Expression of cytochromes P450, conjugating enzymes and nuclear receptors in human hepatoma HepaRG cells

Drug Metabolism and Disposition

Volumn 34, Issue 1, 2006, Pages 75-83

  Aninat, Caroline ^a   Piton, Amélie ^a   Glaise, Denise ^b   Le Charpentier, Typhen ^b   Langouët, Sophie ^a   Morel, Fabrice ^a   Guguen Guillouzo, Christiane ^b   Guillouzo, André ^a  

^a UNIVERSITÉ DE RENNES 1   (France)

^b PONTCHAILLOU UNIVERSITY HOSPITAL   (France)

Author keywords

[No Author keywords available]

Indexed keywords

AROMATIC HYDROCARBON RECEPTOR; CELL NUCLEUS RECEPTOR; CONSTITUTIVE ANDROSTANE RECEPTOR; CYTOCHROME P450; CYTOCHROME P450 1A2; CYTOCHROME P450 2C9; CYTOCHROME P450 2D6; CYTOCHROME P450 3A4; DIMETHYL SULFOXIDE; ENZYME; GLUCURONOSYLTRANSFERASE 1A1; GLUTATHIONE TRANSFERASE A1; GLUTATHIONE TRANSFERASE A4; GLUTATHIONE TRANSFERASE M1; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR; PREGNANE X RECEPTOR; TRANSFERASE; UNCLASSIFIED DRUG;

ARTICLE; CELL CULTURE; CELL DIFFERENTIATION; CELL DIVISION; CELL STRUCTURE; CYTOTOXICITY; DENSITY; DRUG METABOLISM; EPITHELIUM CELL; HEPATOBILIARY SYSTEM; HEPATOMA CELL; HUMAN; HUMAN CELL; LIVER; LIVER CELL; LIVER CELL CARCINOMA; NUCLEOTIDE SEQUENCE; PRIORITY JOURNAL; PROTEIN EXPRESSION; REVERSE TRANSCRIPTION POLYMERASE CHAIN REACTION;

ACETAMINOPHEN; AFLATOXIN B1; AMIODARONE; CARCINOMA, HEPATOCELLULAR; CELL LINE, TUMOR; CELL SURVIVAL; CHLORPROMAZINE; CYTOCHROME P-450 ENZYME SYSTEM; DIMETHYL SULFOXIDE; GENE EXPRESSION; GENE EXPRESSION PROFILING; GLUCURONOSYLTRANSFERASE; HEPATOCYTES; HUMANS; INHIBITORY CONCENTRATION 50; ISOENZYMES; RECEPTORS, CYTOPLASMIC AND NUCLEAR; REVERSE TRANSCRIPTASE POLYMERASE CHAIN REACTION; RNA, MESSENGER; XENOBIOTICS;

EID: 29944444269     PISSN: 00909556     EISSN: 1521009X     Source Type: Journal    
DOI: 10.1124/dmd.105.006759     Document Type: Article

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