Synthesis and antimicrobial evaluation of L-phenylalanine-derived C5-substituted rhodanine and chalcone derivatives containing thiobarbituric acid or 2-thioxo-4-thiazolidinone

European Journal of Medicinal Chemistry

Volumn 56, Issue , 2012, Pages 203-209

  Jin, Xin ^b   Zheng, Chang Ji ^a   Song, Ming Xia ^a   Wu, Yan ^a   Sun, Liang Peng ^a   Li, Yin Jing ^a   Yu, Li Jun ^b   Piao, Hu Ri ^a  

^a YANBIAN UNIVERSITY   (China)

^b INNER MONGOLIA UNIVERSITY FOR NATIONALITIES   (China)

Author keywords

Antibacterial activity; Chalcone; Phenylpropionic acid; Rhodanine; Thiobarbituric acid

Indexed keywords

2 [5 [4 [3 (NAPHTHALEN 2 YL) 3 OXOPROP 1 EN 1 YL]BENZYLIDENE] 4 OXO 2 THIOXOTHIAZOLIDIN 3 YL] 3 PHENYLPROPANOIC ACID; 4 THIAZOLIDINONE DERIVATIVE; CHALCONE DERIVATIVE; NORFLOXACIN; OXACILLIN; PHENYLALANINE DERIVATIVE; RHODANINE; THIOBARBITURIC ACID DERIVATIVE; UNCLASSIFIED DRUG;

ANTIMICROBIAL ACTIVITY; ARTICLE; BACTERIAL STRAIN; BACTERIUM ISOLATE; CONTROLLED STUDY; DRUG POTENCY; DRUG SYNTHESIS; GRAM NEGATIVE BACTERIUM; GRAM POSITIVE BACTERIUM; MINIMUM INHIBITORY CONCENTRATION; NONHUMAN; STAPHYLOCOCCUS AUREUS;

ANTI-BACTERIAL AGENTS; CHALCONE; DOSE-RESPONSE RELATIONSHIP, DRUG; MICROBIAL SENSITIVITY TESTS; MOLECULAR STRUCTURE; PHENYLALANINE; RHODANINE; STAPHYLOCOCCUS AUREUS; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLIDINES; THIOBARBITURATES;

EID: 84865961097     PISSN: 02235234     EISSN: 17683254     Source Type: Journal    
DOI: 10.1016/j.ejmech.2012.08.026     Document Type: Article

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