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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 21, 2013, Pages 5860-5864

Exploring the molecular determinants of substrate-selective inhibition of cyclooxygenase-2 by lumiracoxib

(5) Windsor, Matthew A a Valk, Pieter L a Xu, Shu a Banerjee, Surajit b,c Marnett, Lawrence J a

a VANDERBILT UNIVERSITY SCHOOL OF MEDICINE (United States)

b Cornell University ^* (United States)

c ARGONNE NATIONAL LABORATORY (United States)

Author keywords

COX 2; Endocannabinoids; Lumiracoxib; Prostaglandins; Substrate selective inhibition

Indexed keywords

2 ARACHIDONOYLGLYCEROL; ANANDAMIDE; ANILINE; ARACHIDONIC ACID; CYCLOOXYGENASE 2; CYCLOOXYGENASE 2 INHIBITOR; DES FLUOROLUMIRACOXIB; DICLOFENAC; ENDOCANNABINOID; ETHANOLAMINE DERIVATIVE; FLURBIPROFEN; GLYCEROL DERIVATIVE; INDOMETACIN; LUMIRACOXIB; METHYL GROUP; PHENYLACETIC ACID; PROSTAGLANDIN H2; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; DRUG POTENCY; DRUG SELECTIVITY; DRUG STRUCTURE; ENZYME INHIBITION; HYDROGEN BOND; IC 50; OXYGENATION;

COX-2; ENDOCANNABINOIDS; LUMIRACOXIB; PROSTAGLANDINS; SUBSTRATE-SELECTIVE INHIBITION;

ANIMALS; BINDING SITES; CYCLOOXYGENASE 2; CYCLOOXYGENASE 2 INHIBITORS; DICLOFENAC; ENDOCANNABINOIDS; MICE; MOLECULAR DOCKING SIMULATION;

EID: 84885161313 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.08.097 Document Type: Article

Times cited : (14)

References (22)

1
- 4143107932
- D.L. Simmons, R.M. Botting, and T. Hla Pharmacol. Rev. 56 2004 387
- (2004) Pharmacol. Rev. , vol.56 , pp. 387
- Simmons, D.L.¹ Botting, R.M.² Hla, T.³

2
- 80054080661
- C.A. Rouzer, and L.J. Marnett Chem. Rev. 111 2011 5899
- (2011) Chem. Rev. , vol.111 , pp. 5899
- Rouzer, C.A.¹ Marnett, L.J.²

3
- 0037661996
- T.F. Freund, I. Katona, and D. Piomelli Physiol. Rev. 83 2003 1017
- (2003) Physiol. Rev. , vol.83 , pp. 1017
- Freund, T.F.¹ Katona, I.² Piomelli, D.³

4
- 51649093696
- D.F. Woodward, R.W.C. Carling, C.L. Cornell, H.G. Fliri, J.L. Martos, S.N. Pettit, Y. Liang, and J.W. Wang Pharmacol. Ther. 120 2008 71
- (2008) Pharmacol. Ther. , vol.120 , pp. 71
- Woodward, D.F.¹ Carling, R.W.C.² Cornell, C.L.³ Fliri, H.G.⁴ Martos, J.L.⁵ Pettit, S.N.⁶ Liang, Y.⁷ Wang, J.W.⁸

5
- 68249100483
- J.J. Prusakiewicz, K.C. Duggan, C.A. Rouzer, and L.J. Marnett Biochemistry 48 2009 7353
- (2009) Biochemistry , vol.48 , pp. 7353
- Prusakiewicz, J.J.¹ Duggan, K.C.² Rouzer, C.A.³ Marnett, L.J.⁴

6
- 80054953106
- K.C. Duggan, D.J. Hermanson, J. Musee, J.J. Prusakiewicz, J.L. Scheib, B.D. Carter, S. Banerjee, J.A. Oates, and L.J. Marnett Nat. Chem. Biol. 7 2011 803
- (2011) Nat. Chem. Biol. , vol.7 , pp. 803
- Duggan, K.C.¹ Hermanson, D.J.² Musee, J.³ Prusakiewicz, J.J.⁴ Scheib, J.L.⁵ Carter, B.D.⁶ Banerjee, S.⁷ Oates, J.A.⁸ Marnett, L.J.⁹

7
- 34147119080
- A.L. Blobaum, and L.J. Marnett J. Med. Chem. 50 2007 1425
- (2007) J. Med. Chem. , vol.50 , pp. 1425
- Blobaum, A.L.¹ Marnett, L.J.²

8
- 79956290893
- L. Dong, A.J. Vecchio, N.P. Sharma, B.J. Jurban, M.G. Malkowski, and W.L. Smith J. Biol. Chem. 286 2011 19035
- (2011) J. Biol. Chem. , vol.286 , pp. 19035
- Dong, L.¹ Vecchio, A.J.² Sharma, N.P.³ Jurban, B.J.⁴ Malkowski, M.G.⁵ Smith, W.L.⁶

9
- 76249130338
- G. Rimon, R.S. Sidhu, D.A. Lauver, J.Y. Lee, N.P. Sharma, C. Yuan, R.A. Frieler, R.C. Trievel, B.R. Lucchesi, and W.L. Smith Proc. Natl. Acad. Sci. 107 2010 28
- (2010) Proc. Natl. Acad. Sci. , vol.107 , pp. 28
- Rimon, G.¹ Sidhu, R.S.² Lauver, D.A.³ Lee, J.Y.⁴ Sharma, N.P.⁵ Yuan, C.⁶ Frieler, R.A.⁷ Trievel, R.C.⁸ Lucchesi, B.R.⁹ Smith, W.L.¹⁰

10
- 0030068054
- D.K. Bhattacharyya, M. Lecomte, C.J. Rieke, R.M. Garavito, and W.L. Smith J. Biol. Chem. 271 1996 2179
- (1996) J. Biol. Chem. , vol.271 , pp. 2179
- Bhattacharyya, D.K.¹ Lecomte, M.² Rieke, C.J.³ Garavito, R.M.⁴ Smith, W.L.⁵

11
- 84866355094
- M.A. Windsor, D.J. Hermanson, P.J. Kingsley, S. Xu, B.C. Crews, W. Ho, C.M. Keenan, S. Banerjee, K.A. Sharkey, and L.J. Marnett ACS Med. Chem. Lett. 3 2012 759
- (2012) ACS Med. Chem. Lett. , vol.3 , pp. 759
- Windsor, M.A.¹ Hermanson, D.J.² Kingsley, P.J.³ Xu, S.⁴ Crews, B.C.⁵ Ho, W.⁶ Keenan, C.M.⁷ Banerjee, S.⁸ Sharkey, K.A.⁹ Marnett, L.J.¹⁰

12
- 34447526067
- A.L. Blobaum, and L.J. Marnett J. Biol. Chem. 282 2007 16379
- (2007) J. Biol. Chem. , vol.282 , pp. 16379
- Blobaum, A.L.¹ Marnett, L.J.²

13
- 0242580725
- S.W. Rowlinson, J.R. Kiefer, J.J. Prusakiewicz, J.L. Pawlitz, K.R. Kozak, A.S. Kalgutkar, W.C. Stallings, R.G. Kurumbail, and L.J. Marnett J. Biol. Chem. 278 2003 45763
- (2003) J. Biol. Chem. , vol.278 , pp. 45763
- Rowlinson, S.W.¹ Kiefer, J.R.² Prusakiewicz, J.J.³ Pawlitz, J.L.⁴ Kozak, K.R.⁵ Kalgutkar, A.S.⁶ Stallings, W.C.⁷ Kurumbail, R.G.⁸ Marnett, L.J.⁹

14
- 34547105217
- American Chemical Society Washington, D.C. pp. 22-26
- K. Clark, R. Kulathila, J. Koehn, S. Rieffel, A. Strauss, S. Hu, M. Kalfoglou, D. Szeto, D. Lasala, M. Sabio, X. Wang, and P. Marshall American Chemical Society: Book of Abstracts 2004 American Chemical Society Washington, D.C. pp. 22-26
- (2004) American Chemical Society: Book of Abstracts
- Clark, K.¹ Kulathila, R.² Koehn, J.³ Rieffel, S.⁴ Strauss, A.⁵ Hu, S.⁶ Kalfoglou, M.⁷ Szeto, D.⁸ Lasala, D.⁹ Sabio, M.¹⁰ Wang, X.¹¹ Marshall, P.¹²

15
- 16744369033
- J.R. Kiefer, J.L. Pawlitz, K.T. Moreland, R.A. Stegeman, W.F. Hood, J.K. Gierse, A.M. Stevens, D.C. Goodwin, S.W. Rowlinson, L.J. Marnett, W.C. Stallings, and R.G. Kurumbail Nature 405 2000 97
- (2000) Nature , vol.405 , pp. 97
- Kiefer, J.R.¹ Pawlitz, J.L.² Moreland, K.T.³ Stegeman, R.A.⁴ Hood, W.F.⁵ Gierse, J.K.⁶ Stevens, A.M.⁷ Goodwin, D.C.⁸ Rowlinson, S.W.⁹ Marnett, L.J.¹⁰ Stallings, W.C.¹¹ Kurumbail, R.G.¹²

16
- 0030461132
- R.G. Kurumbail, A.M. Stevens, J.K. Gierse, J.J. McDonald, R.A. Stegeman, J.Y. Pak, D. Gildehaus, J.M. Iyashiro, T.D. Penning, K. Seibert, P.C. Isakson, and W.C. Stallings Nature 384 1996 644
- (1996) Nature , vol.384 , pp. 644
- Kurumbail, R.G.¹ Stevens, A.M.² Gierse, J.K.³ McDonald, J.J.⁴ Stegeman, R.A.⁵ Pak, J.Y.⁶ Gildehaus, D.⁷ Iyashiro, J.M.⁸ Penning, T.D.⁹ Seibert, K.¹⁰ Isakson, P.C.¹¹ Stallings, W.C.¹²

17
- 0015150481
- W.L. Smith, and W.E.M. Lands J. Biol. Chem. 246 1971 6700
- (1971) J. Biol. Chem. , vol.246 , pp. 6700
- Smith, W.L.¹ Lands, W.E.M.²

18
- 0033594911
- T.D. Warner, F. Giuliano, I. Vojnovic, A. Bukasa, J.A. Mitchell, and J.R. Vane Proc. Natl. Acad. Sci. 96 1999 7563
- (1999) Proc. Natl. Acad. Sci. , vol.96 , pp. 7563
- Warner, T.D.¹ Giuliano, F.² Vojnovic, I.³ Bukasa, A.⁴ Mitchell, J.A.⁵ Vane, J.R.⁶

19
- 0022382640
- R.J. Kulmacz, and W.E. Lands J. Biol. Chem. 260 1985 12572
- (1985) J. Biol. Chem. , vol.260 , pp. 12572
- Kulmacz, R.J.¹ Lands, W.E.²

20
- 10644285687
- J.J. Prusakiewicz, A.S. Felts, B.S. Mackenzie, and L.J. Marnett Biochemistry 43 2004 15439
- (2004) Biochemistry , vol.43 , pp. 15439
- Prusakiewicz, J.J.¹ Felts, A.S.² Mackenzie, B.S.³ Marnett, L.J.⁴

21
- 79958009684
- A.J. Vecchio, and M.G. Malkowski J. Biol. Chem. 286 2011 20736
- (2011) J. Biol. Chem. , vol.286 , pp. 20736
- Vecchio, A.J.¹ Malkowski, M.G.²

22
- 77954611060
- A.J. Vecchio, D.M. Simmons, and M.G. Malkowski J. Biol. Chem. 285 2010 22152
- (2010) J. Biol. Chem. , vol.285 , pp. 22152
- Vecchio, A.J.¹ Simmons, D.M.² Malkowski, M.G.³

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