SCOPUS 정보 검색 플랫폼

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 23, 2004, Pages 5863-5866

The impact of spacer structure on 5-HT 7 and 5-HT 1A receptor affinity in the group of long-chain arylpiperazine ligands

(5) Bojarski, Andrzej J a Duszyńska, Beata a Kołaczkowski, Marcin b Kowalski, Piotr c Kowalska, Teresa c

a INSTITUTE OF PHARMACOLOGY (Poland)

b JAGIELLONIAN UNIVERSITY MEDICAL COLLEGE (Poland)

c CRACOW UNIVERSITY OF TECHNOLOGY (Poland)

Author keywords

5 HT 7 receptor ligands; Conformational constraints; Long chain arylpiperazines

Indexed keywords

1 (2 METHOXYPHENYL) 4 (4 PHTHALIMIDOBUTYL)PIPERAZINE; 1 (2 METHOXYPHENYL) 4 (4 SUCCINIMIDOBUTYL)PIPERAZINE; PIPERAZINE DERIVATIVE; SEROTONIN 1 ANTAGONIST; SEROTONIN 1A RECEPTOR; SEROTONIN 7 RECEPTOR; UNCLASSIFIED DRUG;

ARTICLE; CIS TRANS ISOMERISM; CONFORMATION; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; STRUCTURE ANALYSIS;

LIGANDS; MOLECULAR CONFORMATION; PIPERAZINES; PROTEIN BINDING; RECEPTOR, SEROTONIN, 5-HT1A; RECEPTORS, SEROTONIN;

EID: 7044222890 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2004.09.029 Document Type: Article

Times cited : (33)

References (20)

1
- 0027421620
- J.A. Bard, J. Zgombick, N. Adham, P. Vaysse, T.A. Branchek, and R.L. Weinshank J. Biol. Chem. 268 1993 23422
- (1993) J. Biol. Chem. , vol.268 , pp. 23422
- Bard, J.A.¹ Zgombick, J.² Adham, N.³ Vaysse, P.⁴ Branchek, T.A.⁵ Weinshank, R.L.⁶

2
- 0027368668
- T.W. Lovenberg, B.M. Baron, L. de Lecea, J.D. Miller, R.A. Prosser, M.A. Rea, P.E. Foye, M. Racke, A.L. Slone, B.W. Siegel, P.E. Danielson, J.G. Sutcliffe, and M.G. Erlander Neuron 11 1993 449
- (1993) Neuron , vol.11 , pp. 449
- Lovenberg, T.W.¹ Baron, B.M.² De Lecea, L.³ Miller, J.D.⁴ Prosser, R.A.⁵ Rea, M.A.⁶ Foye, P.E.⁷ Racke, M.⁸ Slone, A.L.⁹ Siegel, B.W.¹⁰ Danielson, P.E.¹¹ Sutcliffe, J.G.¹² Erlander, M.G.¹³

3
- 0028168584
- A.P. Tsou, A. Kosaka, C. Bach, P. Zuppan, C. Yee, L. Tom, R. Alvarez, S. Ramsey, D.W. Bonhaus, E. Stefanich, L. Jakeman, R.M. Eglen, and H. Chan J. Neurochem. 63 1994 456
- (1994) J. Neurochem. , vol.63 , pp. 456
- Tsou, A.P.¹ Kosaka, A.² Bach, C.³ Zuppan, P.⁴ Yee, C.⁵ Tom, L.⁶ Alvarez, R.⁷ Ramsey, S.⁸ Bonhaus, D.W.⁹ Stefanich, E.¹⁰ Jakeman, L.¹¹ Eglen, R.M.¹² Chan, H.¹³

4
- 0034628555
- P.J. Lovell, S.M. Bromidge, S. Dabbs, D.M. Duckworth, I.T. Forbes, A.J. Jennings, F.D. King, D.N. Middlemiss, S.K. Rahman, D.V. Saunders, L.L. Collin, J.J. Hagan, G.J. Riley, and D.R. Thomas J. Med. Chem. 43 2000 342
- (2000) J. Med. Chem. , vol.43 , pp. 342
- Lovell, P.J.¹ Bromidge, S.M.² Dabbs, S.³ Duckworth, D.M.⁴ Forbes, I.T.⁵ Jennings, A.J.⁶ King, F.D.⁷ Middlemiss, D.N.⁸ Rahman, S.K.⁹ Saunders, D.V.¹⁰ Collin, L.L.¹¹ Hagan, J.J.¹² Riley, G.J.¹³ Thomas, D.R.¹⁴

5
- 18644367263
- I.T. Forbes, S. Douglas, A.D. Gribble, R.J. Ife, A.P. Lightfoot, A.E. Garner, G.J. Riley, P. Jeffrey, A.J. Stevens, T.O. Stean, and D.R. Thomas Bioorg. Med. Chem. Lett. 12 2002 3341
- (2002) Bioorg. Med. Chem. Lett. , vol.12 , pp. 3341
- Forbes, I.T.¹ Douglas, S.² Gribble, A.D.³ Ife, R.J.⁴ Lightfoot, A.P.⁵ Garner, A.E.⁶ Riley, G.J.⁷ Jeffrey, P.⁸ Stevens, A.J.⁹ Stean, T.O.¹⁰ Thomas, D.R.¹¹

6
- 1642374924
- M. Leopoldo Curr. Med. Chem. 11 2004 629
- (2004) Curr. Med. Chem. , vol.11 , pp. 629
- Leopoldo, M.¹

7
- 3042841937
- D.R. Thomas, and J.J. Hagan Curr. Drug Targets CNS Neurol. Disord. 3 2004 81
- (2004) Curr. Drug Targets CNS Neurol. Disord. , vol.3 , pp. 81
- Thomas, D.R.¹ Hagan, J.J.²

8
- 10744229658
- M.L. Lopez-Rodriguez, E. Porras, M.J. Morcillo, B. Benhamu, L.J. Soto, J.L. Lavandera, J.A. Ramos, M. Olivella, M. Campillo, and L. Pardo J. Med. Chem. 46 2003 5638
- (2003) J. Med. Chem. , vol.46 , pp. 5638
- Lopez-Rodriguez, M.L.¹ Porras, E.² Morcillo, M.J.³ Benhamu, B.⁴ Soto, L.J.⁵ Lavandera, J.L.⁶ Ramos, J.A.⁷ Olivella, M.⁸ Campillo, M.⁹ Pardo, L.¹⁰

9
- 0037434593
- R. Perrone, F. Berardi, N.A. Colabufo, E. Lacivita, M. Leopoldo, and V. Tortorella J. Med. Chem. 46 2003 646
- (2003) J. Med. Chem. , vol.46 , pp. 646
- Perrone, R.¹ Berardi, F.² Colabufo, N.A.³ Lacivita, E.⁴ Leopoldo, M.⁵ Tortorella, V.⁶

10
- 0035570104
- R.E. Wilcox, J.E. Ragan, R.S. Pearlman, M.Y. Brusniak, R.M. Eglen, D.W. Bonhaus, T.E. Tenner Jr., and J.D. Miller J. Comput. Aided Mol. Des. 15 2001 883
- (2001) J. Comput. Aided Mol. Des. , vol.15 , pp. 883
- Wilcox, R.E.¹ Ragan, J.E.² Pearlman, R.S.³ Brusniak, M.Y.⁴ Eglen, R.M.⁵ Bonhaus, D.W.⁶ Tenner Jr., T.E.⁷ Miller, J.D.⁸

11
- 0000209627
- M.J. Mokrosz, E. Chojnacka-Wójcik, E. Tatarczyñska, A. Kłodziñ ska, M. Filip, J. Boksa, S. Charakchieva-Minol, and J.L. Mokrosz Med. Chem. Res. 4 1994 161
- (1994) Med. Chem. Res. , vol.4 , pp. 161
- Mokrosz, M.J.¹ Chojnacka-Wójcik, E.² Tatarczyñska, E.³ Kłodziñ Ska, A.⁴ Filip, M.⁵ Boksa, J.⁶ Charakchieva-Minol, S.⁷ Mokrosz, J.L.⁸

12
- 0023793228
- R.A. Glennon, N.A. Naiman, M.E. Pierson, M. Titeler, R.A. Lyon, and E. Weisberg Eur. J. Pharmacol. 154 1988 339
- (1988) Eur. J. Pharmacol. , vol.154 , pp. 339
- Glennon, R.A.¹ Naiman, N.A.² Pierson, M.E.³ Titeler, M.⁴ Lyon, R.A.⁵ Weisberg, E.⁶

13
- 0037023530
- M.H. Paluchowska, A.J. Bojarski, S. Charakchieva-Minol, and A. Wesołowska Eur. J. Med. Chem. 37 2002 273
- (2002) Eur. J. Med. Chem. , vol.37 , pp. 273
- Paluchowska, M.H.¹ Bojarski, A.J.² Charakchieva-Minol, S.³ Wesołowska, A.⁴

14
- 0033518263
- M.H. Paluchowska, M.J. Mokrosz, A.J. Bojarski, A. Wesołowska, J. Borycz, S. Charakchieva-Minol, and E. Chojnacka-Wójcik J. Med. Chem. 42 1999 4952
- (1999) J. Med. Chem. , vol.42 , pp. 4952
- Paluchowska, M.H.¹ Mokrosz, M.J.² Bojarski, A.J.³ Wesołowska, A.⁴ Borycz, J.⁵ Charakchieva-Minol, S.⁶ Chojnacka-Wójcik, E.⁷

15
- 0032502639
- N. Aguirre, S. Ballaz, B. Lasheras, and J. Del Rio Eur. J. Pharmacol. 346 1998 181
- (1998) Eur. J. Pharmacol. , vol.346 , pp. 181
- Aguirre, N.¹ Ballaz, S.² Lasheras, B.³ Del Rio, J.⁴

16
- 0027211828
- A.J. Bojarski, M.T. Cegła, S. Charakchieva-Minol, M.J. Mokrosz, M. Maćkowiak, and J.L. Mokrosz Pharmazie 48 1993 289
- (1993) Pharmazie , vol.48 , pp. 289
- Bojarski, A.J.¹ Cegła, M.T.² Charakchieva-Minol, S.³ Mokrosz, M.J.⁴ MaćKowiak, M.⁵ Mokrosz, J.L.⁶

17
- 0030043026
- M.H. Norman, D.J. Minick, and G.C. Rigdon J. Med. Chem. 39 1996 149
- (1996) J. Med. Chem. , vol.39 , pp. 149
- Norman, M.H.¹ Minick, D.J.² Rigdon, G.C.³

18
- 0038316776
- M.L. Lopez-Rodriguez, M.J. Morcillo, T.K. Rovat, E. Fernandez, B. Vicente, A.M. Sanz, M. Hernandez, and L. Orensanz J. Med. Chem. 42 1999 36
- (1999) J. Med. Chem. , vol.42 , pp. 36
- Lopez-Rodriguez, M.L.¹ Morcillo, M.J.² Rovat, T.K.³ Fernandez, E.⁴ Vicente, B.⁵ Sanz, A.M.⁶ Hernandez, M.⁷ Orensanz, L.⁸

19
- 0035818892
- R. Perrone, F. Berardi, N.A. Colabufo, M. Leopoldo, E. Lacivita, V. Tortorella, A. Leonardi, E. Poggesi, and R. Testa J. Med. Chem. 44 2001 4431
- (2001) J. Med. Chem. , vol.44 , pp. 4431
- Perrone, R.¹ Berardi, F.² Colabufo, N.A.³ Leopoldo, M.⁴ Lacivita, E.⁵ Tortorella, V.⁶ Leonardi, A.⁷ Poggesi, E.⁸ Testa, R.⁹

20
- 84961980743
- A. Klamt, and G. Schüürmann J. Chem. Soc., Perkin Trans. 2 1993 799
- (1993) J. Chem. Soc., Perkin Trans. 2 , pp. 799
- Klamt, A.¹ Schüürmann, G.²

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.