-
1
-
-
0029070763
-
Review pharmaceutical solids: A strategic approach to regulatory considerations
-
Byrn S, Pfeiffer R, Ganey M, et al. Review. Pharmaceutical solids: A strategic approach to regulatory considerations. Pharm Res 1995;12:945-54
-
(1995)
Pharm Res
, vol.12
, pp. 945-954
-
-
Byrn, S.1
Pfeiffer, R.2
Ganey, M.3
-
3
-
-
84884573249
-
-
ANDAs U.S. Department of Health and Human Services, FDA/Center for Drug Evaluation and Research,. Available from [Last accessed 26 March 13]
-
ANDAs: Pharmaceutical Solid polymorphism chemistry, manufacturing, and controls information. Guidance for Industry. U.S. Department of Health and Human Services, FDA/Center for Drug Evaluation and Research, 2007. Available from: Http://www.fda.gov/downloads/Drugs/GuidanceComplianceRegulatory Information/Guidances/ucm072866.pdf [Last accessed 26 March 13]
-
(2007)
Pharmaceutical Solid Polymorphism Chemistry Manufacturing And Controls Information. Guidance For Industry
-
-
-
4
-
-
4344717272
-
Solid-state of pharmaceutical compounds impact of the ICH Q6 guideline on industrial development
-
Giron D, Mutz M, Garnier S. Solid-state of pharmaceutical compounds impact of the ICH Q6 guideline on industrial development. J Therm Anal Calorim 2004;77:709-47
-
(2004)
J Therm Anal Calorim
, vol.77
, pp. 709-747
-
-
Giron, D.1
Mutz, M.2
Garnier, S.3
-
8
-
-
0034980946
-
Investigation of polymorphism and pseudo-polymorphism in pharmaceutical by combined analytical techniques
-
Giron D. Investigation of polymorphism and pseudo-polymorphism in pharmaceutical by combined analytical techniques. J Therm Anal Calorim 2001;64:37-60
-
(2001)
J Therm Anal Calorim
, vol.64
, pp. 37-60
-
-
Giron, D.1
-
9
-
-
0017188210
-
Relationship between acute toxicity in mice and polymorphic forms of polyene antibiotics
-
Ghielmetti G, Bruzzese T, Bianchi C, Recusani F. Relationship between acute toxicity in mice and polymorphic forms of polyene antibiotics. J Pharm Sci 1976;65:905-7
-
(1976)
J Pharm Sci
, vol.65
, pp. 905-907
-
-
Ghielmetti, G.1
Bruzzese, T.2
Bianchi, C.3
Recusani, F.4
-
10
-
-
0034874245
-
Ritonavir: An extraordinary example of conformational polymorphism
-
Bauer J, Spanton S, Henry R, et al. Ritonavir: An extraordinary example of conformational polymorphism. Pharm Res 2001;18:859-66
-
(2001)
Pharm Res
, vol.18
, pp. 859-866
-
-
Bauer, J.1
Spanton, S.2
Henry, R.3
-
11
-
-
84884540262
-
-
HIV and AIDS Activities. Available from [Last accessed 28 March 13]
-
HIV and AIDS Activities. Office of Health and Constituent Affairs, U.S. Food and Drug Administration. 2013. Available from: Http://www.fda.gov/ ForConsumers/ByAudience/ForPatientAdvocates/HIVandAIDSActivities/ucm200179.htm [Last accessed 28 March 13]
-
(2013)
Office Of Health Constituent Affairs U.S. Food Drug Administration
-
-
-
12
-
-
0002425795
-
Theory and origin of polymorphism
-
Brittain HG, editior Marcel Dekker New York
-
Grant DJW. Theory and origin of polymorphism. In: Polymorphism in pharmaceutical solids. Brittain HG, editior Marcel Dekker; New York: 1999
-
(1999)
Polymorphism in pharmaceutical solids
-
-
Grant, D.J.W.1
-
15
-
-
27944487022
-
Occurrence of pharmaceutically acceptable anions and cations in the Cambridge structural database
-
Haynes DA, Jones W, Motherwell WDS. Occurrence of pharmaceutically acceptable anions and cations in the Cambridge structural database. J Pharm Sci 2005;94:2111-20
-
(2005)
J Pharm Sci
, vol.94
, pp. 2111-2120
-
-
Haynes, D.A.1
Jones, W.2
Motherwell, W.D.S.3
-
17
-
-
0023032232
-
Salt selection for basic drugs
-
Gould PL. Salt selection for basic drugs. Int J Pharm 1986;33:201-17
-
(1986)
Int J Pharm
, vol.33
, pp. 201-217
-
-
Gould, P.L.1
-
18
-
-
43049170351
-
The role of cocrystals in pharmaceutical science
-
Shan N, Zaworotko MJ. The role of cocrystals in pharmaceutical science. Drug Discov Today 2008;13:440-6
-
(2008)
Drug Discov Today
, vol.13
, pp. 440-446
-
-
Shan, N.1
Zaworotko, M.J.2
-
19
-
-
78649683097
-
Benefits of cocrystallization in pharmaceutical materials science: An update
-
Frişçić T, Jones W. Benefits of cocrystallization in pharmaceutical materials science: An update. J Pharm Pharmacol 2010;62:1547-59
-
(2010)
J Pharm Pharmacol
, vol.62
, pp. 1547-1559
-
-
Frişçić, T.1
Jones, W.2
-
20
-
-
84860442899
-
Polymorphs, salts, and cocrystals: What's in a name?
-
Aitipamula S, Banerjee R, Bansal AK, et al. Polymorphs, salts, and cocrystals: What's in a name? Cryst Growth Des 2012;12:2147-52
-
(2012)
Cryst Growth Des
, vol.12
, pp. 2147-2152
-
-
Aitipamula, S.1
Banerjee, R.2
Bansal, A.K.3
-
21
-
-
84876892154
-
Understanding the effects of ionicity in salts, solvates, co-crystals, ionic co-crystals, and ionic liquids, rather than nomenclature, is critical to understanding their behavior
-
Kelley SP, Narita A, Holbrey JD, et al. Understanding the effects of ionicity in salts, solvates, co-crystals, ionic co-crystals, and ionic liquids, rather than nomenclature, is critical to understanding their behavior. Cryst Growth Des 2013;13:965-75
-
(2013)
Cryst Growth Des
, vol.13
, pp. 965-975
-
-
Kelley, S.P.1
Narita, A.2
Holbrey, J.D.3
-
22
-
-
79954998105
-
-
Ionic Liquids: Industrial Applications For Green Chemistry. In: ACS Symposium Series 818. American Chemical Society Washington DC
-
Ionic liquids: Industrial applications for green chemistry. In: Rogers RD, Seddon KR, editors. Ionic liquids: Industrial applications for green chemistry. ACS Symposium Series 818. American Chemical Society; Washington; DC: 2002
-
(2002)
Ionic Liquids: Industrial Applications For Green Chemistry
-
-
Rogers, R.D.1
Seddon, K.R.2
-
23
-
-
79751484932
-
Liquid forms of pharmaceutical cocrystals: Exploring the boundaries of salt formation
-
Bica K, Shamshina J, Hough WL, et al. Liquid forms of pharmaceutical cocrystals: Exploring the boundaries of salt formation. Chem Commun 2011;47:2267-9
-
(2011)
Chem Commun
, vol.47
, pp. 2267-2269
-
-
Bica, K.1
Shamshina, J.2
Hough, W.L.3
-
24
-
-
84889625022
-
Synthesis of ionic liquids
-
In: Endres F, Abbott AP, MacFarlane DR, editors. Wiley-VCH Verlag GmbH & Co. KGaA
-
Beyersdorff T, Schubert TJS, Welz-Biermann U, et al. Synthesis of ionic liquids. In: Endres F, Abbott AP, MacFarlane DR, editors. In Electrodeposition from ionic liquids. Wiley-VCH Verlag GmbH & Co. KGaA; 2008. p. 15-46
-
(2008)
Electrodeposition from ionic liquids
, pp. 15-46
-
-
Beyersdorff, T.1
Schubert, T.J.S.2
Welz-Biermann, U.3
-
25
-
-
75649115343
-
Syn thesis, purification and characterization of ionic liquids
-
Clare B, Sirwardana A, Mac Farlane DR. Synthesis, purification and characterization of ionic liquids. Top Curr Chem 2010;290:1-40
-
(2010)
Top Curr Chem
, vol.290
, pp. 1-40
-
-
Clare, B.1
Sirwardana, A.2
Mac Farlane, D.R.3
-
26
-
-
84891333242
-
-
In: Wasserscheid P Welton T Editor. Ionic Liq. Synth. 2nd Edition. Wiley. VCH Verlag GmbH & Co. KGaA
-
Gordon CM, Muldoon MJ. Synthesis and purification: Synthesis of ionic liquids. In: Wasserscheid P, Welton T, editor. Ionic Liq. Synth. 2nd edition. Wiley-VCH Verlag GmbH & Co. KGaA; 2008. p. 7-25
-
(2008)
Synthesis And Purification: Synthesis Of Ionic Liquids
, pp. 7-25
-
-
Gordon, C.M.1
Muldoon, M.J.2
-
27
-
-
84857323337
-
Designing, synthesis and applications of task specific ionic liquids
-
Hullio AA, Mastoi GM. Designing, synthesis and applications of task specific ionic liquids. Orient J Chem 2011;27:1591-612
-
(2011)
Orient J Chem
, vol.27
, pp. 1591-1612
-
-
Hullio, A.A.1
Mastoi, G.M.2
-
28
-
-
57249114417
-
Ionic liquids based on imidazolium, ammonium and pyrrolidinium salts of the dicyanamide anion
-
MacFarlane DR, Forsyth SA, Golding J, et al. Ionic liquids based on imidazolium, ammonium and pyrrolidinium salts of the dicyanamide anion. Green Chem 2002;4:444-8
-
(2002)
Green Chem
, vol.4
, pp. 444-448
-
-
MacFarlane, D.R.1
Forsyth, S.A.2
Golding, J.3
-
29
-
-
27744578633
-
Influence of ion size asymmetry on the properties of ionic liquid-vapour interfaces
-
Bresme F, González-Melchor M, Alejandre J. Influence of ion size asymmetry on the properties of ionic liquid-vapour interfaces. J Phys Condens Matter 2005;17:S3301-7
-
(2005)
J Phys Condens Matter
, vol.17
-
-
Bresme, F.1
González-Melchor, M.2
Alejandre, J.3
-
30
-
-
33645763725
-
1-N-alkyl-3-methylimidazolium ionic liquids as neat lubricants and lubricant additives in steel-aluminium contacts
-
Jiménez AE, Berm-udez MD, Iglesias P, et al. 1-N-alkyl-3- methylimidazolium ionic liquids as neat lubricants and lubricant additives in steel-aluminium contacts. Wear 2006;260:766-82
-
(2006)
Wear
, vol.260
, pp. 766-782
-
-
Jiménez, A.E.1
Berm-Udez, M.D.2
Iglesias, P.3
-
31
-
-
2342503807
-
Room temperature ionic liquid 1-ethyl-3-hexylimidazolium-bis (trifluoromethylsulfonyl)-imide as lubricant for steel-steel contact
-
Lu Q, Wang H, Ye C, et al. Room temperature ionic liquid 1-ethyl-3-hexylimidazolium-bis (trifluoromethylsulfonyl)-imide as lubricant for steel-steel contact. Tribol Int 2004;37:547-52
-
(2004)
Tribol Int
, vol.37
, pp. 547-552
-
-
Lu, Q.1
Wang, H.2
Ye, C.3
-
32
-
-
3242763786
-
Functional room-temperature ionic liquids as lubricants for an aluminum-on-steel system
-
Mu Z, Liu W, Zhang S, et al. Functional room-temperature ionic liquids as lubricants for an aluminum-on-steel system. Chem Lett 2004;33:524-5
-
(2004)
Chem Lett
, vol.33
, pp. 524-525
-
-
Mu, Z.1
Liu, W.2
Zhang, S.3
-
33
-
-
0035824005
-
Room-temperature ionic liquids: A novel versatile lubricant
-
Ye C, Liu W, Chen Y, et al. Room-temperature ionic liquids: A novel versatile lubricant. Chem Commun 2001;21:2244-5
-
(2001)
Chem Commun
, vol.21
, pp. 2244-2245
-
-
Ye, C.1
Liu, W.2
Chen, Y.3
-
34
-
-
57249114468
-
The greening of explosives and propellants using high-energy nitrogen chemistry
-
Klapotke TM, Holl G. The greening of explosives and propellants using high-energy nitrogen chemistry. Green Chem 2001;3:G75
-
(2001)
Green Chem
, vol.3
-
-
Klapotke, T.M.1
Holl, G.2
-
35
-
-
34548260269
-
Choline-derivative-based ionic liquids
-
Pernak J, Syguda A, Mirska I, et al. Choline-derivative-based ionic liquids. Chem Eur J 2007;13:6817-27
-
(2007)
Chem Eur J
, vol.13
, pp. 6817-6827
-
-
Pernak, J.1
Syguda, A.2
Mirska, I.3
-
36
-
-
34547399045
-
The third evolution of ionic liquids: Active pharmaceutical ingredients
-
Hough WL, Smiglak M, Rodríguez H, et al. The third evolution of ionic liquids: Active pharmaceutical ingredients. New J Chem 2007;31:1429-36
-
(2007)
New J Chem
, vol.31
, pp. 1429-1436
-
-
Hough, W.L.1
Smiglak, M.2
Rodríguez, H.3
-
37
-
-
46149112704
-
Ionic liquids then and now: From solvents to materials to active pharmaceutical ingredients
-
Hough WL, Rogers RD. Ionic liquids then and now: From solvents to materials to active pharmaceutical ingredients. Bull Chem Soc Jpn 2007;80:2262-9
-
(2007)
Bull Chem Soc Jpn
, vol.80
, pp. 2262-2269
-
-
Hough, W.L.1
Rogers, R.D.2
-
38
-
-
84884584566
-
Structure-property relationships in ionic liquids
-
In: Rogers RD, Seddon KR, editors. ACS Symposium Series 818. American Chemical Society; Washington, DC
-
Martin JD. Structure-property relationships in ionic liquids. In: Rogers RD, Seddon KR, editors. In Ionic liquids: Industrial applications for green chemistry. ACS Symposium Series 818. American Chemical Society; Washington, DC: 2002
-
(2002)
Ionic liquids: Industrial applications for green chemistry
-
-
Martin, J.D.1
-
40
-
-
84884574502
-
Dual functioning ionic liquids and salts thereof
-
WO 2010/078300 (2010), US 2012/0046244 A1
-
Rogers RD, Daly DT, MacFarlane D, et al. Dual functioning ionic liquids and salts thereof. PCT Int Appl. WO 2010/078300 (2010), US 2012/0046244 A1; 2012
-
(2012)
PCT Int Appl.
-
-
Rogers, R.D.1
Daly, D.T.2
MacFarlane, D.3
-
41
-
-
84884546545
-
-
U.S. Patent N.o. 8 232265 PCT/US2006/039454 WO 2007/044693 A2 2007), MX 301158
-
Rogers RD, Daly DT, Swatloski RP, et al. Multifunctional ionic liquid compositions for overcoming polymorphism and imparting improved properties for active pharmaceutical, biological, nutritional and energetic ingredients. U.S. Patent No. 8,232,265; PCT/US2006/039454; WO 2007/044693 A2 (2007), MX 301158; 2012
-
(2012)
Multifunctional ionic liquid compositions for overcoming polymorphism and imparting improved properties for active pharmaceutical, biological, nutritional and energetic ingredients.
-
-
Rogers, R.D.1
Daly, D.T.2
Swatloski, R.P.3
-
42
-
-
84884546233
-
Compounds comprising two or more biologically functional ions and method of treating Parkinson's Disease
-
WO 2010078258 A1 20100708
-
Rogers RD, Rijksen C, Daly DT, et al. Compounds comprising two or more biologically functional ions and method of treating Parkinson's Disease. PCT Int. Appl. WO 2010078258 A1 20100708; 2010
-
(2010)
PCT Int. Appl.
-
-
Rogers, R.D.1
Rijksen, C.2
Daly, D.T.3
-
43
-
-
84859412431
-
Development of novel ionic liquids based on ampicillin
-
Ferraz R, Branco LC, Marrucho IM, et al. Development of novel ionic liquids based on ampicillin. MedChemCommun 2012;3:494-7
-
(2012)
Med Chem Commun
, vol.3
, pp. 494-497
-
-
Ferraz, R.1
Branco, L.C.2
Marrucho, I.M.3
-
44
-
-
36749086203
-
Accounting for the unique, doubly dual nature of ionic liquids from a molecular thermodynamic and modeling standpoint
-
Rebelo LPN, Lopes JNC, Esperança JMSS, et al. Accounting for the unique, doubly dual nature of ionic liquids from a molecular thermodynamic and modeling standpoint. Acc Chem Res 2007;40:1114-21
-
(2007)
Acc Chem Res
, vol.40
, pp. 1114-1121
-
-
Rebelo, L.P.N.1
Lopes, J.N.C.2
Esperança, J.M.S.S.3
-
45
-
-
33644749212
-
From dysfunction to bis-function: On the design and applications of functionalised ionic liquids
-
Fei Z, Geldbach TJ, Zhao D, et al. From dysfunction to bis-function: On the design and applications of functionalised ionic liquids. Chem Eur J 2006;12:2122-30
-
(2006)
Chem Eur J
, vol.12
, pp. 2122-2130
-
-
Fei, Z.1
Geldbach, T.J.2
Zhao, D.3
-
46
-
-
61749089401
-
Exploring an anti-crystal engineering approach to the preparation of pharmaceutically active ionic liquids
-
Dean PM, Turanjanin J, Yoshizawa-Fujita M, et al. Exploring an anti-crystal engineering approach to the preparation of pharmaceutically active ionic liquids. Cryst Growth Des 2009;9:1137-45
-
(2009)
Cryst Growth Des
, vol.9
, pp. 1137-1145
-
-
Dean, P.M.1
Turanjanin, J.2
Yoshizawa-Fujita, M.3
-
47
-
-
77149123276
-
In search of pure liquid salt forms of aspirin: Ionic liquid approaches with acetylsalicylic acid and salicylic acid
-
Bica K, Rijksen C, Nieuwenhuyzen M, et al. In search of pure liquid salt forms of aspirin: Ionic liquid approaches with acetylsalicylic acid and salicylic acid. Phys Chem Chem Phys 2010;12:2011-17
-
(2010)
Phys Chem Chem Phys
, vol.12
, pp. 2011-2017
-
-
Bica, K.1
Rijksen, C.2
Nieuwenhuyzen, M.3
-
48
-
-
84862796321
-
New ionic derivatives of betulinic acid as highly potent anti-cancer agents
-
Suresh C, Zhao H, Gumbs A, et al. New ionic derivatives of betulinic acid as highly potent anti-cancer agents. Bioorg Med Chem Lett 2012;22:1734-8
-
(2012)
Bioorg Med Chem Lett
, vol.22
, pp. 1734-1738
-
-
Suresh, C.1
Zhao, H.2
Gumbs, A.3
-
49
-
-
76349107155
-
Confused ionic liquid ions - A liquification and dosage strategy for pharmaceutically active salts
-
Bica K, Rogers RD. Confused ionic liquid ions - a " liquification" and dosage strategy for pharmaceutically active salts. Chem Commun 2010;46:1215-17
-
(2010)
Chem Commun
, vol.46
, pp. 1215-1217
-
-
Bica, K.1
Rogers, R.D.2
-
50
-
-
0348110657
-
Ionic liquids by proton transfer: Vapor pressure, conductivity, and the relevance of DpKa from aqueous solutions
-
Yoshizawa M, Xu W, Angell CA. Ionic liquids by proton transfer: Vapor pressure, conductivity, and the relevance of DpKa from aqueous solutions. J Am Chem Soc 2003;125:15411-19
-
(2003)
J Am Chem Soc
, vol.125
, pp. 15411-15419
-
-
Yoshizawa, M.1
Xu, W.2
Angell, C.A.3
-
51
-
-
2342481809
-
Lessons learned from marketed and investigational prodrugs
-
Ettmayer P, Amidon GL, Clement B, et al. Lessons learned from marketed and investigational prodrugs. J Med Chem 2004;47:2393-404
-
(2004)
J Med Chem
, vol.47
, pp. 2393-2404
-
-
Ettmayer, P.1
Amidon, G.L.2
Clement, B.3
-
52
-
-
34548024418
-
Prodrug strategies to overcome poor water solubility
-
Stella VJ, Nti-Addae KW. Prodrug strategies to overcome poor water solubility. Adv Drug Deliv Rev 2007;59:677-94
-
(2007)
Adv Drug Deliv Rev
, vol.59
, pp. 677-694
-
-
Stella, V.J.1
Nti-Addae, K.W.2
-
54
-
-
80052422613
-
Prodrug strategies in drug design
-
In: Rautio J, editor. Wiley-VCH Verlag GmbH & Co. KgaA; Weinheim
-
Rautio J. Prodrug strategies in drug design. In: Rautio J, editor. In Prodrugs and targeted delivery: Towards better ADME properties. Wiley-VCH Verlag GmbH & Co. KgaA; Weinheim: 2010
-
(2010)
Prodrugs and targeted delivery: Towards better ADME properties
-
-
Rautio, J.1
-
55
-
-
0014104395
-
Effect of polymorphism on the absorption of chloramphenicol from chloramphenicol palmitate
-
Aguiar AJ, Krc J Jr, Kinkel AW, et al. Effect of polymorphism on the absorption of chloramphenicol from chloramphenicol palmitate. J Pharm Sci 1967;56:847-53
-
(1967)
J Pharm Sci
, vol.56
, pp. 847-853
-
-
Aguiar, A.J.1
Krc Jr., J.2
Kinkel, A.W.3
-
56
-
-
84874459413
-
Prodrug ionic liquids: Functionalizing neutral active pharmaceutical ingredients to take advantage of the ionic liquid form
-
Cojocaru OA, Bica K, Gurau G, et al. Prodrug ionic liquids: Functionalizing neutral active pharmaceutical ingredients to take advantage of the ionic liquid form. MedChemCommun 2013;4:559-63
-
(2013)
Med Chem Commun
, vol.4
, pp. 559-563
-
-
Cojocaru, O.A.1
Bica, K.2
Gurau, G.3
-
57
-
-
0038697355
-
From curiosities to commodities: Ionic liquids begin the transition
-
Davis JH, Fox PA. From curiosities to commodities: Ionic liquids begin the transition. Chem Commun 2003;1209-12
-
(2003)
Chem Commun
, pp. 1209-1212
-
-
Davis, J.H.1
Fox, P.A.2
-
58
-
-
33645460351
-
Fluorine-free and hydrophobic room-temperature ionic liquids, tetraalkylammonium bis(2-ethylhexyl) sulfosuccinates, and their ionic liquid-water two-phase properties
-
Nishi N, Kawakami T, Shigematsu F, et al. Fluorine-free and hydrophobic room-temperature ionic liquids, tetraalkylammonium bis(2-ethylhexyl) sulfosuccinates, and their ionic liquid-water two-phase properties. Green Chem 2006;8:349-55
-
(2006)
Green Chem
, vol.8
, pp. 349-355
-
-
Nishi, N.1
Kawakami, T.2
Shigematsu, F.3
-
59
-
-
21844432372
-
Room temperature ionic liquids as novel media for clean liquid-liquid extraction
-
Huddleston JG, Willauer HD, Swatloski RP, et al. Room temperature ionic liquids as novel media for "clean" liquid-liquid extraction. Chem Commun 1998;1765-6
-
(1998)
Chem Commun
, pp. 1765-1766
-
-
Huddleston, J.G.1
Willauer, H.D.2
Swatloski, R.P.3
-
60
-
-
41349092480
-
Room temperature ionic liquids and their mixtures: Potential pharmaceutical solvents
-
Mizuuchi H, Jaitely V, Murdan S, et al. Room temperature ionic liquids and their mixtures: Potential pharmaceutical solvents. Eur J Pharm Sci 2008;33:326-31
-
(2008)
Eur J Pharm Sci
, vol.33
, pp. 326-331
-
-
Mizuuchi, H.1
Jaitely, V.2
Murdan, S.3
-
61
-
-
40849106246
-
Water-immiscible room temperature ionic liquids (RTILs) as drug reservoirs for controlled release
-
Jaitely V, Karatas A, Florence AT. Water-immiscible room temperature ionic liquids (RTILs) as drug reservoirs for controlled release. Int J Pharm 2008;354:168-73
-
(2008)
Int J Pharm
, vol.354
, pp. 168-173
-
-
Jaitely, V.1
Karatas, A.2
Florence, A.T.3
-
62
-
-
84884544247
-
Drug specific, tuning of an ionic liquid's hydrophilic-lipophilic balance to improve water solubility of poorly soluble active pharmaceutical ingredients
-
DOI: 10.1039/C3NJ00454F
-
McCrary PD, Beasley PA, Gurau G, et al. Drug specific, tuning of an ionic liquid's hydrophilic-lipophilic balance to improve water solubility of poorly soluble active pharmaceutical ingredients. New J Chem 2013;DOI: 10.1039/C3NJ00454F
-
(2013)
New J Chem
-
-
McCrary, P.D.1
Beasley, P.A.2
Gurau, G.3
-
63
-
-
39049138900
-
Microemulsions: Applications in transdermal and dermal delivery
-
Date AA, Patravale VB. Microemulsions: Applications in transdermal and dermal delivery. Crit Rev Ther Drug Carrier Syst 2007;24:547-96
-
(2007)
Crit Rev Ther Drug Carrier Syst
, vol.24
, pp. 547-596
-
-
Date, A.A.1
Patravale, V.B.2
-
64
-
-
38349172495
-
Biocompatible microemulsions and their prospective uses in drug delivery
-
Gupta S, Moulik SP. Biocompatible microemulsions and their prospective uses in drug delivery. J Pharm Sci 2008;97:22-45
-
(2008)
J Pharm Sci
, vol.97
, pp. 22-45
-
-
Gupta, S.1
Moulik, S.P.2
-
65
-
-
19744365835
-
Ionic liquid-in-oil microemulsions
-
Eastoe J, Gold S, Rogers SE, et al. Ionic liquid-in-oil microemulsions. J Am Chem Soc 2005;127:7302-3
-
(2005)
J Am Chem Soc
, vol.127
, pp. 7302-7303
-
-
Eastoe, J.1
Gold, S.2
Rogers, S.E.3
-
66
-
-
76949096875
-
Ionic liquid-assisted transdermal delivery of sparingly soluble drugs
-
Moniruzzaman M, Tahara Y, Tamura M, et al. Ionic liquid-assisted transdermal delivery of sparingly soluble drugs. Chem Commun 2010;46:1452-4
-
(2010)
Chem Commun
, vol.46
, pp. 1452-1454
-
-
Moniruzzaman, M.1
Tahara, Y.2
Tamura, M.3
-
67
-
-
77957683026
-
Ionic liquid-in-oil microemulsion as a potential carrier of sparingly soluble drug: Characterization and cytotoxicity evaluation
-
Moniruzzaman M, Tamura M, Tahara Y, et al. Ionic liquid-in-oil microemulsion as a potential carrier of sparingly soluble drug: Characterization and cytotoxicity evaluation. Int J Pharm 2010;400:243-50
-
(2010)
Int J Pharm
, vol.400
, pp. 243-250
-
-
Moniruzzaman, M.1
Tamura, M.2
Tahara, Y.3
-
68
-
-
77956916377
-
Ionic liquid based microemulsion with pharmaceutically accepted components: Formulation and potential applications
-
Moniruzzaman M, Kamiya N, Goto M. Ionic liquid based microemulsion with pharmaceutically accepted components: Formulation and potential applications. J Colloid Interface Sci 2010;352:136-42
-
(2010)
J Colloid Interface Sci
, vol.352
, pp. 136-142
-
-
Moniruzzaman, M.1
Kamiya, N.2
Goto, M.3
-
69
-
-
79960279737
-
Unique role of ionic liquid [bmim][BF4] during curcumin-surfactant association and micellization of cationic, anionic and non-ionic surfactant solutions
-
Patra D, Barakat C. Unique role of ionic liquid [bmim][BF4] during curcumin-surfactant association and micellization of cationic, anionic and non-ionic surfactant solutions. Spectrochim Acta A 2011;79:1823-8
-
(2011)
Spectrochim Acta A
, vol.79
, pp. 1823-1828
-
-
Patra, D.1
Barakat, C.2
-
70
-
-
84858302159
-
An understanding of the modulation of photophysical properties of curcumin inside a micelle formed by an ionic liquid: A new possibility of tunable drug delivery system
-
Ghatak C, Rao VG, Mandal S, et al. An understanding of the modulation of photophysical properties of curcumin inside a micelle formed by an ionic liquid: A new possibility of tunable drug delivery system. J Phys Chem B 2012;116:3369-79
-
(2012)
J Phys Chem B
, vol.116
, pp. 3369-3379
-
-
Ghatak, C.1
Rao, V.G.2
Mandal, S.3
-
71
-
-
84871270302
-
An investigation of drug binding ability of a surface active ionic liquid: Micellization, electrochemical, and spectroscopic studies
-
Mahajan S, Sharma R, Mahajan RK. An investigation of drug binding ability of a surface active ionic liquid: Micellization, electrochemical, and spectroscopic studies. Langmuir 2012;28:17238-46
-
(2012)
Langmuir
, vol.28
, pp. 17238-17246
-
-
Mahajan, S.1
Sharma, R.2
Mahajan, R.K.3
-
72
-
-
34248356918
-
Why products fail in phase III
-
Gordian M, Singh N, Zemmel R, et al. Why products fail in phase III. In Vivo 2006;4:49-54
-
(2006)
Vivo
, vol.4
, pp. 49-54
-
-
Gordian, M.1
Singh, N.2
Zemmel, R.3
-
73
-
-
84859237601
-
An emerging technique for poorly soluble drugs: Self-emulsifying drug delivery system
-
Patel ND. An emerging technique for poorly soluble drugs: Self-emulsifying drug delivery system. Int J Pharm Biol Arch 2011;2:621-9
-
(2011)
Int J Pharm Biol Arch
, vol.2
, pp. 621-629
-
-
Patel, N.D.1
-
75
-
-
0030795298
-
Liposomes in drug delivery: Progress and limitations
-
Sharma A, Sharma US. Liposomes in drug delivery: Progress and limitations. Int J Pharm 1997;154:123-40
-
(1997)
Int J Pharm
, vol.154
, pp. 123-140
-
-
Sharma, A.1
Sharma, U.S.2
-
76
-
-
2342481809
-
Lessons learned from marketed and investigational prodrugs
-
Ettmayer P, Amidon GL, Clement B, et al. Lessons learned from marketed and investigational prodrugs. J Med Chem 2004;47:2393-404
-
(2004)
J Med Chem
, vol.47
, pp. 2393-2404
-
-
Ettmayer, P.1
Amidon, G.L.2
Clement, B.3
-
77
-
-
78049512700
-
Some thoughts and current issues
-
Stella VJ. Some thoughts and current issues. J Pharm Sci 2010;99:4755-65
-
(2010)
J Pharm Sci
, vol.99
, pp. 4755-4765
-
-
Stella, V.J.1
-
78
-
-
34548032742
-
Salt formation to improve drug solubility
-
Serajuddin ATM. Salt formation to improve drug solubility. Adv Drug Deliv Rev 2007;59:603-16
-
(2007)
Adv Drug Deliv Rev
, vol.59
, pp. 603-616
-
-
Serajuddin, A.T.M.1
-
79
-
-
27744484364
-
Saccharin salts of active pharmaceutical ingredients, their crystal structures, and increased water solubilities
-
Banerjee R, Bhatt PM, Ravindra NV, et al. Saccharin salts of active pharmaceutical ingredients, their crystal structures, and increased water solubilities. Cryst Growth Des 2005;5:2299-309
-
(2005)
Cryst Growth Des
, vol.5
, pp. 2299-2309
-
-
Banerjee, R.1
Bhatt, P.M.2
Ravindra, N.V.3
-
80
-
-
80052695630
-
Strategies for solubility enhancement of poorly soluble drugs
-
Patil SK, Wagh KS, Parik VB, et al. Strategies for solubility enhancement of poorly soluble drugs. Int J Pharm Sci Rev Res 2011;8:74-80
-
(2011)
Int J Pharm Sci Rev Res
, vol.8
, pp. 74-80
-
-
Patil, S.K.1
Wagh, K.S.2
Parik, V.B.3
-
81
-
-
0038713880
-
Crystal engineering of novel cocrystals of a triazole drug with 1,4-dicarboxylic acids
-
Remenar JF, Morissette SL, Peterson ML, et al. Crystal engineering of novel cocrystals of a triazole drug with 1,4-dicarboxylic acids. J Am Chem Soc 2003;125:8456-7
-
(2003)
J Am Chem Soc
, vol.125
, pp. 8456-8457
-
-
Remenar, J.F.1
Morissette, S.L.2
Peterson, M.L.3
-
82
-
-
6044264984
-
Crystal engineering approach to forming cocrystals of amine hydrochloride with organic acids
-
Childs SL, Chall LJ, Dunlap JT, et al. Crystal engineering approach to forming cocrystals of amine hydrochloride with organic acids. J Am Chem Soc 2004;126:13335-42
-
(2004)
J Am Chem Soc
, vol.126
, pp. 13335-13342
-
-
Childs, S.L.1
Chall, L.J.2
Dunlap, J.T.3
-
83
-
-
19944371772
-
Pharmaceutical cocrystallization: Engineering a remedy for caffeine hydration
-
Trask AV, Motherwell WDS, Jones W. Pharmaceutical cocrystallization: Engineering a remedy for caffeine hydration. Cryst Growth Des 2005;5:1013-21
-
(2005)
Cryst Growth Des
, vol.5
, pp. 1013-1021
-
-
Trask, A.V.1
Motherwell, W.D.S.2
Jones, W.3
-
84
-
-
84863691005
-
Pharmaceutical cocrystals of nitrofurantoin: Screening, characterization and crystal structure analysis
-
Alhalaweh A, George S, Basavoju S, et al. Pharmaceutical cocrystals of nitrofurantoin: Screening, characterization and crystal structure analysis. CrystEngComm 2012;14:5078-88
-
(2012)
Cryst Eng Comm
, vol.14
, pp. 5078-5088
-
-
Alhalaweh, A.1
George, S.2
Basavoju, S.3
-
85
-
-
0034601240
-
Improving drug solubility for oral delivery using solid dispersions
-
Leuner C, Dressman J. Improving drug solubility for oral delivery using solid dispersions. Eur J Pharm Biopharm 2000;50:47-60
-
(2000)
Eur J Pharm Biopharm
, vol.50
, pp. 47-60
-
-
Leuner, C.1
Dressman, J.2
-
86
-
-
80054870067
-
Review on various techniques of solubility enhancement of poorly soluble drugs with special emphasis on solid dispersion
-
Singh MC, Sayyad AB, Sawant SD. Review on various techniques of solubility enhancement of poorly soluble drugs with special emphasis on solid dispersion. J Pharm Res 2010;3:2494-501
-
(2010)
J Pharm Res
, vol.3
, pp. 2494-2501
-
-
Singh, M.C.1
Sayyad, A.B.2
Sawant, S.D.3
-
87
-
-
0141732214
-
Interfacial solubilization of model amphiphilic molecules in block copolymer micelles
-
Choucair A, Eisenburg A. Interfacial solubilization of model amphiphilic molecules in block copolymer micelles. J Am Chem Soc 2003;125:11993-2000
-
(2003)
J Am Chem Soc
, vol.125
, pp. 11993-12000
-
-
Choucair, A.1
Eisenburg, A.2
-
88
-
-
57649240283
-
Formation direct, atom efficient, and halide free syntheses of azolium azolate energetic ionic liquids and their eutectic mixtures, and method for determining eutectic composition
-
Smiglak M, Bridges NJ, Dilip M, et al. Formation direct, atom efficient, and halide free syntheses of azolium azolate energetic ionic liquids and their eutectic mixtures, and method for determining eutectic composition. Chem Eur J 2008;14:11314-19
-
(2008)
Chem Eur J
, vol.14
, pp. 11314-11319
-
-
Smiglak, M.1
Bridges, N.J.2
Dilip, M.3
-
89
-
-
37349014528
-
The second evolution of ionic liquids: From solvents and separations to advanced materials-energetic examples from the ionic liquid cookbook
-
Smiglak M, Metlen A, Rogers RD. The second evolution of ionic liquids: From solvents and separations to advanced materials-energetic examples from the ionic liquid cookbook. Acc Chem Res 2007;40:1182-92
-
(2007)
Acc Chem Res
, vol.40
, pp. 1182-1192
-
-
Smiglak, M.1
Metlen, A.2
Rogers, R.D.3
-
92
-
-
77955982363
-
Efficacy and safety of etodolac-paracetamol fixed dose combination in patients with knee osteoarthritis flare-up: A randomized, double-blind comparative evaluation
-
Pareek AMD, Chandurkar N, Ambade R, et al. Efficacy and safety of etodolac-paracetamol fixed dose combination in patients with knee osteoarthritis flare-up: A randomized, double-blind comparative evaluation. Clin J Pain 2010;26:561-6
-
(2010)
Clin J Pain
, vol.26
, pp. 561-566
-
-
Pareek, A.M.D.1
Chandurkar, N.2
Ambade, R.3
-
93
-
-
0038681648
-
Double blind randomized comparative trial of etodolac SR versus diclofenac in the treatment of osteoarthritis of the knee
-
Liang TH, Hsu PN. Double blind randomized comparative trial of etodolac SR versus diclofenac in the treatment of osteoarthritis of the knee. Curr Med Res Opin 2003;19:336-41
-
(2003)
Curr Med Res Opin
, vol.19
, pp. 336-341
-
-
Liang, T.H.1
Hsu, P.N.2
-
94
-
-
0026665170
-
Safety and efficacy of etodolac compared with piroxicam in patients with degenerative joint disease of the knee
-
Dick WC, Bulstra S, Schardijin GH, et al. Safety and efficacy of etodolac compared with piroxicam in patients with degenerative joint disease of the knee. Clin Ther 1992;14:517-26
-
(1992)
Clin Ther
, vol.14
, pp. 517-526
-
-
Dick, W.C.1
Bulstra, S.2
Schardijin, G.H.3
-
95
-
-
0028198634
-
A comparative study of efficacy and toxicity of etodolac and naproxen in the treatment of osteoarthritis
-
Chikanza IC, Clarke B, Hopkins R, et al. A comparative study of efficacy and toxicity of etodolac and naproxen in the treatment of osteoarthritis. Br J Clin Pract 1994;48:67-9
-
(1994)
Br J Clin Pract
, vol.48
, pp. 67-69
-
-
Chikanza, I.C.1
Clarke, B.2
Hopkins, R.3
-
97
-
-
84884569035
-
-
Available From [Last accessed 17 May 13]
-
MEDRx news release. Available from: Http://www.medrx.co.jp/english/ newsrelease.html [Last accessed 17 May 13]
-
MEDRx News Release
-
-
-
98
-
-
0348110657
-
Ionic liquids by proton transfer: Vapor pressure, conductivity, and the relevance of DeltapKa from aqueous solutions
-
Yoshizawa M, Xu W, Angell CA. Ionic liquids by proton transfer: Vapor pressure, conductivity, and the relevance of DeltapKa from aqueous solutions. J Am Chem Soc 2003;125:15411-19
-
(2003)
J Am Chem Soc
, vol.125
, pp. 15411-15419
-
-
Yoshizawa, M.1
Xu, W.2
Angell, C.A.3
-
99
-
-
84884557653
-
-
Fehrmann R, Haumann M, Riisager A, editor. Book chapter in supported ionic liquids -fundamentals and applications, Wiley. VCH, ISBN-13 978 3527324293 Weinheim, Germany in press
-
Cojocaru OA, Siriwardana A, Gurau G, et al. Pharmaceutically active supported ionic liquid phases. In: Fehrmann R, Haumann M, Riisager A, editor. Book chapter in supported ionic liquids -fundamentals and applications, Wiley-VCH, ISBN-13: 978-3527324293; Weinheim, Germany: 2013, in press.
-
(2013)
Pharmaceutically Active Supported Ionic Liquid Phases
-
-
Cojocaru, O.A.1
Siriwardana, A.2
Gurau, G.3
-
101
-
-
84884548675
-
Biologically active compounds supported on solid carrier such as silica for controlled release and improved thermal stability
-
2011110662
-
Riisager A, Fehrmann R, Rodriguez R, et al. Biologically active compounds supported on solid carrier such as silica for controlled release and improved thermal stability. PCT Int. Appl. WO 2011110662; 2011
-
(2011)
PCT Int. Appl. WO
-
-
Riisager, A.1
Fehrmann, R.2
Rodriguez, R.3
-
102
-
-
84861626939
-
Pharmaceutically active ionic liquids with solids handling, enhanced thermal stability, and fast release
-
Bica K, Rodríguez H, Gurau G, et al. Pharmaceutically active ionic liquids with solids handling, enhanced thermal stability, and fast release. Chem Commun 2012;48:5422-4
-
(2012)
Chem Commun
, vol.48
, pp. 5422-5424
-
-
Bica, K.1
Rodríguez, H.2
Gurau, G.3
|