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Bioorganic and Medicinal Chemistry Letters

Volumn 24, Issue 19, 2014, Pages 4638-4642

Synthesis, biological evaluation and docking analysis of 3-methyl-1-phenylchromeno[4,3-c]pyrazol-4(1H)-ones as potential cyclooxygenase-2 (COX-2) inhibitors

(4) Grover, Jagdeep a Kumar, Vivek a Sobhia, M Elizabeth a Jachak, Sanjay M a

a NATIONAL INSTITUTE OF PHARMACEUTICAL EDUCATION AND RESEARCH NIPER (India)

Author keywords

3 Methyl 1 phenylchromeno 4,3 c pyrazol; 4(1H) ones; Anti inflammatory; Cyclooxygenase 2; Molecular docking

Indexed keywords

3 METHYL 1 PHENYLCHROMENO[4,3 C]PYRAZOL 4(1H)ONE DERIVATIVE; CELECOXIB; CYCLOOXYGENASE 2 INHIBITOR; UNCLASSIFIED DRUG; 3-METHYL-1-(4-(TRIFLUOROMETHYL)PHENYLCHROMENO(4,3-C)PYRAZOL-4(1H)-ONE; CARRAGEENAN; COUMARIN DERIVATIVE; CYCLOOXYGENASE 2; NONSTEROID ANTIINFLAMMATORY AGENT; PYRAZOLE DERIVATIVE;

ANTIINFLAMMATORY ACTIVITY; ARTICLE; DRUG SYNTHESIS; EDEMA; IC50; MOLECULAR DOCKING; PAW EDEMA; STRUCTURE ACTIVITY RELATION; ANIMAL; CHEMICAL STRUCTURE; CHEMICALLY INDUCED; CHEMISTRY; DOSE RESPONSE; METABOLISM; RAT; SHEEP; SYNTHESIS;

ANIMALS; ANTI-INFLAMMATORY AGENTS, NON-STEROIDAL; CARRAGEENAN; COUMARINS; CYCLOOXYGENASE 2; CYCLOOXYGENASE 2 INHIBITORS; DOSE-RESPONSE RELATIONSHIP, DRUG; EDEMA; MOLECULAR DOCKING SIMULATION; MOLECULAR STRUCTURE; PYRAZOLES; RATS; SHEEP; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84907209878 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2014.08.050 Document Type: Article

Times cited : (24)

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