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MedChemComm

Volumn 6, Issue 7, 2015, Pages 1293-1302

Chromanones: selective and reversible monoamine oxidase B inhibitors with nanomolar potency

(6) Lan, Jin Shuai a Xie, Sai Sai a Huang, Ming a Hu, Ya Jian a Kong, Ling Yi a Wang, Xiao Bing a

a CHINA PHARMACEUTICAL UNIVERSITY (China)

Author keywords

[No Author keywords available]

Indexed keywords

2,2 DIMETHYL 7 [(3 METHYLBENZYL)OXY]CHROMAN 4 ONE; 2,2 DIMETHYL 7 [(4 METHYLBENZYL)OXY]CHROMAN 4 ONE; 4 CHROMANONE DERIVATIVE; 4 [[(2,2 DIMETHYL 4 OXOCHROMAN 7 YL)OXY]METHYL]BENZONITRILE; 6 (3 PHENYLPROPOXY)BENZOFURAN 3(2H) ONE; 6 (BENZYLOXY)BENZOFURAN 3(2H) ONE; 6 PHENETHOXYBENZOFURAN 3(2H) ONE; 7 (3 PHENYLPROPOXY)CHROMAN 4 ONE; 7 (BENZYLOXY) 2,2 DIMETHYLCHROMAN 4 ONE; 7 (BENZYLOXY)CHROMAN 4 ONE; 7 PHENETHOXYCHROMAN 4 ONE; 7 [(2 FLUOROBENZYL)OXY] 2,2 DIMETHYLCHROMAN 4 ONE; 7 [(2 FLUOROBENZYL)OXY]CHROMAN 4 ONE; 7 [(3 BROMOBENZYL)OXY] 2,2 DIMETHYLCHROMAN 4 ONE; 7 [(3 BROMOBENZYL)OXY]CHROMAN 4 ONE; 7 [(3 CHLOROBENZYL)OXY] 2,2 DIMETHYLCHROMAN 4 ONE; 7 [(3 CHLOROBENZYL)OXY]CHROMAN 4 ONE; 7 [(3 FLUOROBENZYL)OXY] 2,2 DIMETHYLCHROMAN 4 ONE; 7 [(3 FLUOROBENZYL)OXY]CHROMAN 4 ONE; 7 [(3 METHYLBENZYL)OXY]CHROMAN 4 ONE; 7 [(4 BROMOBENZYL)OXY] 2,2 DIMETHYLCHROMAN 4 ONE; 7 [(4 BROMOBENZYL)OXY]CHROMAN 4 ONE; 7 [(4 CHLOROBENZYL)OXY] 2,2 DIMETHYLCHROMAN 4 ONE; 7 [(4 CHLOROBENZYL)OXY]CHROMAN 4 ONE; 7 [(4 FLUOROBENZYL)OXY] 2,2 DIMETHYLCHROMAN 4 ONE; 7 [(4 FLUOROBENZYL)OXY]CHROMAN 4 ONE; 7 [(4 METHYLBENZYL)OXY]CHROMAN 4 ONE; 7 [[(4 OXOCHROMAN 7 YL)OXY]METHYL]BENZONITRILE; MONOAMINE OXIDASE B INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; BLOOD BRAIN BARRIER; CONTROLLED STUDY; DEGENERATIVE DISEASE; DRUG SYNTHESIS; ENZYME INHIBITION; IC50; IN VITRO STUDY; MOLECULAR DOCKING; NEUROTOXICITY; PHYSICAL CHEMISTRY; PRIORITY JOURNAL; STRUCTURE ACTIVITY RELATION;

EID: 84936882524 PISSN: 20402503 EISSN: 20402511 Source Type: Journal
DOI: 10.1039/c5md00124b Document Type: Article

Times cited : (22)

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