds that inhibit binding of endothelin to its receptor. I. Isolation and elucidation of structures. J Antibiot (1994) 47:528-535.
-
(1994)
J Antibiot
, vol.47
, pp. 528-535
-
-
Hochlowski, J.F.1
Hill, P.2
Whittem, D.N.3
Scherr, M.H.4
Rasmussen, R.R.5
Dorwin, S.A.6
McAlpine, J.B.7
-
96
-
-
0028240445
-
WS79089A, B and C, new endothelin converting enzyme inhibitors isolated from Streptosporangium roseum. No. 79089. Taxonomy, fermentation, isolation, physico-chemical properties and biological activities
-
Tsurumi Y, Ohhata N, Iwamoto T, Shigematsu K, Nishikawa M, Kiyoto S, Okuhara M: WS79089A, B and C, new endothelin converting enzyme inhibitors isolated from Streptosporangium roseum. No. 79089. Taxonomy, fermentation, isolation, physico-chemical properties and biological activities. J Antibiot (1994) 47:619-630.
-
(1994)
J Antibiot
, vol.47
, pp. 619-630
-
-
Tsurumi, Y.1
Ohhata, N.2
Iwamoto, T.3
Shigematsu, K.4
Nishikawa, M.5
Kiyoto, S.6
Okuhara, M.7
-
97
-
-
0028825317
-
WS75624 a and B, new endothelin converting enzyme inhibitors isolated from Saccharothrix sp. I. Taxonomy, fermentation, isolation, physico-chemical properties and biological activities
-
Tsurumi Y, Ueda H, Hayashi K, Takase S, Nishikawa M, Kiyoto S, Okuhara M: WS75624 A and B, new endothelin converting enzyme inhibitors isolated from Saccharothrix sp. I. Taxonomy, fermentation, isolation, physico-chemical properties and biological activities. J Antibiot (1995) 48:1066-1072.
-
(1995)
J Antibiot
, vol.48
, pp. 1066-1072
-
-
Tsurumi, Y.1
Ueda, H.2
Hayashi, K.3
Takase, S.4
Nishikawa, M.5
Kiyoto, S.6
Okuhara, M.7
-
98
-
-
13344250468
-
Endothelin receptor antagonist triterpenoid, myriceric acid A, isolated from Myrica cerifera and structure activity relationships of its derivatives
-
Sakurawa K, Yasuda F, Tozyo T, Nakamura M, Sato T, Kikuchi J, Terui Y, Ikenishi Y, Iwata T, Takahashi K, Konoike T, Mihara S, Fujimoto M: Endothelin receptor antagonist triterpenoid, myriceric acid A, isolated from Myrica cerifera and structure activity relationships of its derivatives. Chem Pharm Bull (1996) 44:343-351.
-
(1996)
Chem Pharm Bull
, vol.44
, pp. 343-351
-
-
Sakurawa, K.1
Yasuda, F.2
Tozyo, T.3
Nakamura, M.4
Sato, T.5
Kikuchi, J.6
Terui, Y.7
Ikenishi, Y.8
Iwata, T.9
Takahashi, K.10
Konoike, T.11
Mihara, S.12
Fujimoto, M.13
-
99
-
-
0030975485
-
Daleformis, a new phytoalexin from the roots of Dalea filiciformis: An inhibitor of endothelin converting enzyme
-
Patil AD, Freyer AJ, Eggleston DS, Haltiwanger RC, Tomcowicz B, Breen A, Johnson RK: Daleformis, a new phytoalexin from the roots of Dalea filiciformis: an inhibitor of endothelin converting enzyme. J Nat Products (1997) 60:306-308.
-
(1997)
J Nat Products
, vol.60
, pp. 306-308
-
-
Patil, A.D.1
Freyer, A.J.2
Eggleston, D.S.3
Haltiwanger, R.C.4
Tomcowicz, B.5
Breen, A.6
Johnson, R.K.7
-
100
-
-
0027420795
-
Isolation and structure elucidation of 3,4-sulfatobastadin 13, an inhibitor of the endothelin a receptor, from a sponge of the genus Ianthella
-
Gulavita NK, Wright AE, McCarthy PJ, Pomponi SA, Kelly-Borges M, Chin M, Sills MA: Isolation and structure elucidation of 3,4-sulfatobastadin 13, an inhibitor of the endothelin A receptor, from a sponge of the genus Ianthella. J Nat Products (1993) 56:1613-1617.
-
(1993)
J Nat Products
, vol.56
, pp. 1613-1617
-
-
Gulavita, N.K.1
Wright, A.E.2
McCarthy, P.J.3
Pomponi, S.A.4
Kelly-Borges, M.5
Chin, M.6
Sills, M.A.7
-
101
-
-
0029950814
-
Halistanol disulfate B, a novel sulfated sterol from the sponge Pachastrelaa sp: Inhibitor of endothelin converting enzyme
-
Patil AD, Freyer AJ, Breen A, Carte B, Johnson RK: Halistanol disulfate B, a novel sulfated sterol from the sponge Pachastrelaa sp: inhibitor of endothelin converting enzyme. J Nat Products (1996) 59:606-608.
-
(1996)
J Nat Products
, vol.59
, pp. 606-608
-
-
Patil, A.D.1
Freyer, A.J.2
Breen, A.3
Carte, B.4
Johnson, R.K.5
-
102
-
-
0032124784
-
Nahocols and isonahocols, endothelin antagonists from the brown alga, Sargassum automnale
-
Tsuchiya N, Sato A, Haruyama H, Watanabe T, Iijima Y: Nahocols and isonahocols, endothelin antagonists from the brown alga, Sargassum automnale. Phytochemistry (1998) 48:1003-1011.
-
(1998)
Phytochemistry
, vol.48
, pp. 1003-1011
-
-
Tsuchiya, N.1
Sato, A.2
Haruyama, H.3
Watanabe, T.4
Iijima, Y.5
|