-
1
-
-
69949174478
-
Has the era of untreatable infections arrived?
-
Livermore, D.M. Has the era of untreatable infections arrived? J. Antimicrob. Chemother. 2009, 64 (Suppl. 1), i29–i36. [CrossRef] [PubMed]
-
(2009)
J. Antimicrob. Chemother.
, vol.64
, pp. i29-i36
-
-
Livermore, D.M.1
-
2
-
-
85019749032
-
Synthesis and antibacterial evaluation of novel 3-substituted ocotillol-type derivatives as leads
-
Bi, Y.; Liu, X.X.; Zhang, H.Y.; Yang, X.; Liu, Z.Y.; Lu, J.; Lewis, P.J.; Wang, C.Z.; Xu, J.Y.; Meng, Q.G.; et al. Synthesis and Antibacterial Evaluation of Novel 3-Substituted Ocotillol-Type Derivatives as Leads. Molecules 2017, 22, 590. [CrossRef] [PubMed]
-
(2017)
Molecules
, vol.22
, pp. 590
-
-
Bi, Y.1
Liu, X.X.2
Zhang, H.Y.3
Yang, X.4
Liu, Z.Y.5
Lu, J.6
Lewis, P.J.7
Wang, C.Z.8
Xu, J.Y.9
Meng, Q.G.10
-
3
-
-
84944618155
-
Usa300 methicillin-resistant staphylococcus aureus, United States, 2000–2013
-
Carrel, M.; Perencevich, E.N.; David, M.Z. USA300 Methicillin-Resistant Staphylococcus aureus, United States, 2000–2013. Emerg. Infect. Dis. 2015, 21, 1973–1980. [CrossRef] [PubMed]
-
(2015)
Emerg. Infect. Dis.
, vol.21
, pp. 1973-1980
-
-
Carrel, M.1
Perencevich, E.N.2
David, M.Z.3
-
4
-
-
84861205652
-
China takes aim at rampant antibiotic resistance
-
Public health
-
Hvistendahl, M. Public health. China takes aim at rampant antibiotic resistance. Science 2012, 336, 795. [CrossRef] [PubMed]
-
(2012)
Science
, vol.336
, pp. 795
-
-
Hvistendahl, M.1
-
5
-
-
84867402030
-
Antibiotic resistance amongst healthcare-associated pathogens in China
-
Yezli, S.; Li, H. Antibiotic resistance amongst healthcare-associated pathogens in China. Int. J. Antimicrob. Agents 2012, 40, 389–397. [CrossRef] [PubMed]
-
(2012)
Int. J. Antimicrob. Agents
, vol.40
, pp. 389-397
-
-
Yezli, S.1
Li, H.2
-
6
-
-
84927674621
-
Liposomes as novel anti-infectives targeting bacterial virulence factors?
-
Azeredo da Silveira, S.; Perez, A. Liposomes as novel anti-infectives targeting bacterial virulence factors? Expert. Rev. Anti-Infect. Ther. 2015, 13, 531–533. [CrossRef] [PubMed]
-
(2015)
Expert. Rev. Anti-infect. Ther.
, vol.13
, pp. 531-533
-
-
Azeredo da Silveira, S.1
Perez, A.2
-
7
-
-
84911480620
-
Antiadhesion agents against gram-positive pathogens
-
Cascioferro, S.; Cusimano, M.G.; Schillaci, D. Antiadhesion agents against Gram-positive pathogens. Future Microbiol. 2014, 9, 1209–1220. [CrossRef] [PubMed]
-
(2014)
Future Microbiol
, vol.9
, pp. 1209-1220
-
-
Cascioferro, S.1
Cusimano, M.G.2
Schillaci, D.3
-
8
-
-
84893816415
-
Development of quorum-based anti-virulence therapeutics targeting gram negative bacterial pathogens
-
Tay, S.B.; Yew, W.S. Development of quorum-based anti-virulence therapeutics targeting Gram negative bacterial pathogens. Int. J. Mol. Sci. 2013, 14, 16570–16599. [CrossRef] [PubMed]
-
(2013)
Int. J. Mol. Sci.
, vol.14
, pp. 16570-16599
-
-
Tay, S.B.1
Yew, W.S.2
-
10
-
-
84878278251
-
Infectious diseases society of america. 10 x '20 progress–development of new drugs active against gram-negative bacilli: an update from the infectious diseases society of america
-
Boucher, H.W.; Talbot, G.H.; Benjamin, D.K.; Bradley, J.; Guidos, R.J.; Jones, R.N.; Murray, B.E.; Bonomo, R.A.; Gilbert, D. Infectious Diseases Society of America. 10 x '20 Progress–development of new drugs active against gram-negative bacilli: an update from the Infectious Diseases Society of America. Clin. Infect. Dis. 2013, 56, 1685–1694. [CrossRef] [PubMed]
-
(2013)
Clin. Infect. Dis.
, vol.56
, pp. 1685-1694
-
-
Boucher, H.W.1
Talbot, G.H.2
Benjamin, D.K.3
Bradley, J.4
Guidos, R.J.5
Jones, R.N.6
Murray, B.E.7
Bonomo, R.A.8
Gilbert, D.9
-
11
-
-
85014117063
-
Synthesis of extended conjugated indolyl chalcones as potent anti-breast cancer, anti-inflammatory and antioxidant agents
-
Bhale, P.S.; Chavan, H.V.; Dongare, S.B.; Shringare, S.N.; Mule, Y.B.; Nagane, S.S.; Bandgar, B.P. Synthesis of extended conjugated indolyl chalcones as potent anti-breast cancer, anti-inflammatory and antioxidant agents. Bioorg. Med. Chem. Lett. 2017, 27, 1502–1507. [CrossRef] [PubMed]
-
(2017)
Bioorg. Med. Chem. Lett.
, vol.27
, pp. 1502-1507
-
-
Bhale, P.S.1
Chavan, H.V.2
Dongare, S.B.3
Shringare, S.N.4
Mule, Y.B.5
Nagane, S.S.6
Bandgar, B.P.7
-
12
-
-
85017201451
-
Synthesis and biological evaluation of novel indole-pyrimidine hybrids bearing morpholine and thiomorpholine moieties
-
Diao, P.C.; Li, Q.; Hu, M.J.; Ma, Y.F.; You, W.W.; Hong, K.H.; Zhao, P.L. Synthesis and biological evaluation of novel indole-pyrimidine hybrids bearing morpholine and thiomorpholine moieties. Eur. J. Med. Chem. 2017, 13, 110–118. [CrossRef] [PubMed]
-
(2017)
Eur. J. Med. Chem.
, vol.13
, pp. 110-118
-
-
Diao, P.C.1
Li, Q.2
Hu, M.J.3
Ma, Y.F.4
You, W.W.5
Hong, K.H.6
Zhao, P.L.7
-
13
-
-
85021121982
-
Novel indole-based tambjamine-analogues induce apoptotic lung cancer cell death through p38 mitogen-activated protein kinase activation
-
in press
-
Manuel-Manresa, P.; Korrodi-Gregório, L.; Hernando, E.; Villanueva, A.; Martínez-García, D.; Rodilla, A.M.; Ramos, R.; Fardilha, M.; Moya, J.; Quesada, R.; et al. Novel indole-based tambjamine-analogues induce apoptotic lung cancer cell death through p38 mitogen-activated protein kinase activation. Mol. Cancer. Ther. 2017, in press. [CrossRef] [PubMed]
-
(2017)
Mol. Cancer. Ther.
-
-
Manuel-Manresa, P.1
Korrodi-Gregório, L.2
Hernando, E.3
Villanueva, A.4
Martínez-García, D.5
Rodilla, A.M.6
Ramos, R.7
Fardilha, M.8
Moya, J.9
Quesada, R.10
-
14
-
-
84993965476
-
Synthesis and evaluation of novel hybrids ?-carboline-4-thiazolidinones as potential antitumor and antiviral agents
-
Barbosa, V.A.; Baréa, P.; Mazia, R.S.; Ueda-Nakamura, T.; Costa, W.F.; Foglio, M.A.; Goes Ruiz, A.L.; Carvalho, J.E.; Vendramini-Costa, D.B.; Nakamura, C.V.; et al. Synthesis and evaluation of novel hybrids ?-carboline-4-thiazolidinones as potential antitumor and antiviral agents. Eur. J. Med. Chem. 2016, 124, 1093–1104. [CrossRef] [PubMed]
-
(2016)
Eur. J. Med. Chem.
, vol.124
, pp. 1093-1104
-
-
Barbosa, V.A.1
Baréa, P.2
Mazia, R.S.3
Ueda-Nakamura, T.4
Costa, W.F.5
Foglio, M.A.6
Goes Ruiz, A.L.7
Carvalho, J.E.8
Vendramini-Costa, D.B.9
Nakamura, C.V.10
-
15
-
-
85018423823
-
Antibacterial and anti-tubercular evaluation of dihydronaphthalenone-indole hybrid analogues
-
in press
-
Kumar, V.P.; Renjitha, J.; Salfeena, C.F.; Ashitha, K.T.; Keri, R.S.; Varughese, S.; Sasidhar, B.S. Antibacterial and anti-tubercular evaluation of Dihydronaphthalenone-indole hybrid analogues. Chem. Biol. Drug. Des. 2017, in press. [CrossRef]
-
(2017)
Chem. Biol. Drug. Des.
-
-
Kumar, V.P.1
Renjitha, J.2
Salfeena, C.F.3
Ashitha, K.T.4
Keri, R.S.5
Varughese, S.6
Sasidhar, B.S.7
-
16
-
-
85016459322
-
Medicinal applications of (benz)imidazole- and indole-based macrocycles
-
Patil, S.A.; Patil, S.A.; Patil, R. Medicinal applications of (benz)imidazole- and indole-based macrocycles. Chem. Biol. Drug. Des. 2017, 89, 639–649. [CrossRef] [PubMed]
-
(2017)
Chem. Biol. Drug. Des.
, vol.89
, pp. 639-649
-
-
Patil, S.A.1
Patil, S.A.2
Patil, R.3
-
17
-
-
85010426169
-
Identification of 5-methoxy-2-(diformylmethylidene)-3,3-dimethylindole as an anti-influenza a virus agent
-
Tan, M.C.; Wong, W.Y.; Ng, W.L.; Yeo, K.S.; Mohidin, T.B.; Lim, Y.Y.; Lafta, F.; Mohd Ali, H.; Ea, C.K. Identification of 5-Methoxy-2-(Diformylmethylidene)-3,3-Dimethylindole as an Anti-Influenza A Virus Agent. PLoS ONE 2017, 12, e0170352. [CrossRef] [PubMed]
-
(2017)
Plos ONE
, vol.12
, pp. e0170352
-
-
Tan, M.C.1
Wong, W.Y.2
Ng, W.L.3
Yeo, K.S.4
Mohidin, T.B.5
Lim, Y.Y.6
Lafta, F.7
Mohd Ali, H.8
Ea, C.K.9
-
18
-
-
85006489409
-
Discovery of novel multi-target indole-based derivatives as potent and selective inhibitors of chikungunya virus replication
-
Scuotto, M.; Abdelnabi, R.; Collarile, S.; Schiraldi, C.; Delang, L.; Massa, A.; Ferla, S.; Brancale, A.; Leyssen, P.; Neyts, J.; et al. Discovery of novel multi-target indole-based derivatives as potent and selective inhibitors of chikungunya virus replication. Bioorg. Med. Chem. 2017, 25, 327–337. [CrossRef] [PubMed]
-
(2017)
Bioorg. Med. Chem.
, vol.25
, pp. 327-337
-
-
Scuotto, M.1
Abdelnabi, R.2
Collarile, S.3
Schiraldi, C.4
Delang, L.5
Massa, A.6
Ferla, S.7
Brancale, A.8
Leyssen, P.9
Neyts, J.10
-
19
-
-
84974794716
-
Synthesis and in vitro anti-HIV-1 activity of a series of n-arylsulfonyl-3-propionylindoles.
-
Che, Z.; Tian, Y.; Hu, Z.; Chen, Y.; Liu, S.; Chen, G. Synthesis and in vitro anti-HIV-1 activity of a series of N-arylsulfonyl-3-propionylindoles. Z. Naturforsch. C 2016, 71, 105–109. [CrossRef] [PubMed]
-
(2016)
Z. Naturforsch. C
, vol.71
, pp. 105-109
-
-
Che, Z.1
Tian, Y.2
Hu, Z.3
Chen, Y.4
Liu, S.5
Chen, G.6
-
20
-
-
12444315080
-
Novel indolyl aryl sulfones active against HIV-1 carrying NNRTI resistance mutations: Synthesis and sar studies
-
Silvestri, R.; De Martino, G.; La Regina, G.; Artico, M.; Massa, S.; Vargiu, L.; Mura, M.; Loi, A.G.; Marceddu, T.; La Colla, P. Novel indolyl aryl sulfones active against HIV-1 carrying NNRTI resistance mutations: Synthesis and SAR studies. J. Med. Chem. 2003, 46, 2482–2493. [CrossRef] [PubMed]
-
(2003)
J. Med. Chem.
, vol.46
, pp. 2482-2493
-
-
Silvestri, R.1
De Martino, G.2
La Regina, G.3
Artico, M.4
Massa, S.5
Vargiu, L.6
Mura, M.7
Loi, A.G.8
Marceddu, T.9
La Colla, P.10
-
21
-
-
84983315315
-
Extended N-Arylsulfonylindoles as 5-HT6 receptor antagonists: Design, synthesis & amp; biological evaluation
-
Vera, G.; Lagos, C.F.; Almendras, S.; Hebel, D.; Flores, F.; Valle-Corvalán, G.; Pessoa-Mahana, C.D.; Mella-Raipán, J.; Montecinos, R.; Recabarren-Gajardo, G. Extended N-Arylsulfonylindoles as 5-HT6 Receptor Antagonists: Design, Synthesis & amp; Biological Evaluation. Molecules 2016, 21, 1070.
-
(2016)
Molecules
, vol.21
, pp. 1070
-
-
Vera, G.1
Lagos, C.F.2
Almendras, S.3
Hebel, D.4
Flores, F.5
Valle-Corvalán, G.6
Pessoa-Mahana, C.D.7
Mella-Raipán, J.8
Montecinos, R.9
Recabarren-Gajardo, G.10
-
22
-
-
68149103322
-
Anti human immunodeficiency virus-1 (HIV-1) agents 3. Synthesis and in vitro anti-HIV-1 activity of some n-arylsulfonylindoles
-
Fan, L.L.; Liu, W.Q.; Xu, H.; Yang, L.M.; Lv, M.; Zheng, Y.T. Anti human immunodeficiency virus-1 (HIV-1) agents 3. synthesis and in vitro anti-HIV-1 activity of some N-arylsulfonylindoles. Chem. Pharm. Bull. (Tokyo) 2009, 57, 797–800. [CrossRef] [PubMed]
-
(2009)
Chem. Pharm. Bull. (Tokyo)
, vol.57
, pp. 797-800
-
-
Fan, L.L.1
Liu, W.Q.2
Xu, H.3
Yang, L.M.4
Lv, M.5
Zheng, Y.T.6
-
23
-
-
78549254120
-
Antifungal agents. Part 5: synthesis and antifungal activities of aminoguanidine derivatives of N-arylsulfonyl-3-acylindoles
-
Xu, H.; Wang, Y.Y. Antifungal agents. Part 5: Synthesis and antifungal activities of aminoguanidine derivatives of N-arylsulfonyl-3-acylindoles. Bioorg. Med. Chem. Lett. 2010, 20, 7274–7277. [CrossRef] [PubMed]
-
(2010)
Bioorg. Med. Chem. Lett.
, vol.20
, pp. 7274-7277
-
-
Xu, H.1
Wang, Y.Y.2
-
24
-
-
84907057145
-
Synthesis and biological evaluation of (E)-1-(substituted)-3-phenylprop-2-en-1-ones bearing rhodanines as potent antimicrobial agents
-
Song, M.X.; Deng, X.Q.; Li, Y.R.; Zheng, C.J.; Hong, L.; Piao, H.R. Synthesis And biological evaluation of (E)-1-(substituted)-3-phenylprop-2-en-1-ones bearing rhodanines as potent antimicrobial agents. J. Enzym. Inhib. Med. Chem. 2014, 29, 647–653. [CrossRef] [PubMed]
-
(2014)
J. Enzym. Inhib. Med. Chem.
, vol.29
, pp. 647-653
-
-
Song, M.X.1
Deng, X.Q.2
Li, Y.R.3
Zheng, C.J.4
Hong, L.5
Piao, H.R.6
-
25
-
-
85008972630
-
The synthesis and anti-bacterial activities of N-carboxymethyl rhodanines
-
Song, M.X.; Zheng, C.J.; Deng, X.Q.; Wei, Z.Y.; Piao, H.R. The Synthesis and Anti-Bacterial Activities of N-carboxymethyl Rhodanines. Med. Chem. 2014, 4, 441–448.
-
(2014)
Med. Chem.
, vol.4
, pp. 441-448
-
-
Song, M.X.1
Zheng, C.J.2
Deng, X.Q.3
Wei, Z.Y.4
Piao, H.R.5
-
26
-
-
84872119409
-
Synthesis and antibacterial evaluation of rhodanine-based 5-aryloxy pyrazoles against selected methicillin resistant and quinolone-resistant staphylococcus aureus (MRSA and QRSA)
-
Song, M.X.; Zheng, C.J.; Sun, L.P.; Wu, Y.; Hong, L.; Li, Y.J.; Liu, Y.; Wei, Z.Y.; Jin, M.J.; Piao, H.R. Synthesis and antibacterial evaluation of rhodanine-based 5-aryloxy pyrazoles against selected methicillin resistant and quinolone-resistant Staphylococcus aureus (MRSA and QRSA). Eur. J. Med. Chem. 2013, 60, 376–385. [CrossRef] [PubMed]
-
(2013)
Eur. J. Med. Chem.
, vol.60
, pp. 376-385
-
-
Song, M.X.1
Zheng, C.J.2
Sun, L.P.3
Wu, Y.4
Hong, L.5
Li, Y.J.6
Liu, Y.7
Wei, Z.Y.8
Jin, M.J.9
Piao, H.R.10
-
27
-
-
84864418734
-
Synthesis and bioactivity evaluation of rhodanine derivatives as potential anti-bacterial agents
-
Song, M.X.; Zheng, C.J.; Deng, X.Q.; Wang, Q.; Hou, S.P.; Liu, T.T.; Xing, X.L.; Piao, H.R. Synthesis and bioactivity evaluation of rhodanine derivatives as potential anti-bacterial agents. Eur. J. Med. Chem. 2012, 54, 403–412. [CrossRef] [PubMed]
-
(2012)
Eur. J. Med. Chem.
, vol.54
, pp. 403-412
-
-
Song, M.X.1
Zheng, C.J.2
Deng, X.Q.3
Wang, Q.4
Hou, S.P.5
Liu, T.T.6
Xing, X.L.7
Piao, H.R.8
-
28
-
-
84869096131
-
Synthesis and biological evaluation of 5-aryloxypyrazole derivatives bearing a rhodanine-3-aromatic acid as potential antimicrobial agents
-
Zheng, C.J.; Song, M.X.; Sun, L.P.; Wu, Y.; Hong, L.; Piao, H.R. Synthesis and biological evaluation of 5-aryloxypyrazole derivatives bearing a rhodanine-3-aromatic acid as potential antimicrobial agents. Bioorg. Med. Chem. Lett. 2012, 22, 7024–7028. [CrossRef] [PubMed]
-
(2012)
Bioorg. Med. Chem. Lett.
, vol.22
, pp. 7024-7028
-
-
Zheng, C.J.1
Song, M.X.2
Sun, L.P.3
Wu, Y.4
Hong, L.5
Piao, H.R.6
-
29
-
-
84865961097
-
Synthesis and antimicrobial evaluation of l-phenylalanine-derived c5-substituted rhodanine and chalcone derivatives containing thiobarbituric acid or 2-thioxo-4-thiazolidinone
-
Jin, X.; Zheng, C.J.; Song, M.X.; Wu, Y.; Sun, L.P.; Li, Y.J.; Yu, L.J.; Piao, H.R. Synthesis and antimicrobial evaluation of L-phenylalanine-derived C5-substituted rhodanine and chalcone derivatives containing thiobarbituric acid or 2-thioxo-4-thiazolidinone. Eur. J. Med. Chem. 2012, 56, 203–209. [CrossRef] [PubMed]
-
(2012)
Eur. J. Med. Chem.
, vol.56
, pp. 203-209
-
-
Jin, X.1
Zheng, C.J.2
Song, M.X.3
Wu, Y.4
Sun, L.P.5
Li, Y.J.6
Yu, L.J.7
Piao, H.R.8
-
30
-
-
78649325633
-
Synthesis of new chalcone derivatives containing a rhodanine-3-acetic acid moiety with potential anti-bacterial activity
-
Chen, Z.H.; Zheng, C.J.; Sun, L.P.; Piao, H.R. Synthesis of new chalcone derivatives containing a rhodanine-3-acetic acid moiety with potential anti-bacterial activity. Eur. J. Med. Chem. 2010, 45, 5739–5743. [CrossRef] [PubMed]
-
(2010)
Eur. J. Med. Chem.
, vol.45
, pp. 5739-5743
-
-
Chen, Z.H.1
Zheng, C.J.2
Sun, L.P.3
Piao, H.R.4
|