SCOPUS 정보 검색 플랫폼

Beilstein Journal of Organic Chemistry

Volumn 9, Issue , 2013, Pages 2696-2708

Stereoselectively fluorinated N-heterocycles: A brief survey

(2) Hu, Xiang Guo a Hunter, Luke a

a UNIVERSITY OF NEW SOUTH WALES (Australia)

Author keywords

Conformation; Fluorine; Iminosugars; Medicinal chemistry; N heterocycles; Organo fluorine

Indexed keywords

EID: 84890462953 PISSN: None EISSN: 18605397 Source Type: Journal
DOI: 10.3762/bjoc.9.306 Document Type: Review

Times cited : (72)

References (78)

1
- 0036882589
- doi:10.1016/S0022-1139(02)00201-4
- Ismail, F. M. D. J. Fluorine Chem. 2002, 118, 27-33. doi:10.1016/S0022- 1139(02)00201-4
- (2002) J. Fluorine Chem. , vol.118 , pp. 27-33
- Ismail, F.M.D.¹

2
- 77958039726
- doi:10.1016/j.jfluchem.2010.03.003
- O'Hagan, D. J. Fluorine Chem. 2010, 131, 1071-1081. doi:10.1016/j. jfluchem.2010.03.003
- (2010) J. Fluorine Chem. , vol.131 , pp. 1071-1081
- O'Hagan, D.¹

3
- 75449093256
- doi:10.1021/ar9001763
- Grushin, V. V. Acc. Chem. Res. 2010, 43, 160-171. doi:10.1021/ar9001763
- (2010) Acc. Chem. Res. , vol.43 , pp. 160-171
- Grushin, V.V.¹

4
- 79957603696
- doi:10.1038/nature10108
- Furuya, T.; Kamlet, A. S.; Ritter, T. Nature 2011, 473, 470-477. doi:10.1038/nature10108
- (2011) Nature , vol.473 , pp. 470-477
- Furuya, T.¹ Kamlet, A.S.² Ritter, T.³

5
- 11844274689
- doi:10.1002/anie.200460441
- Shimizu, M.; Hiyama, T. Angew. Chem., Int. Ed. 2004, 44, 214-231. doi:10.1002/anie.200460441
- (2004) Angew. Chem., Int. Ed. , vol.44 , pp. 214-231
- Shimizu, M.¹ Hiyama, T.²

6
- 79958141712
- doi:10.1021/cr1004293
- Tomashenko, O. A.; Grushin, V. V. Chem. Rev. 2011, 111, 4475-4521. doi:10.1021/cr1004293
- (2011) Chem. Rev. , vol.111 , pp. 4475-4521
- Tomashenko, O.A.¹ Grushin, V.V.²

7
- 84870541226
- doi:10.1038/nature11680
- Fujiwara, Y.; Dixon, J. A.; O'Hara, F.; Daa Funder, E.; Dixon, D. D.; Rodriguez, R. A.; Baxter, R. D.; Herlé, B.; Sach, N.; Collins, M. R.; Ishihara, Y.; Baran, P. S. Nature 2012, 492, 95-99. doi:10.1038/nature11680
- (2012) Nature , vol.492 , pp. 95-99
- Fujiwara, Y.¹ Dixon, J.A.² O'Hara, F.³ Daa Funder, E.⁴ Dixon, D.D.⁵ Rodriguez, R.A.⁶ Baxter, R.D.⁷ Herlé, B.⁸ Sach, N.⁹ Collins, M.R.¹⁰ Ishihara, Y.¹¹ Baran, P.S.¹²

8
- 84882268052
- doi:10.1002/anie.201206566
- Liang, T.; Neumann, C. N.; Ritter, T. Angew. Chem., Int. Ed. 2013, 52, 8214-8264. doi:10.1002/anie.201206566
- (2013) Angew. Chem., Int. Ed. , vol.52 , pp. 8214-8264
- Liang, T.¹ Neumann, C.N.² Ritter, T.³

9
- 84890444186
- doi:10.1007/7081-2011-63
- Sandford, G. Top. Heterocycl. Chem. 2012, 27, 1-32. doi:10.1007/7081- 2011-63
- (2012) Top. Heterocycl. Chem. , vol.27 , pp. 1-32
- Sandford, G.¹

10
- 84855221489
- Al-Maharik, N.; O'Hagan, D. Aldrichimica Acta 2011, 44, 65-75.
- (2011) Aldrichimica Acta , vol.44 , pp. 65-75
- Al-Maharik, N.¹ O'Hagan, D.²

11
- 11144341001
- Asymmetric fluorination, trifluoromethylation, and perfluoroalkylation reactions
- DOI 10.1021/cr030143e
- Ma, J.-A.; Cahard, D. Chem. Rev. 2004, 104, 6119-6146. doi:10.1021/cr030143e (Pubitemid 40025735)
- (2004) Chemical Reviews , vol.104 , Issue.12 , pp. 6119-6146
- Ma, J.-A.¹ Cahard, D.²

12
- 84890981047
- John Wiley & Sons: Hoboken, NJ, USA
- Petrov, C. A., Ed. Fluorinated Heterocyclic Compounds: Synthesis, Chemistry and Applications; John Wiley & Sons: Hoboken, NJ, USA, 2009.
- (2009) Fluorinated Heterocyclic Compounds: Synthesis, Chemistry and Applications
- Petrov, C.A.¹

13
- 83455243028
- doi:10.1002/anie.201102027
- Zimmer, L. E.; Sparr, C.; Gilmour, R. Angew. Chem., Int. Ed. 2011, 50, 11860-11871. doi:10.1002/anie.201102027
- (2011) Angew. Chem., Int. Ed. , vol.50 , pp. 11860-11871
- Zimmer, L.E.¹ Sparr, C.² Gilmour, R.³

14
- 38149016915
- doi:10.1039/b711844a
- O'Hagan, D. Chem. Soc. Rev. 2008, 37, 308-319. doi:10.1039/b711844a
- (2008) Chem. Soc. Rev. , vol.37 , pp. 308-319
- O'Hagan, D.¹

15
- 34547209700
- doi:10.1021/ol071127x
- van Hende, E.; Verniest, G.; Surmont, R.; De Kimpe, N. Org. Lett. 2007, 9, 2935-2937. doi:10.1021/ol071127x
- (2007) Org. Lett. , vol.9 , pp. 2935-2937
- Van Hende, E.¹ Verniest, G.² Surmont, R.³ De Kimpe, N.⁴

16
- 35548934674
- Synthesis and reactivity of 1-substituted 2-fluoro- and 2,2-difluoroaziridines
- DOI 10.1021/jo071253e
- Verniest, G.; Colpaert, F.; Van Hende, E.; De Kimpe, N. J. Org. Chem. 2007, 72, 8569-8572. doi:10.1021/jo071253e (Pubitemid 350012880)
- (2007) Journal of Organic Chemistry , vol.72 , Issue.22 , pp. 8569-8572
- Verniest, G.¹ Colpaert, F.² Van Hende, E.³ De Kimpe, N.⁴

17
- 33750021720
- The profound effect of fluorine substitution on the reactivity and regioselectivity of nucleophilic substitution reactions of strained heterocycles. A study of aziridine and its derivatives
- DOI 10.1021/jo061255j
- Banks, H. D. J. Org. Chem. 2006, 71, 8089-8097. doi:10.1021/jo061255j (Pubitemid 44571814)
- (2006) Journal of Organic Chemistry , vol.71 , Issue.21 , pp. 8089-8097
- Banks, H.D.¹

18
- 34547423776
- Enantioselective acylation of alcohols with fluorinated β-phenyl-β-lactams in the presence of Burkholderia cepacia lipase
- DOI 10.1016/j.tetasy.2007.06.033, PII S0957416607004946
- Li, X.-G.; Lähitie, M.; Päiviö, M.; Kanerva, L. T. Tetrahedron: Asymmetry 2007, 18, 1567-1573. doi:10.1016/j.tetasy.2007.06.033 (Pubitemid 47161127)
- (2007) Tetrahedron Asymmetry , vol.18 , Issue.13 , pp. 1567-1573
- Li, X.-G.¹ Lahitie, M.² Paivio, M.³ Kanerva, L.T.⁴

19
- 77952688640
- doi:10.3762/bjoc.6.38
- Hunter, L. Beilstein J. Org. Chem. 2010, 6, No. 38. doi:10.3762/bjoc.6.38
- (2010) Beilstein J. Org. Chem. , vol.6 , Issue.38
- Hunter, L.¹

20
- 33746410059
- The intramolecular β-fluorine ammonium interaction in 4- and 8-membered rings
- DOI 10.1039/b606334a
- Gooseman, N. E. J.; O'Hagan, D.; Slawin, A. M. Z.; Teale, A. M.; Tozer, D. J.; Young, R. J. Chem. Commun. 2006, 3190-3192. doi:10.1039/b606334a (Pubitemid 44126562)
- (2006) Chemical Communications , Issue.30 , pp. 3190-3192
- Gooseman, N.E.J.¹ O'Hagan, D.² Slawin, A.M.Z.³ Teale, A.M.⁴ Tozer, D.J.⁵ Young, R.J.⁶

21
- 0015932846
- doi:10.1021/ja00798a046
- Gerig, J. T.; McLeod, R. S. J. Am. Chem. Soc. 1973, 95, 5725-5729. doi:10.1021/ja00798a046
- (1973) J. Am. Chem. Soc. , vol.95 , pp. 5725-5729
- Gerig, J.T.¹ McLeod, R.S.²

22
- 79951657834
- doi:10.1039/c0ob00886a
- Campbell, N. H.; Smith, D. L.; Reszka, A. P.; Neidle, S.; O'Hagan, D. Org. Biomol. Chem. 2011, 9, 1328-1331. doi:10.1039/c0ob00886a
- (2011) Org. Biomol. Chem. , vol.9 , pp. 1328-1331
- Campbell, N.H.¹ Smith, D.L.² Reszka, A.P.³ Neidle, S.⁴ O'Hagan, D.⁵

23
- 0033079679
- A hyperstable collagen mimic
- DOI 10.1016/S1074-5521(99)80003-9
- Holmgren, S. K.; Bretscher, L. E.; Taylor, K. M.; Raines, R. T. Chem. Biol. 1999, 6, 63-70. doi:10.1016/S1074-5521(99)80003-9 (Pubitemid 29363157)
- (1999) Chemistry and Biology , vol.6 , Issue.2 , pp. 63-70
- Holmgren, S.K.¹ Bretscher, L.E.² Taylor, K.M.³ Raines, R.T.⁴

24
- 84891565619
- Wiley-VCH: Weinheim, Germany, doi:10.1002/352760393X
- Kirsch, P. Modern Fluoroorganic Chemistry: Synthesis, Reactivity, Applications; Wiley-VCH: Weinheim, Germany, 2004. doi:10.1002/352760393X
- (2004) Modern Fluoroorganic Chemistry: Synthesis, Reactivity, Applications
- Kirsch, P.¹

25
- 0032537113
- Code for collagen's stability deciphered [9]
- DOI 10.1038/33573
- Holmgren, S. K.; Taylor, K. M.; Bretscher, L. E.; Raines, R. T. Nature 1998, 392, 666-667. doi:10.1038/33573 (Pubitemid 28207776)
- (1998) Nature , vol.392 , Issue.6677 , pp. 666-667
- Holmgren, S.K.¹ Taylor, K.M.² Bretscher, L.E.³ Raines, R.T.⁴

26
- 81755187358
- doi:10.1002/chem.201102757
- Quintard, A.; Langlois, J.-B.; Emery, D.; Mareda, J.; Guénée, L.; Alexakis, A. Chem.-Eur. J. 2011, 17, 13433-13437. doi:10.1002/chem.201102757
- (2011) Chem.-Eur. J. , vol.17 , pp. 13433-13437
- Quintard, A.¹ Langlois, J.-B.² Emery, D.³ Mareda, J.⁴ Guénée, L.⁵ Alexakis, A.⁶

27
- 0001267759
- doi:10.1021/ja00061a055
- Lankin, D. C.; Chandrakumar, N. S.; Rao, S. N.; Spangler, D. P.; Snyder, J. P. J. Am. Chem. Soc. 1993, 115, 3356-3357. doi:10.1021/ja00061a055
- (1993) J. Am. Chem. Soc. , vol.115 , pp. 3356-3357
- Lankin, D.C.¹ Chandrakumar, N.S.² Rao, S.N.³ Spangler, D.P.⁴ Snyder, J.P.⁵

28
- 0034716326
- The unexpected diaxial orientation of cis-3,5-difluoropiperidine in water: A potent CF-NH charge-dipole effect
- DOI 10.1021/ja9934504
- Snyder, J. P.; Chandrakumar, N. S.; Sato, H.; Lankin, D. C. J. Am. Chem. Soc. 2000, 122, 544-545. doi:10.1021/ja9934504 (Pubitemid 30075497)
- (2000) Journal of the American Chemical Society , vol.122 , Issue.3 , pp. 544-545
- Snyder, J.P.¹ Chandrakumar, N.S.² Sato, H.³ Lankin, D.C.⁴

29
- 84962377223
- 3-Fluoropiperidines and N-methyl-3-fluoropiperidinium salts: The persistence of axial fluorine
- DOI 10.1002/chem.200400835
- Sum, A. M.; Lankin, D. C.; Hardcastle, K.; Snyder, J. P. Chem.-Eur. J. 2005, 11, 1579-1591. doi:10.1002/chem.200400835 (Pubitemid 40341887)
- (2005) Chemistry - A European Journal , vol.11 , Issue.5 , pp. 1579-1591
- Sun, A.¹ Lankin, D.C.² Hardcastle, K.³ Snyder, J.P.⁴

30
- 84890448457
- doi:10.1039/c3ob40391b
- Patel, A. R.; Ball, G.; Hunter, L.; Liu, F. Org. Biomol. Chem. 2013, 11, 3781-3785. doi:10.1039/c3ob40391b
- (2013) Org. Biomol. Chem. , vol.11 , pp. 3781-3785
- Patel, A.R.¹ Ball, G.² Hunter, L.³ Liu, F.⁴

31
- 84889478479
- Wiley-VCH: Chichester, UK
- Compain, P.; Martin, O. R., Eds. Iminosugars: From Synthesis to Therapeutic Applications; Wiley-VCH: Chichester, UK, 2007.
- (2007) Iminosugars: From Synthesis to Therapeutic Applications
- Compain, P.¹ Martin, O.R.²

32
- 0003532642
- Wiley-VCH: Weinheim, Germany
- Stütz, A. E., Ed. Iminosugars as Glycosidase Inhibitors: Nojirimycin and Beyond; Wiley-VCH: Weinheim, Germany, 1999.
- (1999) Iminosugars As Glycosidase Inhibitors: Nojirimycin and beyond
- Stütz, A.E.¹

33
- 0034607947
- Sugar-mimic glycosidase inhibitors: Natural occurrence, biological activity and prospects for therapeutic application
- DOI 10.1016/S0957-4166(00)00113-0, PII S0957416600001130
- Asano, N.; Nash, R. J.; Molyneux, R. J.; Fleet, G. W. J. Tetrahedron: Asymmetry 2000, 11, 1645-1680. doi:10.1016/S0957-4166(00)00113-0 (Pubitemid 30320886)
- (2000) Tetrahedron Asymmetry , vol.11 , Issue.8 , pp. 1645-1680
- Asano, N.¹ Nash, R.J.² Molyneux, R.J.³ Fleet, G.W.J.⁴

34
- 0035925104
- Polyhydroxylated alkaloids - Natural occurrence and therapeutic applications
- DOI 10.1016/S0031-9422(00)00451-9, PII S0031942200004519
- Watson, A. A.; Fleet, G. W. J.; Asano, N.; Molyneux, R. J.; Nash, R. J. Phytochemistry 2001, 56, 265-295. doi:10.1016/S0031-9422(00)00451-9 (Pubitemid 32162799)
- (2001) Phytochemistry , vol.56 , Issue.3 , pp. 265-295
- Watson, A.A.¹ Fleet, G.W.J.² Asano, N.³ Molyneux, R.J.⁴ Nash, R.J.⁵

35
- 0036462605
- Recent developments of transition-state analogue glycosidase inhibitors of non-natural product origin
- DOI 10.1021/cr000433k
- Lillelund, V. H.; Jensen, H. H.; Liang, X.; Bols, M. Chem. Rev. 2002, 102, 515-554. doi:10.1021/cr000433k (Pubitemid 35381638)
- (2002) Chemical Reviews , vol.102 , Issue.2 , pp. 515-553
- Lillelund, V.H.¹ Jensen, H.H.² Liang, X.³ Bols, M.⁴

36
- 33745728992
- Whalen, L. J.; Wong, C.-H. Aldrichimica Acta 2006, 39, 63-71.
- (2006) Aldrichimica Acta , vol.39 , pp. 63-71
- Whalen, L.J.¹ Wong, C.-H.²

37
- 80052454406
- doi:10.4155/fmc.11.117
- Nash, R. J.; Kato, A.; Yu, C.-Y.; Fleet, G. W. J. Future Med. Chem. 2011, 3, 1513-1521. doi:10.4155/fmc.11.117
- (2011) Future Med. Chem. , vol.3 , pp. 1513-1521
- Nash, R.J.¹ Kato, A.² Yu, C.-Y.³ Fleet, G.W.J.⁴

38
- 84867381413
- doi:10.1021/jo301327s
- Thaharn, W.; Bootwicha, T.; Soorukram, D.; Kuhakarn, C.; Prabpai, S.; Kongsaeree, P.; Tuchinda, P.; Reutrakul, V.; Pohmakotr, M. J. Org. Chem. 2012, 77, 8465-8479. doi:10.1021/jo301327s
- (2012) J. Org. Chem. , vol.77 , pp. 8465-8479
- Thaharn, W.¹ Bootwicha, T.² Soorukram, D.³ Kuhakarn, C.⁴ Prabpai, S.⁵ Kongsaeree, P.⁶ Tuchinda, P.⁷ Reutrakul, V.⁸ Pohmakotr, M.⁹

39
- 0025778594
- doi:10.1021/jo00006a031
- Reymond, J.-L.; Pinkerton, A. A.; Vogel, P. J. Org. Chem. 1991, 56, 2128-2135. doi:10.1021/jo00006a031
- (1991) J. Org. Chem. , vol.56 , pp. 2128-2135
- Reymond, J.-L.¹ Pinkerton, A.A.² Vogel, P.³

40
- 0028233603
- The chemistry of castanospermine, Part II: Synthesis of deoxyfluoro analogues of castanospermine
- DOI 10.1016/S0040-4039(00)76852-3
- Fumeaux, R. H.; Mason, J. M.; Tyler, P. C. Tetrahedron Lett. 1994, 35, 3143-3146. doi:10.1016/S0040-4039(00)76852-3 (Pubitemid 24162697)
- (1994) Tetrahedron Letters , vol.35 , Issue.19 , pp. 3143-3146
- Furneaux, R.H.¹ Mason, J.M.² Tyler, P.C.³

41
- 0028297871
- The chemistry of castanospermine, part I: Synthetic modifications at C-6
- DOI 10.1016/S0040-4020(01)85075-4
- Furneaux, R. H.; Gainsford, G. J.; Mason, J. M.; Tyler, P. C. Tetrahedron 1994, 50, 2131-2160. doi:10.1016/S0040-4020(01)85075-4 (Pubitemid 24098895)
- (1994) Tetrahedron , vol.50 , Issue.7 , pp. 2131-2160
- Furneaux, R.H.¹ Gainsford, G.J.² Mason, J.M.³ Tyler, P.C.⁴

42
- 0028861072
- doi:10.1016/0040-4020(95)00803-G
- Furneaux, R. H.; Gainsford, G. J.; Mason, J. M.; Tyler, P. C.; Hartley, O.; Winchester, B. G. Tetrahedron 1995, 51, 12611-12630. doi:10.1016/0040- 4020(95)00803-G
- (1995) Tetrahedron , vol.51 , pp. 12611-12630
- Furneaux, R.H.¹ Gainsford, G.J.² Mason, J.M.³ Tyler, P.C.⁴ Hartley, O.⁵ Winchester, B.G.⁶

43
- 79954437989
- doi:10.1039/c0ob01063d
- Li, Y.-X.; Huang, M.-H.; Yamashita, Y.; Kato, A.; Jia, Y.-M.; Wang, W.-B.; Fleet, G. W. J.; Nash, R. J.; Yu, C.-Y. Org. Biomol. Chem. 2011, 9, 3405-3414. doi:10.1039/c0ob01063d
- (2011) Org. Biomol. Chem. , vol.9 , pp. 3405-3414
- Li, Y.-X.¹ Huang, M.-H.² Yamashita, Y.³ Kato, A.⁴ Jia, Y.-M.⁵ Wang, W.-B.⁶ Fleet, G.W.J.⁷ Nash, R.J.⁸ Yu, C.-Y.⁹

44
- 0001765832
- doi:10.1021/ja00016a039
- Kajimoto, T.; Liu, K. K. C.; Derson, R. L.; Zhong, Z. Y.; Ichikawa, Y.; Porco, J. A.; Wong, C. H. J. Am. Chem. Soc. 1991, 113, 6187-6196. doi:10.1021/ja00016a039
- (1991) J. Am. Chem. Soc. , vol.113 , pp. 6187-6196
- Kajimoto, T.¹ Liu, K.K.C.² Derson, R.L.³ Zhong, Z.Y.⁴ Ichikawa, Y.⁵ Porco, J.A.⁶ Wong, C.H.⁷

45
- 0030917175
- Two isosteric fluorinated derivatives of the powerful glucosidase inhibitors, 1-deoxynojirimycin and 2,5-dideoxy-2,5-imino-D-mannitol: Syntheses and glycosidase-inhibitory activities of 1,2,5-trideoxy-2-fluoro-1,5-imino-D- glucitol and of 1,2,5-trideoxy-1-fluoro-2,5-imino-D-mannitol
- DOI 10.1016/S0008-6215(97)00099-2, PII S0008621597000992
- Anderson, S. M.; Ebner, M.; Ekhart, C. W.; Gradnig, G.; Legler, G.; Lundt, I.; Stütz, A. E.; Withers, S. G.; Wrodnigg, T. Carbohydr. Res. 1997, 301, 155-166. doi:10.1016/S0008-6215(97)00099-2 (Pubitemid 27272238)
- (1997) Carbohydrate Research , vol.301 , Issue.3-4 , pp. 155-166
- Andersen, S.M.¹ Ebner, M.² Ekhart, C.W.³ Gradnig, G.⁴ Legler, G.⁵ Lundt, I.⁶ Stutz, A.E.⁷ Withers, S.G.⁸ Wrodnigg, T.⁹

46
- 69949091359
- doi:10.1016/j.bmcl.2009.08.012
- Prell, E.; Csuk, R. Bioorg. Med. Chem. Lett. 2009, 19, 5673-5674. doi:10.1016/j.bmcl.2009.08.012
- (2009) Bioorg. Med. Chem. Lett. , vol.19 , pp. 5673-5674
- Prell, E.¹ Csuk, R.²

47
- 78349238135
- doi:10.1002/ardp.200900256
- Prell, E.; Korb, C.; Kluge, R.; Ströhl, D.; Csuk, R. Arch. Pharm. 2010, 343, 583-589. doi:10.1002/ardp.200900256
- (2010) Arch. Pharm. , vol.343 , pp. 583-589
- Prell, E.¹ Korb, C.² Kluge, R.³ Ströhl, D.⁴ Csuk, R.⁵

48
- 0035837068
- 2A receptor antagonists
- DOI 10.1021/jm0004998
- Rowley, M.; Hallett, D. J.; Goodacre, S.; Moyes, C.; Crawforth, J.; Sparey, T. J.; Patel, S.; Marwood, R.; Patel, S.; Thomas, S.; Hitzel, L.; O'Connor, D.; Szeto, N.; Castro, J. L.; Hutson, P. H.; Macleod, A. M. J. Med. Chem. 2001, 44, 1603-1614. doi:10.1021/jm0004998 (Pubitemid 32852203)
- (2001) Journal of Medicinal Chemistry , vol.44 , Issue.10 , pp. 1603-1614
- Rowley, M.¹ Hallett, D.J.² Goodacre, S.³ Moyes, C.⁴ Crawforth, J.⁵ Sparey, T.J.⁶ Patel, S.⁷ Marwood, R.⁸ Patel, S.⁹ Thomas, S.¹⁰ Hitzel, L.¹¹ O'Connor, D.¹² Szeto, N.¹³ Castro, J.L.¹⁴ Hutson, P.H.¹⁵ Macleod, A.M.¹⁶

49
- 0027977494
- doi:10.1002/anie.199417781
- Jespersen, T. M.; Dong, W.; Sierks, M. R.; Skrydstrup, T.; Lundt, I.; Bols, M. Angew. Chem., Int. Ed. Engl. 1994, 33, 1778-1779. doi:10.1002/anie. 199417781
- (1994) Angew. Chem., Int. Ed. Engl. , vol.33 , pp. 1778-1779
- Jespersen, T.M.¹ Dong, W.² Sierks, M.R.³ Skrydstrup, T.⁴ Lundt, I.⁵ Bols, M.⁶

50
- 63249088271
- doi:10.1016/j.tet.2009.02.079
- Li, R.-J.; Bols, M.; Rousseau, C.; Zhang, X.-G.; Wang, R.-W.; Qing, F.-L. Tetrahedron 2009, 65, 3717-3727. doi:10.1016/j.tet.2009.02.079
- (2009) Tetrahedron , vol.65 , pp. 3717-3727
- Li, R.-J.¹ Bols, M.² Rousseau, C.³ Zhang, X.-G.⁴ Wang, R.-W.⁵ Qing, F.-L.⁶

51
- 80051796424
- doi:10.1016/j.jfluchem.2011.05.031
- Yang, Y.; Zheng, F.; Bols, M.; Marinescu, L. G.; Qing, F.-L. J. Fluorine Chem. 2011, 838-845. doi:10.1016/j.jfluchem.2011.05.031
- (2011) J. Fluorine Chem. , pp. 838-845
- Yang, Y.¹ Zheng, F.² Bols, M.³ Marinescu, L.G.⁴ Qing, F.-L.⁵

52
- 84880573820
- doi:10.1016/j.bmc.2013.03.003
- López, O.; Qing, F.-L.; Pedersen, C. M.; Bols, M. Bioorg. Med. Chem. 2013, 21, 4755-4761. doi:10.1016/j.bmc.2013.03.003
- (2013) Bioorg. Med. Chem. , vol.21 , pp. 4755-4761
- López, O.¹ Qing, F.-L.² Pedersen, C.M.³ Bols, M.⁴

53
- 4544316921
- The polar hydrophobicity of fluorinated compounds
- DOI 10.1002/cbic.200300910
- Biffinger, J. C.; Kim, H. W.; DiMagno, S. G. ChemBioChem 2004, 5, 622-627. doi:10.1002/cbic.200300910 (Pubitemid 39257083)
- (2004) ChemBioChem , vol.5 , Issue.5 , pp. 622-627
- Biffinger, J.C.¹ Kim, H.W.² DiMagno, S.G.³

54
- 80053473935
- doi:10.1039/c1cc13956h
- Ioannou, A.; Cini, E.; Timofte, R. S.; Flitsch, S. L.; Turner, N. J.; Linclau, B. Chem. Commun. 2011, 47, 11228-11230. doi:10.1039/c1cc13956h
- (2011) Chem. Commun. , vol.47 , pp. 11228-11230
- Ioannou, A.¹ Cini, E.² Timofte, R.S.³ Flitsch, S.L.⁴ Turner, N.J.⁵ Linclau, B.⁶

55
- 0036500382
- Stereoelectronic substituent effects in polyhydroxylated piperidines and hexahydropyridazines
- DOI 10.1002/1521-3765(20020301)8:5<1218::AID-CHEM1218>3.0.CO;2-X
- Jensen, H. H.; Lyngbye, L.; Jensen, A.; Bols, M. Chem.-Eur. J. 2002, 8, 1218-1226. doi:10.1002/1521-3765(20020301)8:5<1218::AID-CHEM1218>3.0.CO;2- X (Pubitemid 34256361)
- (2002) Chemistry - A European Journal , vol.8 , Issue.5 , pp. 1218-1226
- Jensen, H.H.¹ Lyngbye, L.² Jensen, A.³ Bols, M.⁴

56
- 79960881545
- doi:10.1021/ja2048072
- Tang, P.; Wang, W.; Ritter, T. J. Am. Chem. Soc. 2011, 133, 11482-11484. doi:10.1021/ja2048072
- (2011) J. Am. Chem. Soc. , vol.133 , pp. 11482-11484
- Tang, P.¹ Wang, W.² Ritter, T.³

57
- 84874047432
- doi:10.1021/ja3125405
- Sladojevich, F.; Arlow, S. I.; Tang, P.; Ritter, T. J. Am. Chem. Soc. 2013, 135, 2470-2473. doi:10.1021/ja3125405
- (2013) J. Am. Chem. Soc. , vol.135 , pp. 2470-2473
- Sladojevich, F.¹ Arlow, S.I.² Tang, P.³ Ritter, T.⁴

58
- 77953398186
- doi:10.3998/ark.5550190.0011.812
- Ferret, H.; Déchamps, I.; Gomez Pardo, D.; Van Hijfte, L.; Cossy, J. ARKIVOC 2010, No. 8, 126-159. doi:10.3998/ark.5550190.0011.812
- (2010) ARKIVOC , Issue.8 , pp. 126-159
- Ferret, H.¹ Déchamps, I.² Gomez Pardo, D.³ Van Hijfte, L.⁴ Cossy, J.⁵

59
- 45749106438
- Rearrangement of 2-hydroxyalkylazetidines into 3-fluoropyrrolidines
- DOI 10.1055/s-2008-1072770
- Drouillat, B.; Couty, F.; David, O.; Evano, G.; Marrot, J. Synlett 2008, 1345-1348. doi:10.1055/s-2008-1072770 (Pubitemid 351870876)
- (2008) Synlett , Issue.9 , pp. 1345-1348
- Drouillat, B.¹ Couty, F.² David, O.³ Evano, G.⁴ Marrot, J.⁵

60
- 33847043960
- doi:10.1055/s-2007-967989
- Déchamps, I.; Gomez Pardo, D.; Cossy, J. Synlett 2007, 263-267. doi:10.1055/s-2007-967989
- (2007) Synlett , pp. 263-267
- Déchamps, I.¹ Gomez Pardo, D.² Cossy, J.³

61
- 34548361266
- doi:10.1002/ejoc.200700237
- Déchamps, I.; Gomez Pardo, D.; Cossy, J. Eur. J. Org. Chem. 2007, 4224-4234. doi:10.1002/ejoc.200700237
- (2007) Eur. J. Org. Chem. , pp. 4224-4234
- Déchamps, I.¹ Gomez Pardo, D.² Cossy, J.³

62
- 84878887864
- doi:10.1016/j.tet.2012.10.078
- Patel, A. R.; Liu, F. Tetrahedron 2012, 69, 744-752. doi:10.1016/j.tet. 2012.10.078
- (2012) Tetrahedron , vol.69 , pp. 744-752
- Patel, A.R.¹ Liu, F.²

63
- 0036779376
- Synthesis of fluoroalkyl substituted heterocycles using fluorine-containing building blocks
- DOI 10.2174/1385272023373635
- Zhu, S. Z.; Wang, Y. L.; Peng, W. M. Curr. Org. Chem. 2002, 6, 1057-1096. doi:10.2174/1385272023373635 (Pubitemid 34951191)
- (2002) Current Organic Chemistry , vol.6 , Issue.12 , pp. 1057-1096
- Zhu, S.Z.¹ Wang, Y.L.² Peng, W.M.³ Song, L.P.⁴ Jin, G.F.⁵

64
- 0002551083
- Building block approaches to aliphatic organofluorine compounds
- Chambers, R. D., Ed.; Springer-Verlag: Berlin, Germany
- Percy, J. M. Building Block Approaches to Aliphatic Organofluorine Compounds. In Organofluorine Chemistry: Techniques and Synthons; Chambers, R. D., Ed.; Springer-Verlag: Berlin, Germany, 1997; pp 131-195.
- (1997) Organofluorine Chemistry: Techniques and Synthons , pp. 131-195
- Percy, J.M.¹

65
- 84856108104
- doi:10.1021/jo2022845
- Kyne, S. H.; Miles, J. A. L.; Percy, J. M.; Singh, K. J. Org. Chem. 2012, 77, 991-998. doi:10.1021/jo2022845
- (2012) J. Org. Chem. , vol.77 , pp. 991-998
- Kyne, S.H.¹ Miles, J.A.L.² Percy, J.M.³ Singh, K.⁴

66
- 77953417458
- doi:10.4155/fmc.09.47
- Wilkinson, S. C.; Salmon, R.; Gouverneur, V. Future Med. Chem. 2009, 1, 847-863. doi:10.4155/fmc.09.47
- (2009) Future Med. Chem. , vol.1 , pp. 847-863
- Wilkinson, S.C.¹ Salmon, R.² Gouverneur, V.³

67
- 0035803748
- Synthesis of fluorogypsetin and fluorobrevianamide E by a novel fluorination - Cyclization of cyclo-L-Trp-L-AAs
- DOI 10.1002/1521-3773(20011203)40:23<4461::AID-ANIE4461>3.0.CO;2-E
- Shibata, N.; Tarui, T.; Doi, Y.; Kirk, K. L. Angew. Chem., Int. Ed. 2001, 40, 4461-4463. doi:10.1002/1521-3773(20011203)40:23<4461::AID-ANIE4461>3. 0.CO;2-E (Pubitemid 33150784)
- (2001) Angewandte Chemie - International Edition , vol.40 , Issue.23 , pp. 4461-4463
- Shibata, N.¹ Tarui, T.² Doi, Y.³ Kirk, K.L.⁴

68
- 37049114857
- doi:10.1039/C2969000644B
- Birch, A. J.; Wright, J. J. J. Chem. Soc. D 1969, 644b-645. doi:10.1039/C2969000644B
- (1969) J. Chem. Soc. D
- Birch, A.J.¹ Wright, J.J.²

69
- 0028299465
- doi:10.7164/antibiotics.47.163
- Shinohara, C.; Hasumi, K.; Takei, Y.; Endo, A. J. Antibiot. 1994, 47, 163-167. doi:10.7164/antibiotics.47.163
- (1994) J. Antibiot. , vol.47 , pp. 163-167
- Shinohara, C.¹ Hasumi, K.² Takei, Y.³ Endo, A.⁴

70
- 0028294112
- doi:10.7164/antibiotics.47.168
- Nuber, B.; Hansske, F.; Shinohara, C.; Miura, S.; Hasumi, K.; Endo, A. J. Antibiot. 1994, 47, 168-172. doi:10.7164/antibiotics.47.168
- (1994) J. Antibiot. , vol.47 , pp. 168-172
- Nuber, B.¹ Hansske, F.² Shinohara, C.³ Miura, S.⁴ Hasumi, K.⁵ Endo, A.⁶

71
- 80051775032
- doi:10.1002/anie.201103151
- Lozano, O.; Blessley, G.; del Campo, T. M.; Thompson, A. L.; Giuffredi, G. T.; Bettati, M.; Walker, M.; Borman, R.; Gouverneur, V. Angew. Chem., Int. Ed. 2011, 50, 8105-8109. doi:10.1002/anie.201103151
- (2011) Angew. Chem., Int. Ed. , vol.50 , pp. 8105-8109
- Lozano, O.¹ Blessley, G.² Del Campo, T.M.³ Thompson, A.L.⁴ Giuffredi, G.T.⁵ Bettati, M.⁶ Walker, M.⁷ Borman, R.⁸ Gouverneur, V.⁹

72
- 0343610039
- doi:10.1021/ja00728a056
- Kollonitsch, J.; Barash, L.; Doldouras, G. A. J. Am. Chem. Soc. 1970, 92, 7494-7495. doi:10.1021/ja00728a056
- (1970) J. Am. Chem. Soc. , vol.92 , pp. 7494-7495
- Kollonitsch, J.¹ Barash, L.² Doldouras, G.A.³

73
- 34250877795
- 2SPh: Synthesis of chiral 2,4-disubstituted 3,3-difluoropyrrolidines
- DOI 10.1002/anie.200604783
- Li, Y.; Hu, J. Angew. Chem., Int. Ed. 2007, 46, 2489-2492. doi:10.1002/anie.200604783 (Pubitemid 46973596)
- (2007) Angewandte Chemie - International Edition , vol.46 , Issue.14 , pp. 2489-2492
- Li, Y.¹ Hu, J.²

74
- 33748366516
- doi:10.1016/S0040-4020(01)98839-8
- Beckwith, A. L. J. Tetrahedron 1981, 37, 3073-3100. doi:10.1016/S0040- 4020(01)98839-8
- (1981) Tetrahedron , vol.37 , pp. 3073-3100
- Beckwith, A.L.J.¹

75
- 33845282341
- doi:10.1021/jo00382a001
- Spellmeyer, D. C.; Houk, K. N. J. Org. Chem. 1987, 52, 959-974. doi:10.1021/jo00382a001
- (1987) J. Org. Chem. , vol.52 , pp. 959-974
- Spellmeyer, D.C.¹ Houk, K.N.²

76
- 79959631387
- doi:10.1021/jo200813a
- Hunter, L.; Chung, J. H. J. Org. Chem. 2011, 76, 5502-5505. doi:10.1021/jo200813a
- (2011) J. Org. Chem. , vol.76 , pp. 5502-5505
- Hunter, L.¹ Chung, J.H.²

77
- 79951621675
- doi:10.1002/chem.201003320
- Hunter, L.; Jolliffe, K. A. J.; Jordan, M. J. T.; Jensen, P.; Macquart, R. B. Chem.-Eur. J. 2011, 17, 2340-2343. doi:10.1002/chem.201003320
- (2011) Chem.-Eur. J. , vol.17 , pp. 2340-2343
- Hunter, L.¹ Jolliffe, K.A.J.² Jordan, M.J.T.³ Jensen, P.⁴ Macquart, R.B.⁵

78
- 84866715184
- Hunter, L. Chim. Oggi 2012, 30 (3), 20-22.
- (2012) Chim. Oggi , vol.30 , Issue.3 , pp. 20-22
- Hunter, L.¹

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.