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Archiv der Pharmazie

Volumn 346, Issue 5, 2013, Pages 339-348

New arylpiperazines with flexible versus partly constrained linker as serotonin 5-HT1A/5-HT7 receptor ligands

(5) Kowalski, Piotr a Mitka, Katarzyna a Jaśkowska, Jolanta a Duszyńska, Beata b Bojarski, Andrzej J b

a CRACOW UNIVERSITY OF TECHNOLOGY (Poland)

b INSTITUTE OF PHARMACOLOGY (Poland)

Author keywords

Arylpiperazines; NAN 190; Serotonin 5 HT1A 5 HT7 receptor ligands; Structure activity relationship (SAR)

Indexed keywords

1 (2 METHOXYPHENYL) 4 (4 PHTHALIMIDOBUTYL)PIPERAZINE; 3 [(1,2,3,4 TETRAHYDROISOQUINOLIN 2 YL)METHYL]TOLUENE; 3 [[4 (2 METHOXYPHENYL)PIPERAZIN 1 YL]METHYL]TOLUENE; 4 [(1,2,3,4 TETRAHYDROISOQUINOLIN 2 YL)METHYL]TOLUENE; 4 [[4 (2 METHOXYPHENYL)PIPERAZIN 1 YL]METHYL]TOLUENE; ARYLPIPERAZINE DERIVATIVE; N [3 (1,2,3,4 TETRAHYDROISOQUINOLIN 2 YL)BENZYL]PHTHALIMIDE; N [3 [(1,2,3,4 TETRAHYDROISOQUINOLIN 2 YL)METHYL]BENZYL]PHTHALIMIDE; N [3 [[4 (2 METHOXYPHENYL)PIPERAZIN 1YL]BENZYL] 2H 1,3 BENZOXAZINE 2,4 (3H) DIONE; N [3 [[4 (2 METHOXYPHENYL)PIPERAZIN 1YL]METHYL]BENZYL]PHTHALIMIDE; N [4 (1,2,3,4 TETRAHYDROISOQUINOLIN 2 YL)PENTYL]2H 1,3 BENZOXAZINE 2,4(3H)DIONE; N [4 [(1,2,3,4 TETRAHYDROISOQUINOLIN 2 YL)METHYL]BENZYL]PHTHALIMIDE; N [4 [[4 (2 METHOXYPHENYL)PIPERAZIN 1YL]BENZYL] 2H 1,3 BENZOXAZINE 2,4 (3H) DIONE; N [4 [[4 (2 METHOXYPHENYL)PIPERAZIN 1YL]METHYL]BENZYL]PHTHALIMIDE; N [5 (1,2,3,4 TETRAHYDROISOQUINOLIN 2 YL)PENTYL]2H 1,3 BENZOXAZINE 2,4(3H)DIONE; N [5 (1,2,3,4 TETRAHYDROISOQUINOLIN 2 YL)PENTYL]PHTHALIMIDE; N [5 [4 (2 METHOXYPHENYL)PIPERAZIN 1YL]PENTYL]PHTHALIMIDE; N [5 [[4 (2 METHOXYPHENYL)PIPERAZIN 1YL]PENTYL] 2H 1,3 BENZOXAZINE 2,4 (3H) DIONE; N [6 (1,2,3,4 TETRAHYDROISOQUINOLIN 2 YL)HEXYL] 2H 1,3 BENZOXAZINE 2,4 (3H)DIONE; N [6 (1,2,3,4 TETRAHYDROISOQUINOLIN 2 YL)HEXYL]PHTHALIMIDE; N [6 [4 (2 METHOXYPHENYL)PIPERAZIN 1YL]HEXYL]PHTHALIMIDE; N [6 [[4 (2 METHOXYPHENYL)PIPERAZIN 1YL]HEXYL] 2H 1,3 BENZOXAZINE 2,4 (3H) DIONE; PIPERAZINE DERIVATIVE; SEROTONIN 1A RECEPTOR; SEROTONIN 7 RECEPTOR; SEROTONIN RECEPTOR AFFECTING AGENT; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; DRUG BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; HUMAN CELL; IN VITRO STUDY; PRIORITY JOURNAL; RADIOACTIVITY; STRUCTURE ACTIVITY RELATION;

ANIMALS; HUMANS; LIGANDS; PIPERAZINES; RATS; RECEPTOR, SEROTONIN, 5-HT1A; RECEPTORS, SEROTONIN; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84877769113 PISSN: 03656233 EISSN: 15214184 Source Type: Journal
DOI: 10.1002/ardp.201300011 Document Type: Article

Times cited : (24)

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