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MedChemComm

Volumn 5, Issue 12, 2014, Pages 1863-1870

3,5-Diamino-1,2,4-triazoles as a novel scaffold for potent, reversible LSD1 (KDM1A) inhibitors

(4) Kutz, Craig J a Holshouser, Steven L a Marrow, Ethan A a Woster, Patrick M a

a MEDICAL UNIVERSITY OF SOUTH CAROLINA (United States)

Author keywords

[No Author keywords available]

Indexed keywords

AMIDOXIME; AMINE OXIDASE (FLAVIN CONTAINING) ISOENZYME A; AMINE OXIDASE (FLAVIN CONTAINING) ISOENZYME B; CYCLOPEPTIDE; GUANAZOLE; HISTONE H3; LYSINE; LYSINE SPECIFIC DEMETHYLASE 1 INHIBITOR; N3 (2 CHLORO 6 PHENOXYBENZYL) 4H 1,2,4 TRIAZOLE 3,5 DIAMINE; N3,N5 BIS(2 METHOXYBENZYL) 1H 1,2,4 TRIAZOLE 3,5 DIAMINE; OXYGENASE INHIBITOR; THIOUREA DERIVATIVE; TRANYLCYPROMINE; UNCLASSIFIED DRUG; VERLINDAMYCIN;

ARTICLE; CELL DEATH; CONTROLLED STUDY; CYTOTOXICITY; DRUG IDENTIFICATION; DRUG STRUCTURE; DRUG SYNTHESIS; GENETIC TRANSCRIPTION; HUMAN; HUMAN CELL; IC50; IN VITRO STUDY; IN VIVO STUDY; MAMMAL CELL; TRANSCRIPTION INITIATION;

EID: 84911931554 PISSN: 20402503 EISSN: 20402511 Source Type: Journal
DOI: 10.1039/c4md00283k Document Type: Article

Times cited : (45)

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