Mutation of Cys242 of Human Monoacylglycerol Lipase Disrupts Balanced Hydrolysis of 1-and 2-Monoacylglycerols and Selectively Impairs Inhibitor Potency s

Molecular Pharmacology

Volumn 85, Issue 3, 2014, Pages 510-519

  Laitinen, Tuomo ^a   Navia Paldanius, Dina ^a   Rytilahti, Roosa ^a   Marjamaa, Joona J T ^a   Karízková, Julie ^a   Parkkari, Teija ^a   Pantsar, Tatu ^a   Poso, Antti ^a   Laitinen, Jarmo T ^a   Savinainen, Juha R ^a  

^a UNIVERSITY OF EASTERN FINLAND   (Finland)

Author keywords

[No Author keywords available]

Indexed keywords

ARACHIDONIC ACIDS; CATALYSIS; CELL LINE; CYSTEINE; ENDOCANNABINOIDS; ENZYME INHIBITORS; GLYCERIDES; HEK293 CELLS; HUMANS; HYDROLYSIS; MONOACYLGLYCEROL LIPASES; MONOGLYCERIDES; MUTATION;

EID: 84894085407     PISSN: 0026895X     EISSN: 15210111     Source Type: Journal    
DOI: 10.1124/mol.113.090795     Document Type: Article

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