Interactions of endosulfan and methoxychlor involving CYP3A4 and CYP2B6 in human HepaRG cells

Drug Metabolism and Disposition

Volumn 42, Issue 8, 2014, Pages 1234-1240

  Savary, Camille C ^a   Jossé, Rozenn ^a   Bruyère, Arnaud ^b   Guillet, Fabrice ^b   Robin, Marie Anne ^a   Guillouzo, André ^a  

^a UNIVERSITÉ DE RENNES 1   (France)

^b Xenoblis   (France)

Author keywords

[No Author keywords available]

Indexed keywords

CONSTITUTIVE ANDROSTANE RECEPTOR; CYTOCHROME P450 2B6; CYTOCHROME P450 3A4; ENDOSULFAN; MESSENGER RNA; METHOXYCHLOR; ORGANOCHLORINE PESTICIDE; PREGNANE X RECEPTOR; CELL RECEPTOR; CYP2B6 PROTEIN, HUMAN; CYP3A4 PROTEIN, HUMAN; CYTOCHROME P450 3A; PESTICIDE; STEROID RECEPTOR;

ARTICLE; CELL VIABILITY; CHEMICAL INTERACTION; CONCENTRATION (PARAMETERS); CYTOTOXICITY; ENZYME ACTIVITY; ENZYME INHIBITION; HUMAN; HUMAN CELL; LIVER CELL; LIVER MICROSOME; PRIORITY JOURNAL; REGULATORY MECHANISM; GENETICS; HEPG2 CELL LINE; METABOLISM; TUMOR CELL LINE;

CELL LINE, TUMOR; CYTOCHROME P-450 CYP2B6; CYTOCHROME P-450 CYP3A; ENDOSULFAN; HEP G2 CELLS; HUMANS; METHOXYCHLOR; MICROSOMES, LIVER; PESTICIDES; RECEPTORS, CYTOPLASMIC AND NUCLEAR; RECEPTORS, STEROID; RNA, MESSENGER;

EID: 84904191354     PISSN: 00909556     EISSN: 1521009X     Source Type: Journal    
DOI: 10.1124/dmd.114.057786     Document Type: Article

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